Target Details
| UniProt AC | P33981 |
|---|---|
| Gene Symbol | TTK |
| Protein Name | Dual specificity protein kinase TTK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 178
- Clinical molecules 17
- Avg pChEMBL 7.57
KEGG Pathways (1)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SGWLRDAOCLITOM
|
8.2 | IC50 | 7 | — | |
RNRUHOJYKQGQGN
|
8.2 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
OMONHEJVJYRTAT
|
8.2 | IC50 | 3 | — | |
KXMLNXWIFJZEJN
|
8.2 | IC50 | 3 | — | |
URWRFSMVDXZMJH
|
8.2 | IC50 | 3 | — | |
LKZXAQZZOSZHLE
|
8.1 | IC50 | 3 | — | |
WROHCHCGJIWAPG
|
8.1 | IC50 | 3 | — | |
QZZFLPGPIFLIDL
|
8.1 | IC50 | 3 | — | |
FVXILEFBMIKZCO
|
8.1 | IC50 | 3 | — | |
CWJLAVRXVFHDSJ
|
8.1 | IC50 | 13 | — | |
XDEFNAWAKYQBQY
|
8.1 | IC50 | 3 | — | |
DIBCUQSRSKMAFL
|
8.1 | IC50 | 3 | — | |
NBCVGOXDQJIDNF
|
8.1 | IC50 | 3 | — | |
XTJZKALDRPVFSN
|
8.1 | IC50 | 3 | — | |
GXKIHPXGVQZMIN
|
8.0 | IC50 | 3 | — | |
IUWWRSQCDUQDEZ
|
8.0 | IC50 | 8 | — | |
IUWWRSQCDUQDEZ
|
8.0 | IC50 | 9 | — | |
YZTLHDUNASRPOV
|
8.0 | IC50 | 2 | — | |
CQOOBCLBMYGVDE
|
8.0 | IC50 | 3 | — | |
PUJKNBHSGMNWBW
|
8.0 | IC50 | 2 | — | |
XTJZKALDRPVFSN
|
8.0 | IC50 | 5 | — | |
NHAUZBMUXRGRCV
|
7.9 | IC50 | 3 | — | |
OQGWFLXBPGEVIM
|
7.9 | IC50 | 3 | — | |
GBAHUNGQGRGJAX
|
7.8 | IC50 | 3 | — | |
BNSPEWBMGVWZFC
|
7.8 | IC50 | 7 | — | |
IIBNWMLKRSXDKD
|
7.8 | IC50 | 3 | — | |
NKFDCMFJEHBWMX
|
7.8 | IC50 | 2 | — | |
NMJXLTYBAJJXCO
|
7.8 | IC50 | 2 | — | |
VTYQURZUYOUAOK
|
7.8 | IC50 | 3 | — | |
WSTCEYSBWKYEDE
|
7.8 | IC50 | 3 | — | |
COJCXGYVLBGQIH
|
7.7 | IC50 | 2 | — | |
RIOJOTOJNAHBST
|
7.7 | IC50 | 2 | — | |
VDYTVNXJBMDQBM
|
7.7 | IC50 | 3 | — | |
FTZQWKAIKYEWPM
|
7.7 | IC50 | 2 | — | |
QKBGNVCABCTNCY
|
7.7 | IC50 | 3 | — | |
JRZGFHZNTXYGPL
|
7.7 | IC50 | 3 | Yes | |
XSJWROYTYXTZKU
|
7.7 | IC50 | 3 | — | |
ZSURBDONNIPHHP
|
7.7 | IC50 | 3 | — | |
VGVIWBCNXYVLQY
|
7.7 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
7.7 | Kd | 165 | Yes | |
VHRZLROQUWIXSC
|
7.7 | IC50 | 3 | — | |
RJGLNSNPZNKTGL
|
7.6 | IC50 | 2 | — | |
GMIIXDTZSKOUIW
|
7.6 | IC50 | 2 | — | |
ONQYZCIVDNVJRE
|
7.6 | Ki | 2 | — | |
PSDOGBDKRWOMIK
|
7.6 | IC50 | 3 | — | |
UIEXDKQSWATHMD
|
7.6 | IC50 | 3 | — | |
CITPEYUXGCJVRV
|
7.6 | IC50 | 2 | — | |
IEZVBDUJVUPHKM
|
7.5 | IC50 | 3 | — | |
XJNGZIGUKNHSJB
|
7.5 | IC50 | 2 | — |