Target Details
| UniProt AC | P32298 |
|---|---|
| Gene Symbol | GRK4 |
| Protein Name | G protein-coupled receptor kinase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00615 (RGS) |
Summary
- Multi-target molecules 22
- Clinical molecules 8
- Avg pChEMBL 6.73
KEGG Pathways (3)
Active Molecules (22)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UIARLYUEJFELEN
|
7.9 | Kd | 289 | Yes | |
XZXHXSATPCNXJR
|
7.8 | Kd | 165 | Yes | |
ACLLLJSNOCYQOJ
|
7.7 | IC50 | 8 | — | |
HKSZLNNOFSGOKW
|
7.2 | IC50 | 408 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
GYMOXCZIQHPXOH
|
7.0 | IC50 | 6 | — | |
PIQCTGMSNWUMAF
|
7.0 | Kd | 137 | Yes | |
BMGQWWVMWDBQGC
|
7.0 | Kd | 147 | Yes | |
WINHZLLDWRZWRT
|
6.8 | Kd | 201 | Yes | |
JOOXLOJCABQBSG
|
6.8 | Kd | 139 | — | |
PTJBMQVUHYZJLN
|
6.7 | IC50 | 5 | — | |
LYADGAGFYYXXIO
|
6.6 | IC50 | 82 | — | |
XYUFCXJZFZPEJD
|
6.6 | IC50 | 23 | Yes | |
CTNPALGJUAXMMC
|
6.4 | Kd | 151 | — | |
GCIKSSRWRFVXBI
|
6.4 | Kd | 109 | Yes | |
OYONTEXKYJZFHA
|
6.4 | Kd | 69 | Yes | |
NHHQJBCNYHBUSI
|
6.3 | Kd | 220 | — | |
ZCBUQCWBWNUWSU
|
6.2 | Kd | 59 | — | |
NGFGTMFVWSDFPS
|
6.2 | IC50 | 32 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |