Target Details
| UniProt AC | P33981 |
|---|---|
| Gene Symbol | TTK |
| Protein Name | Dual specificity protein kinase TTK |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 178
- Clinical molecules 17
- Avg pChEMBL 7.57
KEGG Pathways (1)
Active Molecules (178)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TXGCEDYNBXDZEI
|
9.2 | IC50 | 2 | — | |
WHJIHZSXTQRCNX
|
9.1 | Kd | 10 | — | |
LZKFDPIUYGTKHZ
|
9.0 | IC50 | 3 | — | |
UVHDAKLRGJSVKQ
|
9.0 | IC50 | 4 | — | |
MCYPGAGHAANYON
|
8.9 | IC50 | 3 | — | |
DUKJABPGWUISRC
|
8.9 | IC50 | 3 | — | |
JQONSQMAQRQLRF
|
8.9 | IC50 | 2 | — | |
PMQUGSPFUBGJCZ
|
8.9 | IC50 | 2 | — | |
PMDUMOUXISSZED
|
8.8 | IC50 | 3 | — | |
SPYVZMIWNDEJND
|
8.8 | IC50 | 2 | — | |
CCGBGSFDXIBQHC
|
8.8 | IC50 | 3 | — | |
IEEIUNGYFLCIKQ
|
8.8 | IC50 | 3 | — | |
NRJKIOCCERLIDG
|
8.8 | IC50 | 6 | — | |
RJPWVZWPESKSOM
|
8.8 | IC50 | 3 | — | |
XRBFZYFJBUZBIE
|
8.8 | IC50 | 2 | — | |
CLYMONPGUOMIQL
|
8.7 | IC50 | 3 | — | |
WNMOTZHMKYYWSU
|
8.7 | IC50 | 3 | — | |
XEADJJXUBNVGAN
|
8.7 | IC50 | 3 | — | |
KFENBNGSHOHELN
|
8.7 | IC50 | 2 | — | |
VZBGYKSZEPEEDD
|
8.7 | IC50 | 3 | — | |
DUZMKFLMNMTYDM
|
8.7 | IC50 | 4 | — | |
JNOGLIZMJJRCIW
|
8.7 | IC50 | 2 | — | |
TWPZRFZCHZSVKG
|
8.7 | IC50 | 4 | — | |
YMYOREROCXXANC
|
8.6 | IC50 | 4 | — | |
YDGTUAFFLKCKEE
|
8.6 | IC50 | 3 | — | |
IRGIWNWHHPMOLO
|
8.6 | IC50 | 3 | — | |
XRBFZYFJBUZBIE
|
8.6 | IC50 | 2 | — | |
IYBGHBZUXSMOKI
|
8.6 | IC50 | 3 | — | |
DUKJABPGWUISRC
|
8.5 | IC50 | 10 | — | |
JBZRAEUHDPMQSF
|
8.5 | IC50 | 34 | — | |
XTULNCWAJUYUIA
|
8.5 | IC50 | 4 | — | |
FMRUHQLKCRUMNL
|
8.5 | IC50 | 4 | — | |
JAHXQCZCZURPTI
|
8.4 | IC50 | 34 | — | |
MLMUOABLNWGSQB
|
8.4 | IC50 | 3 | — | |
UVHDAKLRGJSVKQ
|
8.4 | IC50 | 3 | — | |
CHAZIKNZOXHZJA
|
8.4 | IC50 | 3 | — | |
HKIZNKMCQOQZTI
|
8.4 | IC50 | 3 | — | |
KTPMQAQBFZCIRN
|
8.4 | IC50 | 3 | — | |
GFUQINLLDUOCSK
|
8.4 | IC50 | 3 | — | |
VTWYCQYMWJLMTC
|
8.4 | IC50 | 2 | — | |
WGEHOPBYUQXTMK
|
8.4 | IC50 | 2 | — | |
YPJRHEKCFKOVRT
|
8.4 | Kd | 12 | — | |
VTWYCQYMWJLMTC
|
8.4 | IC50 | 2 | — | |
AFPQNJFINOFINI
|
8.4 | IC50 | 3 | — | |
LFMAIWOVKYCOOZ
|
8.4 | IC50 | 3 | — | |
JQONSQMAQRQLRF
|
8.3 | IC50 | 2 | — | |
AFPQNJFINOFINI
|
8.3 | IC50 | 4 | — | |
HMSPYGGDZVMDBA
|
8.3 | IC50 | 3 | — | |
SIBUVHVSIBBFAL
|
8.3 | IC50 | 3 | — | |
JQBMRWMXRCFFOP
|
8.3 | IC50 | 2 | — |