Target Details
| UniProt AC | P33032 |
|---|---|
| Gene Symbol | MC5R |
| Protein Name | Melanocortin receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 383
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (383)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KWBYYFKCXHSTPA
|
8.4 | IC50 | 4 | — | |
NEVVXMYOTHZJES
|
8.4 | IC50 | 3 | — | |
NEVVXMYOTHZJES
|
8.4 | IC50 | 3 | — | |
ORPOIIFPKJKKPO
|
8.4 | IC50 | 2 | — | |
IVRFZQRHPFZUMZ
|
8.4 | Ki | 4 | — | |
JMFDAPXKXHNPIL
|
8.4 | Ki | 3 | — | |
YBWGYSWBATYFBD
|
8.4 | IC50 | 4 | — | |
FDLHDUZIGJCBAK
|
8.3 | IC50 | 3 | — | |
FDLHDUZIGJCBAK
|
8.3 | IC50 | 3 | — | |
BBJOQSQVKOIBHK
|
8.3 | IC50 | 4 | — | |
FHNLUGMXKXPEFR
|
8.3 | IC50 | 4 | — | |
LMTCYYTZYVZVDJ
|
8.3 | Ki | 4 | — | |
DLVAKQPHOINITK
|
8.2 | IC50 | 4 | — | |
KZXNIFOXWZLCOK
|
8.2 | IC50 | 4 | — | |
KRKYTJXTDCSSJS
|
8.2 | IC50 | 4 | — | |
UAISFSHHKXHKOI
|
8.2 | IC50 | 4 | — | |
GGYWLZFXFKFWKL
|
8.2 | IC50 | 4 | — | |
ILTSJNSAHXKVSQ
|
8.2 | Ki | 3 | — | |
PIHBUAVCWXDWIB
|
8.2 | Ki | 3 | — | |
JDKLPDJLXHXHNV
|
8.1 | IC50 | 4 | — | |
ZPANOUCVWZTSLE
|
8.1 | IC50 | 4 | — | |
RVVLJWZWXHPMLS
|
8.1 | IC50 | 4 | — | |
AMLJFTMENZUCBN
|
8.1 | Ki | 3 | — | |
JGBGNKDRAKSUHZ
|
8.0 | Ki | 4 | — | |
QQCJWXXVYXUARZ
|
8.0 | IC50 | 3 | — | |
UAHFGYDRQSXQEB
|
8.0 | Ki | 3 | — | |
FPYYFGFPTJRMBR
|
8.0 | IC50 | 4 | — | |
CZCIDYFBUVIGBB
|
7.9 | IC50 | 3 | — | |
CZCIDYFBUVIGBB
|
7.9 | IC50 | 3 | — | |
KXCTVHIJPZQMDC
|
7.9 | IC50 | 4 | — | |
PBZOSRKDAHPMMH
|
7.9 | IC50 | 2 | — | |
BGQGGVJRXUWNNU
|
7.9 | Ki | 3 | — | |
CETOWTIWZXCWLA
|
7.9 | Ki | 3 | — | |
CQUKLRIOLMQYDE
|
7.9 | IC50 | 4 | — | |
ZTSQVRSYAGAZPG
|
7.8 | Ki | 4 | — | |
QBPUPEUBMHTUDK
|
7.8 | Ki | 3 | — | |
UYKWHGIEHONMDL
|
7.8 | IC50 | 4 | — | |
RBZTXCPXQHRLIB
|
7.8 | Ki | 3 | — | |
XATASKINOVYSLA
|
7.8 | IC50 | 3 | — | |
XATASKINOVYSLA
|
7.8 | IC50 | 3 | — | |
CHPABUPLIAAUIT
|
7.8 | IC50 | 4 | — | |
QTGLDSNZORTQEK
|
7.8 | IC50 | 4 | — | |
GSECRIQNUWHRKM
|
7.8 | Ki | 3 | — | |
KDTZLQMUHBEBMZ
|
7.8 | IC50 | 3 | — | |
PZVZJDCUPVOTTP
|
7.7 | IC50 | 4 | — | |
RVEIEULWMVBMRD
|
7.7 | IC50 | 4 | — | |
VESJJEZSWHFEGA
|
7.7 | Ki | 3 | — | |
KYRVGEKZJIYJKZ
|
7.7 | Ki | 3 | — | |
ZRCSDDHAGXRMLM
|
7.7 | IC50 | 4 | — | |
RQCWCCUAQKMWGM
|
7.7 | IC50 | 4 | — |