Target Details
| UniProt AC | P32297 |
|---|---|
| Gene Symbol | CHRNA3 |
| Protein Name | Neuronal acetylcholine receptor subunit alpha-3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb) |
Summary
- Multi-target molecules 506
- Clinical molecules 0
- Avg pChEMBL 7.36
KEGG Pathways (4)
Associated Diseases (1)
Active Molecules (506)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RFLDYHWWEJNDMO
|
8.9 | Ki | 2 | — | |
JNFVNWDQFKSBOK
|
8.8 | Ki | 2 | — | |
QYLKSFXBRALDIS
|
8.8 | IC50 | 9 | — | |
AZKMTKVSVYHHAA
|
8.8 | IC50 | 4 | — | |
FBNWGQBXLLCHJM
|
8.8 | Ki | 2 | — | |
PAKVZEJOMQOKAO
|
8.8 | IC50 | 3 | — | |
DUQYFGMBLOPGBY
|
8.8 | IC50 | 3 | — | |
UBFPRQOOAXMTBD
|
8.8 | IC50 | 6 | — | |
YDGOUEKZXBLUDG
|
8.8 | IC50 | 8 | — | |
ZUQVZTJFSCBLOT
|
8.8 | IC50 | 3 | — | |
OHKBIDDJISYEHL
|
8.8 | Ki | 2 | — | |
RSEXFRQQJHVYPG
|
8.8 | IC50 | 4 | — | |
WJMKWBQPBBUJHD
|
8.7 | IC50 | 2 | — | |
RCSZDVCUNQPLHO
|
8.7 | Ki | 7 | — | |
DGQVZUDAKWRJPY
|
8.7 | IC50 | 8 | — | |
HGIKFFRIFIJEOP
|
8.7 | IC50 | 3 | — | |
WXTQMACZCSXJTB
|
8.7 | Ki | 4 | — | |
PLUODXWJLHWDCV
|
8.7 | Ki | 2 | — | |
MXJPOFBPCRQRTD
|
8.7 | IC50 | 3 | — | |
NBSDOPKWFMNCQW
|
8.7 | Ki | 2 | — | |
PEYVELBXXMIVMU
|
8.7 | Ki | 2 | — | |
SGVSOCSOUHHZAS
|
8.7 | IC50 | 3 | — | |
UIRMNVOEQMAKFM
|
8.7 | IC50 | 7 | — | |
TZWVPYLQJDFQHL
|
8.7 | Ki | 5 | — | |
SLZOZHRDAPBUAU
|
8.6 | IC50 | 2 | — | |
ISACHQOCISQFPP
|
8.6 | Ki | 4 | — | |
BMWDQBTXNBGORC
|
8.6 | IC50 | 8 | — | |
IELBAACIVCODPI
|
8.6 | IC50 | 8 | — | |
ZRCMYKLGYHVJGO
|
8.6 | Ki | 5 | — | |
JRPWUGPYWRJACU
|
8.6 | IC50 | 8 | — | |
NYPLKEHGCMPSAD
|
8.6 | Ki | 2 | — | |
SWPVFHZSTTYORI
|
8.6 | IC50 | 5 | — | |
YSSBTWFASLVAGY
|
8.6 | IC50 | 5 | — | |
UZJWAFOJOSGEKL
|
8.6 | Ki | 15 | — | |
GLNHQLYIFATJOO
|
8.6 | IC50 | 3 | — | |
YRTJBUGCGGXTRV
|
8.6 | IC50 | 5 | — | |
HVTMEGQWQQUDIH
|
8.5 | IC50 | 3 | — | |
PFEJBPNFLAFPKN
|
8.5 | IC50 | 10 | — | |
PUMYSIXHQPYXGX
|
8.5 | Ki | 4 | — | |
GTVWKLSULFFQST
|
8.5 | Ki | 7 | — | |
AGNZBWKVIGAWTQ
|
8.5 | Ki | 5 | — | |
ZKFFJBXJJFDBJM
|
8.5 | IC50 | 8 | — | |
SYMAJWVHHBJSJV
|
8.5 | IC50 | 8 | — | |
COKJMTQIZQACLZ
|
8.5 | IC50 | 3 | — | |
FIRBQKFGNFGBRC
|
8.5 | IC50 | 2 | — | |
LYGZRGMHPFAAMR
|
8.5 | Ki | 7 | — | |
ZRCMYKLGYHVJGO
|
8.5 | Ki | 5 | — | |
VLLKJTHFWNJPCE
|
8.4 | IC50 | 9 | — | |
OUHSMVDDOPDHGW
|
8.4 | Ki | 2 | — | |
ZZWUEOYQVWAKCJ
|
8.4 | IC50 | 9 | — |