Target Details
| UniProt AC | P33032 |
|---|---|
| Gene Symbol | MC5R |
| Protein Name | Melanocortin receptor 5 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 383
- Clinical molecules 0
- Avg pChEMBL 7.18
KEGG Pathways (2)
Active Molecules (383)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QXDWLOZJHHTTCF
|
10.6 | IC50 | 3 | — | |
QXDWLOZJHHTTCF
|
10.6 | IC50 | 3 | — | |
JNEKRCCXHUFBPL
|
10.5 | IC50 | 3 | — | |
JNEKRCCXHUFBPL
|
10.5 | IC50 | 3 | — | |
GGYWLZFXFKFWKL
|
10.1 | Ki | 3 | — | |
KHGZKFBKKYRZCD
|
10.0 | IC50 | 3 | — | |
KHGZKFBKKYRZCD
|
10.0 | IC50 | 3 | — | |
QOZPHXSKYHWXNY
|
9.8 | IC50 | 4 | — | |
BUVGQEXSQXRZQG
|
9.8 | Ki | 4 | — | |
XDLJELQQEILLFZ
|
9.6 | Ki | 4 | — | |
GGYWLZFXFKFWKL
|
9.6 | IC50 | 4 | — | |
XUCSIJVANOTEDW
|
9.4 | Ki | 3 | — | |
SPJYDEIJYHHMBB
|
9.4 | IC50 | 3 | — | |
UBKGFMZTCLCOLM
|
9.3 | Ki | 4 | — | |
AOMUTEUZPCRNFD
|
9.2 | Ki | 3 | — | |
REMHNXQVRVXAGT
|
9.2 | IC50 | 4 | — | |
WSDYWWDQJYPQDS
|
9.1 | Ki | 3 | — | |
ZSONGANRJTVTCP
|
9.1 | Ki | 4 | — | |
UAHFGYDRQSXQEB
|
9.1 | IC50 | 5 | — | |
UMHVNRYGRKBTCG
|
9.0 | IC50 | 4 | — | |
SNEMRJZDOOLWPZ
|
8.9 | Ki | 4 | — | |
UVUOMESIOOEXGA
|
8.9 | IC50 | 3 | — | |
FDPBRBMLLVILMV
|
8.8 | Ki | 3 | — | |
TUOOEJAUOYDGGA
|
8.8 | IC50 | 4 | — | |
XTFWFFODDNNYFQ
|
8.8 | Ki | 4 | — | |
WSDYWWDQJYPQDS
|
8.7 | IC50 | 4 | — | |
RNCVEEUMKRRHLC
|
8.7 | IC50 | 4 | — | |
UKMQKNTZNHDSPD
|
8.7 | IC50 | 4 | — | |
UYOAPGITMAMCFT
|
8.7 | IC50 | 4 | — | |
TWDTYJMEGITLBP
|
8.7 | IC50 | 3 | — | |
GVZTZLFKKLVBJF
|
8.7 | IC50 | 3 | — | |
RDCIPOBDQMOUKD
|
8.7 | IC50 | 4 | — | |
REMHNXQVRVXAGT
|
8.7 | IC50 | 4 | — | |
AYKQERUAGGPJLP
|
8.6 | IC50 | 3 | — | |
UHCXNXMBPAFWDS
|
8.6 | IC50 | 3 | — | |
KRZXMSMNMZEKGP
|
8.6 | Ki | 4 | — | |
QBYHLGIJWBFDGJ
|
8.6 | IC50 | 4 | — | |
RVKSMTBVJXMWFD
|
8.6 | IC50 | 4 | — | |
UMHVNRYGRKBTCG
|
8.6 | IC50 | 4 | — | |
DFDCZNQATCGDRV
|
8.6 | IC50 | 3 | — | |
XMQSVPKHHVWBGS
|
8.6 | IC50 | 4 | — | |
JMNUTDPHHUFMOG
|
8.5 | Ki | 4 | — | |
BINHUIMAVHQSOM
|
8.5 | Ki | 4 | — | |
XPWIQGFRIVVHRC
|
8.5 | Ki | 4 | — | |
OHFMRHZLQMSCRN
|
8.5 | IC50 | 4 | — | |
BEGFBZSFSWOZDK
|
8.5 | Ki | 4 | — | |
UBWLAYRWNUNYHG
|
8.5 | IC50 | 4 | — | |
OKHXBJLIBJDJMV
|
8.5 | IC50 | 4 | — | |
TYFFXNLNRYRUAU
|
8.4 | IC50 | 3 | — | |
DQDUAZXNONBSMT
|
8.4 | Ki | 3 | — |