Target Details
UniProt ACP32297
Gene SymbolCHRNA3
Protein NameNeuronal acetylcholine receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 506
  • Clinical molecules 0
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (506)
InChIKey pChEMBL Type Targets Clinical
AQYPBNGIIYVIBQ 7.6 Ki 5
ZAGVNQCMOLWFKV 7.6 Ki 5
ZUVFSXFHLMSSND 7.6 IC50 2
CRPBMTGSCRKOBR 7.5 Ki 5
QSEXENQMJGVARI 7.5 Ki 2
BFESRXFYMDMQQS 7.5 IC50 3
GPLPNYTYTRIAGH 7.5 IC50 3
HENZQJYUUUBJJV 7.5 Ki 2
IAPFRWYGZQXILQ 7.5 Ki 2
NURHOKYPHUZXFQ 7.5 IC50 4
OHTDTNHLFFCQRH 7.5 Ki 5
RPQSOKSDYSMFBW 7.5 IC50 3
JSWKSMHGVJDZBY 7.5 IC50 3
DTIFFHAURKBXJT 7.5 IC50 2
NGGVRPGLGXDGKP 7.5 Ki 7
UDGISDAHRCDXMV 7.5 IC50 6
FAEVMLINNNVLLK 7.4 Ki 5
UPRSNEUCMGKPCF 7.4 IC50 3
TZLUIMYGRBSVIB 7.4 Ki 3
UYZAXUWVJGHEFL 7.4 IC50 3
ZLLCEWCZDFPICU 7.4 Ki 5
GKNSLBAHDKWDHQ 7.4 Ki 5
PQBYYZBQJKBZMS 7.4 Ki 5
XUFHNWWGOZPOSG 7.4 Ki 2
AIKMSOHWSGWCNX 7.4 IC50 3
MZBXNOWXAZNDIQ 7.4 Ki 2
AQYPBNGIIYVIBQ 7.4 Ki 5
IKBFUAJBNDCGFQ 7.4 Ki 7
YCKUJRLTYLJWTR 7.4 Ki 5
GGPOGZSZLWNUEK 7.3 Ki 3
DEXLAAAKAUMETM 7.3 Ki 5
MFIANXNGKGYYND 7.3 Ki 2
WINQUAHGULGZED 7.3 IC50 5
ZTPUIOSCXSOSPV 7.3 Ki 2
QGZBKYBWQCGNTH 7.3 IC50 3
WHRKMMNRCVIVON 7.3 Ki 2
LTLFRBMKBHQUTH 7.3 IC50 2
LVYRPIRSEMMFEE 7.3 IC50 3
AQYPBNGIIYVIBQ 7.3 Ki 5
GGSJOBXYOUMOBW 7.2 Ki 2
TWVKXXKMLUVNDJ 7.2 Ki 5
AMMQVZPHMBRHME 7.2 IC50 3
BOLXMIIYJAOMEO 7.2 Ki 5
DJSUCHMXQOIATH 7.2 Ki 2
IEYQINPEMQKRDC 7.2 IC50 3
LKXXWFDWZQRZKV 7.2 IC50 3
ILLGYRJAYAAAEW 7.2 IC50 3
XMYWPQXQUQJAEN 7.2 Ki 2
ZWSIFNIMWCIVIU 7.2 IC50 3
DEGGHZFPJGYWCK 7.2 IC50 2
2D structure