Target Details
| UniProt AC | P33527 |
|---|---|
| Gene Symbol | ABCC1 |
| Protein Name | Multidrug resistance-associated protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00664 (ABC_membrane) PF00005 (ABC_tran) PF24357 (TMD0_ABC) |
Summary
- Multi-target molecules 23
- Clinical molecules 0
- Avg pChEMBL 6.63
KEGG Pathways (6)
Associated Diseases (1)
Active Molecules (23)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SGTNSNPWRIOYBX
|
7.5 | Kd | 2 | — | |
RDMBCGVGRBUTKT
|
7.4 | IC50 | 2 | — | |
BLIMNWSQDQYNMP
|
7.1 | IC50 | 2 | — | |
SGTNSNPWRIOYBX
|
7.1 | IC50 | 19 | — | |
LWMRNOHPZGMUEC
|
7.0 | IC50 | 2 | — | |
SGTNSNPWRIOYBX
|
7.0 | Kd | 2 | — | |
KFCQYUZRWULLQM
|
6.9 | IC50 | 2 | — | |
VNMQONKZFZQPCT
|
6.8 | IC50 | 3 | — | |
XPNBVAOZAHYCST
|
6.8 | IC50 | 3 | — | |
WHQCHUCQKNIQEC
|
6.7 | Ki | 6 | — | |
NECCTVFNAYKBCX
|
6.5 | IC50 | 3 | — | |
OEIXJPAIZADICN
|
6.5 | IC50 | 3 | — | |
OEIXJPAIZADICN
|
6.5 | IC50 | 3 | — | |
WSQDGWOFRGACTF
|
6.4 | IC50 | 2 | — | |
ARBDURHEPGRPSR
|
6.4 | IC50 | 2 | — | |
VNMQONKZFZQPCT
|
6.4 | IC50 | 3 | — | |
XPNBVAOZAHYCST
|
6.4 | IC50 | 3 | — | |
JKKFKPJIXZFSSB
|
6.3 | Ki | 2 | — | |
AZSNMRSAGSSBNP
|
6.3 | Ki | 2 | — | |
AXUZQJFHDNNPFG
|
6.2 | Ki | 3 | — | |
OIKGUIRGSMTFAP
|
6.1 | IC50 | 2 | — | |
SCJLWMXOOYZBTH
|
6.1 | IC50 | 2 | — | |
SCJLWMXOOYZBTH
|
6.1 | IC50 | 2 | — |