Target Details
UniProt ACP32297
Gene SymbolCHRNA3
Protein NameNeuronal acetylcholine receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 506
  • Clinical molecules 0
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (506)
InChIKey pChEMBL Type Targets Clinical
GSEMJTPMJBMBRO 7.9 Ki 3
DLZUIBOQBIXZPS 7.9 IC50 3
OCEAINWYIRTVGD 7.9 Ki 5
RCSZDVCUNQPLHO 7.9 Ki 5
MFMVYBPYDSNLTE 7.9 IC50 3
GJKKKELBGQEBIU 7.9 Ki 2
PFEBDEOEEICVBY 7.9 Ki 2
VAPDPQSECMWOFE 7.9 IC50 3
JTTBYCVBUXQDTE 7.9 IC50 3
KBCGDBMDBJDDGG 7.9 Ki 3
HZRJVZGFTVHZGZ 7.8 Ki 2
INYNWEUTASDACG 7.8 Ki 5
LNIKTCCVSHMIFS 7.8 IC50 2
UEQZFAGVRGWPDK 7.8 IC50 3
YSVOMDFBWJGXEL 7.8 Ki 5
AMOKJMKEFDPTPN 7.8 IC50 7
DEXLAAAKAUMETM 7.8 Ki 5
GIUMMCXYLUQIND 7.8 Ki 5
LNIKTCCVSHMIFS 7.8 IC50 2
DWDCLEHDNICBMI 7.8 IC50 2
MLCFZENIQJYRSR 7.8 IC50 3
VIWKHXNVEIOPSC 7.8 IC50 10
DEXLAAAKAUMETM 7.8 Ki 5
HXZFPBBYBMMKAQ 7.8 Ki 2
KEJDQVGYGBHLMC 7.8 Ki 4
DJUPOXJVHQDKPZ 7.7 IC50 3
NZWMSQXPQAEDAS 7.7 Ki 4
QQODMJRPCBCHDU 7.7 IC50 3
GGPOGZSZLWNUEK 7.7 Ki 3
XTMVSVQIYRTKIW 7.7 IC50 5
GSEMJTPMJBMBRO 7.7 Ki 3
HBRLNTBOOKFZCC 7.7 Ki 5
RNOBTWYQAWEZHH 7.7 Ki 4
RVAVBFSGDWYYEQ 7.7 Ki 2
VIKPJXVYULNEFB 7.7 Ki 2
YJEMXDJGZIOQLT 7.7 IC50 3
RFCWACSNWRAYNU 7.7 IC50 3
SJGHGXWQPNNDCN 7.7 Ki 5
WXJMNOKWJJRHJY 7.7 IC50 3
BACMDOCEIHERJI 7.7 Ki 3
RVUUCOAHJHAFBX 7.6 IC50 3
YEYNZFAXDZFOHU 7.6 Ki 2
QWEBUPURHNWVEK 7.6 IC50 5
BEBIEORUESJWFE 7.6 Ki 5
ZQHLHLOXNNOIQM 7.6 Ki 2
BRSAFVDQMOMDOC 7.6 IC50 2
ASNYTHIFAFBQFH 7.6 IC50 3
DMDHFLXQSOBORU 7.6 Ki 5
HPZRKLOXXPCXBA 7.6 Ki 4
RPHSTODYKZLNFU 7.6 IC50 4
2D structure