Target Details
| UniProt AC | P33032 |
|---|---|
| Gene Symbol | MC5R |
| Protein Name | Melanocortin receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 383
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (383)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YMEXHIACKAXZLZ
|
7.7 | IC50 | 3 | — | |
AODONYDDQNDROG
|
7.7 | IC50 | 2 | — | |
HRTHPANNFOMYJE
|
7.6 | IC50 | 4 | — | |
IFDBWKFSUPQKCA
|
7.6 | IC50 | 4 | — | |
WMMWJBFBADMJIK
|
7.6 | Ki | 3 | — | |
WZIILWAZGXRRFZ
|
7.6 | IC50 | 4 | — | |
XQMPAWYRHAOJTE
|
7.6 | Ki | 4 | — | |
OUFAADNZNCCMJZ
|
7.6 | Ki | 4 | — | |
GGYWLZFXFKFWKL
|
7.6 | Ki | 3 | — | |
JKPIUTPQBDXSRH
|
7.6 | Ki | 3 | — | |
CHNMWUKSZIMHIX
|
7.6 | Ki | 3 | — | |
UKCAJRRGLXHDRO
|
7.6 | Ki | 3 | — | |
YUUZCRILYWDWPO
|
7.6 | IC50 | 3 | — | |
CRWGRYHHKDTXFC
|
7.6 | IC50 | 3 | — | |
QVLFTJGCGVDBFK
|
7.5 | Ki | 3 | — | |
SZCLBSHELXLOEC
|
7.5 | Ki | 4 | — | |
QDDPPGFVMRPNTQ
|
7.5 | IC50 | 2 | — | |
WWDUVSWFUPRTGG
|
7.5 | Ki | 4 | — | |
IXQMIHWLSWEYPU
|
7.5 | IC50 | 4 | — | |
NMZQXNVSJCWFFD
|
7.5 | IC50 | 4 | — | |
BGNHNMCZDLGXJG
|
7.5 | Ki | 3 | — | |
IDDVSLRYKLDACE
|
7.5 | Ki | 4 | — | |
MRFZKAWUCKFKJV
|
7.5 | IC50 | 3 | — | |
PIVHBXZYYYPXHW
|
7.5 | IC50 | 4 | — | |
SFGAMHAXMGIWOF
|
7.4 | IC50 | 3 | — | |
DZOXHHUQYQUKJB
|
7.4 | IC50 | 4 | — | |
MNSNXOUQPSOGHN
|
7.4 | IC50 | 3 | — | |
VJXLJBSRIOMQLS
|
7.4 | IC50 | 4 | — | |
LZYYGZAXFMYSBE
|
7.4 | Ki | 4 | — | |
LKIXKBAXFLOUEW
|
7.4 | Ki | 4 | — | |
XLDGDUSCVKLZIR
|
7.4 | IC50 | 4 | — | |
YENCSZMEVJAKQJ
|
7.4 | IC50 | 4 | — | |
KIFNALNSUOJQPJ
|
7.4 | Ki | 4 | — | |
ZKFHMXVIVJCDFY
|
7.4 | IC50 | 4 | — | |
PAILFUNFWZLMMN
|
7.4 | IC50 | 3 | — | |
PIBQDSQILSXEKV
|
7.3 | IC50 | 2 | — | |
QIKIYIZHGOCQOO
|
7.3 | Ki | 3 | — | |
XVOPWUWRTVGXCT
|
7.3 | IC50 | 3 | — | |
YRPCDHHSQYGEDU
|
7.3 | IC50 | 4 | — | |
LKFLMXAGXFBGSV
|
7.3 | IC50 | 3 | — | |
ZWUGIRDPPFGGRP
|
7.3 | IC50 | 2 | — | |
BHIQIMLFSJYURU
|
7.3 | IC50 | 4 | — | |
ORPYCWJPNJKZIA
|
7.3 | IC50 | 4 | — | |
SZGSXARYIZZWDD
|
7.3 | IC50 | 3 | — | |
ANGMCMXZFGHVPX
|
7.2 | Ki | 3 | — | |
UNHHVHLFOZEIIS
|
7.2 | IC50 | 2 | — | |
XGLRKMGBEOEUSM
|
7.2 | IC50 | 2 | — | |
WQIHSOXKRYCWEW
|
7.2 | IC50 | 4 | — | |
PWVUYOZSIWYFJW
|
7.2 | Ki | 4 | — | |
KXWAHHUIDLURNT
|
7.2 | IC50 | 4 | — |