Target Details
| UniProt AC | P33032 |
|---|---|
| Gene Symbol | MC5R |
| Protein Name | Melanocortin receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 383
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (383)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DABVBFWVYRMYNW
|
6.1 | IC50 | 3 | — | |
JCWSTHXQYUMWKE
|
6.1 | IC50 | 3 | — | |
VHZUXXIKZIQBLB
|
6.1 | IC50 | 2 | — | |
HIYNTZOLQGBWSI
|
6.1 | IC50 | 2 | — | |
HIYNTZOLQGBWSI
|
6.1 | IC50 | 2 | — | |
XJIWJTAALOWWFJ
|
6.1 | Ki | 3 | — | |
WBTHAPYEEKFPSX
|
6.1 | IC50 | 4 | — | |
YMCLJESYNLOGEG
|
6.1 | IC50 | 2 | — | |
GDRJSPPVRGELGB
|
6.1 | Ki | 3 | — | |
WETYFBSRFBUFCI
|
6.1 | IC50 | 3 | — | |
CGANDSYNDFLFKG
|
6.1 | Ki | 4 | — | |
IVOZSKOYXPHCOQ
|
6.1 | IC50 | 3 | — | |
DADQHECQKQBHAW
|
6.1 | Ki | 3 | — | |
JBPCVEBLPIKYKT
|
6.1 | IC50 | 3 | — | |
VFHJQMPJMWPJBF
|
6.1 | IC50 | 2 | — | |
XHTPNLWJKHXMSN
|
6.1 | Ki | 3 | — | |
HHHGGOMKUAYOJZ
|
6.0 | Ki | 3 | — | |
NSFFFSYEDFVOOT
|
6.0 | Ki | 2 | — | |
RBLCKVWSBGCRJN
|
6.0 | Ki | 2 | — | |
ARFBDECCXOFCBN
|
6.0 | IC50 | 3 | — | |
KHTORJRLHSSEND
|
6.0 | IC50 | 3 | — | |
JUZSSTZMGZLRNQ
|
6.0 | Ki | 2 | — | |
PUBNSQFRKLLQSF
|
6.0 | Ki | 2 | — | |
IKTNZHMAWQNOLP
|
6.0 | Ki | 2 | — | |
GRAFEEBFOIOLGS
|
6.0 | Ki | 3 | — | |
GWQJQMUYAJRYAV
|
6.0 | Ki | 2 | — | |
HPVULTYLDIMYRI
|
6.0 | IC50 | 3 | — | |
RSKJGGLMXZWIBS
|
6.0 | IC50 | 2 | — | |
RSZGGZUMSYSTES
|
6.0 | Ki | 3 | — | |
RSZGGZUMSYSTES
|
6.0 | Ki | 3 | — | |
RZLPZBLBQNNVLZ
|
6.0 | Ki | 2 | — | |
SPKUFMODEUMWTR
|
6.0 | Ki | 2 | — | |
YEUMEJHOKABUMX
|
6.0 | Ki | 2 | — |