Target Details
UniProt ACP32297
Gene SymbolCHRNA3
Protein NameNeuronal acetylcholine receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 506
  • Clinical molecules 0
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (506)
InChIKey pChEMBL Type Targets Clinical
OHKODMIWVVUDGL 7.2 Ki 4
VHTBVZBRBLYBGN 7.2 IC50 3
ASEWWVGXMJQYTD 7.2 Ki 8
VHNSVCKCMBYGSB 7.2 Ki 5
IMYZQPCYWPFTAG 7.2 IC50 8
KKFHJNUEMBWTSM 7.2 Ki 2
QAIHOBDHHLOTET 7.2 IC50 3
BEXHXBAKDDOWBF 7.1 Ki 5
VHRLLJQAIUCUDP 7.1 IC50 3
BVYJHUNIDYEALI 7.1 IC50 3
GMXMIEACANMTOP 7.1 Ki 2
VXQLPXYMYHKASH 7.1 Ki 5
NJDRDZZUJLQOGS 7.1 Ki 2
WESGVHHRAFNWER 7.1 Ki 7
BGRDESOBNOVWPL 7.1 Ki 5
CIDBGGRUVLVTTA 7.1 Ki 2
DNTSAGFCYYBUKZ 7.1 Ki 5
HDEHBUBBSWDVRP 7.1 Ki 2
JQSHBVHOMNKWFT 7.1 Ki 6
YBSIIWUTXMMWKC 7.1 Ki 2
XQMFLUIVLXDXEJ 7.1 Ki 2
FVKMUNYZQFUOQQ 7.1 IC50 5
FAGJOGGAOOMVGD 7.1 IC50 3
GDXUHGVVRIPSQZ 7.1 Ki 5
UDMJZFWTHJHTRH 7.0 IC50 3
INYNWEUTASDACG 7.0 Ki 5
XNXRWSAXXLYNOY 7.0 Ki 2
LIWLPYIJYFIYKQ 7.0 Ki 2
ILEWLUJOKLLBMF 7.0 Ki 7
PMLHYFDQPIWSKJ 7.0 Ki 4
HTJXMVNJPKRWQD 7.0 IC50 2
LKHNWNJXVYAMBI 7.0 IC50 4
PJOMWQDGOKINIH 7.0 Ki 2
YOWFIQDENDEMRP 7.0 IC50 3
KPHRNXIFUJLFNL 7.0 Ki 5
KPHRNXIFUJLFNL 7.0 Ki 5
XKTDZPFHTDLVPX 7.0 Ki 2
CHUVPNWRFUBJRL 7.0 Ki 5
FANPYQPRSROCKC 7.0 IC50 3
SWFOYAMAGZFBGV 7.0 Ki 2
UQFKSUCKQFVMKL 7.0 Ki 2
WPIOOGNLSRYEIU 7.0 Ki 2
ZRTUGMRLPXGKGZ 7.0 Ki 3
AUBPMADJYNSPOA 7.0 Ki 2
NDEYLYXEJFWGDB 7.0 Ki 2
HFALPZZGNQXIMP 7.0 Ki 5
SKFPODQWUBSOEM 7.0 Ki 5
JZJRDFFBFLJGOB 7.0 Ki 2
XXWAUQHHHXAXMR 7.0 Ki 3
LJZVEMPJGOKQGQ 6.9 Ki 2
2D structure