Target Details
| UniProt AC | P33176 |
|---|---|
| Gene Symbol | KIF5B |
| Protein Name | Kinesin-1 heavy chain |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00225 (Kinesin) |
Summary
- Multi-target molecules 46
- Clinical molecules 4
- Avg pChEMBL 7.23
KEGG Pathways (11)
Active Molecules (46)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FWEAPVSZAHZTHG
|
8.9 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.8 | IC50 | 408 | — | |
YRBWLEAMGAGYBK
|
8.8 | IC50 | 6 | — | |
ZTIHSLVMCONHQU
|
8.5 | IC50 | 5 | — | |
GBLBJPZSROAGMF
|
8.3 | IC50 | 4 | — | |
CRQNIBKIWTWDFL
|
8.3 | IC50 | 3 | — | |
WOEVJDXDZJWENO
|
8.2 | IC50 | 3 | — | |
BLYRPGBSIKAIAU
|
8.2 | IC50 | 24 | Yes | |
JCCUAVDBGXASEC
|
8.1 | IC50 | 3 | — | |
WOSKHXYHFSIKNG
|
8.0 | IC50 | 24 | — | |
UKYJKXMPIDEQFF
|
8.0 | IC50 | 16 | — | |
JIBBGYSUSKAPDY
|
8.0 | IC50 | 19 | — | |
UYXYKLOTLJDLNL
|
7.8 | IC50 | 4 | — | |
NWKUBTQEYKTRNT
|
7.7 | IC50 | 4 | — | |
FJTQBVRKZLEDPK
|
7.7 | IC50 | 4 | — | |
ZVVQDNWRXSSQDL
|
7.5 | IC50 | 3 | — | |
YZNIHXUBUWEUCM
|
7.4 | IC50 | 14 | — | |
XHXOJKOXEKXDSQ
|
7.4 | IC50 | 5 | Yes | |
PAFIGBIGZBXCGJ
|
7.4 | IC50 | 2 | — | |
YFVCYTODGMGPAD
|
7.4 | IC50 | 4 | — | |
FHZCSNTVCRCIKT
|
7.3 | IC50 | 3 | — | |
RNIXZCQWBPDHPR
|
7.3 | IC50 | 3 | — | |
ZHPRBIFEDSMSRL
|
7.2 | IC50 | 2 | — | |
ATYKMHIJRBRZOA
|
7.2 | IC50 | 2 | — | |
QZKXRJMVQTZACR
|
7.1 | IC50 | 3 | — | |
TXFSECOZKAKHMC
|
7.1 | IC50 | 3 | — | |
HLOASMXRJBZZAG
|
7.0 | IC50 | 3 | — | |
UXWNRDQAMADNES
|
6.9 | IC50 | 3 | — | |
AAQXIFQQTLXRNG
|
6.9 | IC50 | 2 | — | |
ONIQOQHATWINJY
|
6.7 | IC50 | 25 | — | |
FASQTICQHQVOKY
|
6.7 | IC50 | 3 | — | |
DZPXNXYARLTMGL
|
6.6 | IC50 | 2 | — | |
NRBCZVLKKQZZNF
|
6.6 | IC50 | 2 | — | |
UHKNINGWQKGQGB
|
6.6 | IC50 | 3 | — | |
OPRQSQDMYPVYOV
|
6.6 | IC50 | 7 | — | |
BNDYIYYKEIXHNK
|
6.4 | IC50 | 7 | Yes | |
UHTHHESEBZOYNR
|
6.4 | IC50 | 66 | Yes | |
OYIGMLCBXUNGGL
|
6.3 | IC50 | 3 | — | |
XPEVSMSGIHLOSK
|
6.3 | IC50 | 3 | — | |
IKZPPFXCBWIVPC
|
6.3 | IC50 | 3 | — | |
XRFFUVUJIBWJII
|
6.3 | IC50 | 3 | — | |
ARRUJZPOJKKPKY
|
6.2 | IC50 | 3 | — | |
GITWBPKQKQFIAW
|
6.2 | IC50 | 2 | — | |
NMJIPDOHEVXEHN
|
6.2 | IC50 | 3 | — | |
HDWGWERBFXSKLX
|
6.1 | IC50 | 2 | — | |
CEQUQTKEVIQAMX
|
6.0 | IC50 | 3 | — |