Target Details
| UniProt AC | P33981 |
|---|---|
| Gene Symbol | TTK |
| Protein Name | Dual specificity protein kinase TTK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 178
- Clinical molecules 17
- Avg pChEMBL 7.57
KEGG Pathways (1)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JCICCACMYITOCI
|
6.4 | IC50 | 3 | — | |
LOQIJPHCNFJJTO
|
6.4 | IC50 | 2 | — | |
SERJTVXHERVFCQ
|
6.4 | IC50 | 2 | — | |
WGZHCNCLATVGMN
|
6.4 | IC50 | 2 | — | |
WMVFYJNFGFTSCQ
|
6.4 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
6.4 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
6.4 | Kd | 149 | — | |
LXGHIBLIRSFIIW
|
6.4 | IC50 | 2 | — | |
JOOXLOJCABQBSG
|
6.3 | Kd | 139 | — | |
NAGOZOOVQLAGAY
|
6.3 | IC50 | 2 | — | |
HFNKQEVNSGCOJV
|
6.3 | Kd | 65 | — | |
FAPBUMXELNHUHE
|
6.3 | IC50 | 2 | — | |
PCTWMWBDQSWVBE
|
6.3 | IC50 | 2 | — | |
UTHWBIPHRYUJSU
|
6.3 | IC50 | 11 | Yes | |
LHQIHZSYSNEJIN
|
6.3 | IC50 | 2 | — | |
LTQRUCOWRVPXHK
|
6.2 | IC50 | 2 | — | |
PSFMCOGQKUBLKM
|
6.2 | IC50 | 3 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes | |
MUSBPXCQBAUPOW
|
6.2 | IC50 | 2 | — | |
ZJVKSKNRXMNPQJ
|
6.2 | IC50 | 2 | — | |
XGWVDWGXBYRXIX
|
6.1 | IC50 | 2 | — | |
XHEYSFJJPSXTHP
|
6.1 | IC50 | 3 | — | |
FRANNCVVJFQWOT
|
6.1 | IC50 | 3 | — | |
WUDDKNUPJTYVAB
|
6.0 | IC50 | 2 | — | |
ATUUNJCZCOMUKD
|
6.0 | IC50 | 7 | — | |
SKLZRGKNDWBPBV
|
6.0 | IC50 | 2 | — | |
UJBJWYNPUOLFIZ
|
6.0 | IC50 | 49 | — | |
YDMGJNNVRFAERS
|
6.0 | IC50 | 2 | — |