Target Details
| UniProt AC | P33032 |
|---|---|
| Gene Symbol | MC5R |
| Protein Name | Melanocortin receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 383
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (383)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WZIILWAZGXRRFZ
|
6.8 | IC50 | 4 | — | |
XFQWSJOXRAVFGY
|
6.8 | Ki | 3 | — | |
BBYTXRAQNPWSMC
|
6.8 | IC50 | 3 | — | |
HAIHKNYZIMVIIW
|
6.8 | Ki | 3 | — | |
STCDJTWBNWJNLP
|
6.8 | Ki | 2 | — | |
LGJDLKCHZMGHIM
|
6.8 | IC50 | 2 | — | |
MSRUJRYKGIBVTG
|
6.8 | IC50 | 4 | — | |
OBNLGUMWGVRYJW
|
6.8 | IC50 | 3 | — | |
VFJOTTZGMDRNPT
|
6.8 | Ki | 3 | — | |
WLIRRQCYHFOXGC
|
6.8 | IC50 | 4 | — | |
JLMVHMLMBIPZSW
|
6.8 | IC50 | 4 | — | |
UICVQJGBBAMKDX
|
6.8 | IC50 | 4 | — | |
GZWUQPQBOGLSIM
|
6.8 | IC50 | 3 | — | |
PVVLKBSYHAGXBD
|
6.8 | IC50 | 4 | — | |
QEQUHVRIJFFOKD
|
6.8 | IC50 | 4 | — | |
DTYOAGHBUMBHBH
|
6.8 | IC50 | 3 | — | |
LDHOENQCWMSQTE
|
6.8 | IC50 | 3 | — | |
RETXHZDMGJHDNV
|
6.8 | Ki | 3 | — | |
UVJBRYNBZSRMBZ
|
6.8 | IC50 | 4 | — | |
CZTOIAMYLKDGSL
|
6.8 | IC50 | 3 | — | |
KNWLOSLCTAQNSO
|
6.8 | IC50 | 4 | — | |
RCULCPVSLOFQPR
|
6.8 | IC50 | 4 | — | |
FRHMEXCWIHUKBH
|
6.8 | IC50 | 3 | — | |
KBLNYXZHILRCGF
|
6.8 | IC50 | 4 | — | |
HICQRDPLMADMBD
|
6.7 | IC50 | 4 | — | |
LAHUDBCXWRATGM
|
6.7 | Ki | 3 | — | |
NTMXDNFEFWCVSA
|
6.7 | IC50 | 3 | — | |
TUEXZDIGHDGDGO
|
6.7 | IC50 | 3 | — | |
IVQPGYKGSXUDKV
|
6.7 | IC50 | 4 | — | |
KWTLWMHGSUOSHU
|
6.7 | IC50 | 4 | — | |
NMMRTJBOGUWCEQ
|
6.7 | Ki | 4 | — | |
ROTHBSFMHAHRTG
|
6.7 | IC50 | 4 | — | |
UHMCIGUGJPINOI
|
6.7 | IC50 | 3 | — | |
VLMJSBZOGGFEED
|
6.7 | Ki | 3 | — | |
VOCXANHYYBVTET
|
6.7 | Ki | 4 | — | |
FFHBJDQSGDNCIV
|
6.7 | IC50 | 4 | — | |
FPYYFGFPTJRMBR
|
6.7 | IC50 | 3 | — | |
KSMXNEYOFKPWFI
|
6.7 | IC50 | 4 | — | |
WRXWCWIFEFKMJL
|
6.7 | IC50 | 3 | — | |
FIPGSBWOMGALGM
|
6.7 | IC50 | 4 | — | |
NCLQWDCIPKHQBS
|
6.7 | IC50 | 2 | — | |
QAXKNGODUAVCKD
|
6.7 | IC50 | 4 | — | |
KPAXZSMXFNRRAR
|
6.7 | IC50 | 3 | — | |
SMAWMSUKCNWJNR
|
6.7 | Ki | 3 | — | |
VWRQHODLDKRSNP
|
6.7 | IC50 | 4 | — | |
GUUMVPUVSBGKBI
|
6.7 | IC50 | 3 | — | |
UKCAJRRGLXHDRO
|
6.7 | Ki | 2 | — | |
VKDMHINLWUJYEZ
|
6.7 | IC50 | 3 | — | |
HCIQMSLDYBLSJK
|
6.7 | Ki | 4 | — | |
MENIABFEGRBVAB
|
6.6 | Ki | 4 | — |