Target Details
UniProt ACP32297
Gene SymbolCHRNA3
Protein NameNeuronal acetylcholine receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 506
  • Clinical molecules 0
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (506)
InChIKey pChEMBL Type Targets Clinical
CCGVLNAUEKVICK 8.4 IC50 8
WWXZQSSSEUIZDN 8.3 Ki 2
ZMRXSORFBXMBCB 8.3 IC50 8
RCSZDVCUNQPLHO 8.3 Ki 7
ZVMQAHYHODITTD 8.3 Ki 2
NTFKOQBZSNCLLA 8.3 Ki 4
MOMRLMDRIJFWPM 8.3 IC50 5
TZWVPYLQJDFQHL 8.3 Ki 5
ZLLCEWCZDFPICU 8.3 Ki 5
HQBAWNLKYLZICH 8.2 IC50 3
WHDFCXQEDDAKHI 8.2 IC50 3
GTMXEEZPDPKGRK 8.2 Ki 2
QCSSDCOJCQOKNU 8.2 Ki 5
TVSNVPGPFGAKPT 8.2 Ki 2
QGPJNUIJAGMDMT 8.2 Ki 5
VJEPFPRUUZASOL 8.2 Ki 5
MXUDEADPGZWZCH 8.2 IC50 9
VVDRDHLUVVGURR 8.2 IC50 5
AYYXJYPIJMOLEL 8.2 Ki 2
IMWUFTIDVKJBTJ 8.2 Ki 5
KBCGDBMDBJDDGG 8.1 Ki 5
VJEPFPRUUZASOL 8.1 Ki 5
DTWANULJDRVTFI 8.1 IC50 5
LOWDJVQAZMFOLZ 8.1 IC50 10
MVLJPWPLDPHKST 8.1 Ki 2
MLPOWHAMUPIMTC 8.1 IC50 4
JPNUKJAOPRHHRY 8.1 Ki 5
ZDTSCWZPUHXKPB 8.1 Ki 2
ZNRNCCOAWBUSNP 8.1 Ki 4
MVQIWKVEEIZQLL 8.1 IC50 5
ZLLCEWCZDFPICU 8.1 Ki 5
AGNZBWKVIGAWTQ 8.1 Ki 5
FLAHTCIVXKKZAR 8.1 IC50 3
CRXFCGUGNWJSEY 8.0 Ki 5
RNQSYWWRXUJHPF 8.0 Ki 2
YFMOKOLWGKJNCJ 8.0 IC50 3
AOTZFTGAQIRWOB 8.0 IC50 3
CXOPDJYVJZLVSY 8.0 Ki 6
KFULFWHCQIMTLB 8.0 Ki 4
MQVPACXYSJDEHQ 8.0 IC50 5
NMIIKXFGCKOYRV 8.0 IC50 5
JBABGZDZOMSKLX 8.0 IC50 8
KPHRNXIFUJLFNL 8.0 Ki 5
CFVHNYYHCCJXDK 8.0 IC50 9
CRXFCGUGNWJSEY 8.0 Ki 5
DDDMGCMKOCLAAT 8.0 IC50 8
DNVMLFGJFSQQDE 8.0 IC50 9
SNXCJPFZRZMRKK 8.0 IC50 3
VMEDIUSDIYRUSA 8.0 IC50 10
VYRZFHOORZTMRI 8.0 IC50 3
2D structure