Target Details
| UniProt AC | P33032 |
|---|---|
| Gene Symbol | MC5R |
| Protein Name | Melanocortin receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 383
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (383)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IFDBWKFSUPQKCA
|
7.2 | IC50 | 4 | — | |
UTARRQKZBUCQBR
|
7.2 | Ki | 3 | — | |
MIAUOPQGTJQSKK
|
7.2 | IC50 | 2 | — | |
IPSFANQKYGITFT
|
7.2 | Ki | 3 | — | |
OVCXMKITXFVUSL
|
7.2 | IC50 | 3 | — | |
WGLOHHGRWPHJBM
|
7.2 | IC50 | 3 | — | |
YQOPVQXIKMEFFV
|
7.2 | IC50 | 4 | — | |
MWAZOIYNZZSBNG
|
7.1 | IC50 | 2 | — | |
IQLBYPCPYGLSQC
|
7.1 | IC50 | 3 | — | |
RANDNDRFMFBRFD
|
7.1 | IC50 | 3 | — | |
KYLMYZLCQJJVMF
|
7.1 | IC50 | 4 | — | |
XLLJFSCSXTYVTN
|
7.1 | Ki | 4 | — | |
YHYBBOPOIUAVHY
|
7.1 | IC50 | 3 | — | |
KMNARKQYUZICHM
|
7.1 | IC50 | 3 | — | |
HQACQGVVMYJUAG
|
7.1 | Ki | 3 | — | |
YXIBEMYOGWJEQC
|
7.1 | IC50 | 4 | — | |
QUNJOVXJJGQTDV
|
7.1 | IC50 | 3 | — | |
APHPBWUTFHDTLW
|
7.0 | IC50 | 4 | — | |
PBZOSRKDAHPMMH
|
7.0 | IC50 | 2 | — | |
BLUHVPTUPSCCBC
|
7.0 | IC50 | 2 | — | |
YEXGHTGVNJDCFJ
|
7.0 | IC50 | 3 | — | |
GUWAZMLXUQIQKT
|
7.0 | IC50 | 4 | — | |
GYFGNZUSQUDKII
|
7.0 | IC50 | 3 | — | |
AWLXWEMCGRJJAO
|
7.0 | IC50 | 2 | — | |
JKJKHYOUTNOITO
|
7.0 | IC50 | 3 | — | |
JWVUTJWCWBNVDW
|
7.0 | IC50 | 3 | — | |
APAIPJOPPUMQFD
|
7.0 | IC50 | 4 | — | |
DFCJPPDAOZROBS
|
7.0 | IC50 | 4 | — | |
GUUMVPUVSBGKBI
|
7.0 | IC50 | 3 | — | |
MCJFEKJJFCZAHM
|
7.0 | Ki | 3 | — | |
STHTUYXXUBUJIE
|
7.0 | IC50 | 2 | — | |
TVCZNUJSXSNMJP
|
7.0 | Ki | 3 | — | |
PHHQWWPLQKXGDH
|
6.9 | IC50 | 4 | — | |
TVKPENPJQKTJFK
|
6.9 | IC50 | 3 | — | |
OFPOZEFXTIZAHE
|
6.9 | Ki | 4 | — | |
PGOKBMWPBDRDGN
|
6.9 | IC50 | 8 | — | |
WHNFPRLDDSXQCL
|
6.9 | IC50 | 4 | — | |
YTZPUJBWCYPFRS
|
6.9 | IC50 | 3 | — | |
YTZPUJBWCYPFRS
|
6.9 | IC50 | 3 | — | |
BCFFSQJVHOEAAU
|
6.9 | IC50 | 3 | — | |
SHVFCFMJFUMOGL
|
6.9 | IC50 | 2 | — | |
DOVNDOSDULTCGE
|
6.9 | IC50 | 3 | — | |
FWQGDGPDBUUACD
|
6.9 | Ki | 3 | — | |
IXLVDOBKTIIMBE
|
6.9 | IC50 | 4 | — | |
PWADIMGJQZHREF
|
6.9 | IC50 | 2 | — | |
CMKWAAKJKOZNBH
|
6.9 | Ki | 4 | — | |
BVHVEJVRGYHQTC
|
6.9 | IC50 | 3 | — | |
NOLFWMRTIVNJFP
|
6.9 | IC50 | 4 | — | |
HAIHKNYZIMVIIW
|
6.8 | Ki | 3 | — | |
WZIILWAZGXRRFZ
|
6.8 | IC50 | 3 | — |