Target Details
| UniProt AC | P33981 |
|---|---|
| Gene Symbol | TTK |
| Protein Name | Dual specificity protein kinase TTK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 178
- Clinical molecules 17
- Avg pChEMBL 7.57
KEGG Pathways (1)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KOZFSFOOLUUIGY
|
7.5 | Kd | 88 | Yes | |
RIZAQRVECMBTPF
|
7.5 | IC50 | 2 | — | |
ATKPMPVOTNGCIB
|
7.5 | IC50 | 2 | — | |
GUBJNPWVIUFSTR
|
7.5 | Kd | 103 | — | |
ZWRLLBAFCKACAL
|
7.4 | IC50 | 3 | Yes | |
MFVOIPKDSOFMQO
|
7.4 | IC50 | 3 | — | |
MFVOIPKDSOFMQO
|
7.4 | IC50 | 3 | — | |
UGXCBYVBIJACEK
|
7.3 | IC50 | 8 | — | |
QQWUGDVOUVUTOY
|
7.3 | Kd | 231 | Yes | |
SXJKXTZFHYHUNX
|
7.3 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.2 | Kd | 213 | — | |
WINHZLLDWRZWRT
|
7.2 | Kd | 201 | Yes | |
XSLQRBBJXSFSGV
|
7.2 | IC50 | 3 | — | |
PMCMCUYADWVHJI
|
7.2 | IC50 | 3 | — | |
XEMJTISGDXHELX
|
7.2 | IC50 | 8 | Yes | |
LTKUHPWNVCRTSA
|
7.1 | IC50 | 2 | — | |
HZTYDQRUAWIZRE
|
7.1 | Kd | 40 | Yes | |
HKSZLNNOFSGOKW
|
7.1 | Kd | 408 | — | |
RGZXAQQHXALOBL
|
7.1 | Kd | 10 | — | |
WGZYFFJOGZFXBF
|
7.1 | IC50 | 2 | — | |
ACPOUJIDANTYHO
|
7.0 | IC50 | 17 | Yes | |
HJJSEANNATVFNW
|
7.0 | IC50 | 4 | — | |
KRIUNPBAQZGFQA
|
7.0 | Kd | 76 | — | |
CIJWGWNHXQYIJC
|
7.0 | IC50 | 5 | — | |
UBGUCDLLEIGHHP
|
7.0 | IC50 | 6 | — | |
YYLKKYCXAOBSRM
|
7.0 | Kd | 191 | — | |
GELSCYBDXQYAMW
|
6.9 | IC50 | 2 | — | |
NMJMRSQTDLRCRQ
|
6.9 | IC50 | 7 | — | |
DCQJOTPFAGUJNC
|
6.9 | IC50 | 2 | — | |
XDILVFHMVAJWKP
|
6.8 | IC50 | 3 | — | |
ALSJOMXUZWBKMB
|
6.8 | IC50 | 4 | — | |
CUIHSIWYWATEQL
|
6.8 | Kd | 61 | Yes | |
ZPPUMAMZIMPJGP
|
6.8 | Ki | 3 | — | |
CTNPALGJUAXMMC
|
6.7 | Kd | 151 | — | |
UITZSWYAMHHKPO
|
6.7 | IC50 | 4 | — | |
GGWPAZYQWVWDSD
|
6.7 | IC50 | 2 | — | |
KDKUVYLMPJIGKA
|
6.7 | Kd | 91 | Yes | |
UBQLTEZUAMOROQ
|
6.7 | Kd | 2 | — | |
HDAJDNHIBCDLQF
|
6.7 | IC50 | 14 | — | |
ATTXFDBPVDTNAP
|
6.7 | IC50 | 2 | — | |
MTDJJMFQQXOEPJ
|
6.7 | IC50 | 5 | — | |
ODPGGGTTYSGTGO
|
6.6 | Kd | 153 | — | |
OXPLZKSKLWBEIM
|
6.6 | IC50 | 8 | Yes | |
WVXNSAVVKYZVOE
|
6.5 | IC50 | 92 | — | |
KBILTEUAXWLXKP
|
6.5 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.5 | Kd | 91 | Yes | |
JHYPYJLPMJWBRK
|
6.5 | IC50 | 2 | — | |
YIGQSLKUNKHIBI
|
6.5 | IC50 | 2 | — | |
ZBKPGGYJBKTHQF
|
6.4 | IC50 | 2 | — |