Target Details
UniProt ACP32297
Gene SymbolCHRNA3
Protein NameNeuronal acetylcholine receptor subunit alpha-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 506
  • Clinical molecules 0
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (506)
InChIKey pChEMBL Type Targets Clinical
QYIIVMFJYKZTIQ 9.9 Ki 4
XUMSFYBHKWTENQ 9.8 Ki 2
BKXZRLFPGYWHTM 9.8 IC50 7
JEYWCUOEFNZIIU 9.8 Ki 4
FEXJEKNXTSHUSJ 9.7 Ki 2
RFLDYHWWEJNDMO 9.7 Ki 4
NLPRAJRHRHZCQQ 9.7 Ki 7
KAJDVWZFXDCPSN 9.6 Ki 2
GUBZKNSUJVFLNU 9.6 IC50 3
NLPRAJRHRHZCQQ 9.6 Ki 7
AGSIVKJWYGTAIM 9.6 IC50 3
URCPIVZAKGXXGX 9.5 IC50 5
JLHNNIALZUDMPM 9.5 IC50 4
NBNDFLJNAYAZMD 9.4 IC50 4
WXTQMACZCSXJTB 9.4 Ki 4
ORNGHPVNFVLRNV 9.4 Ki 4
WONBUILDJNKYCB 9.4 Ki 5
KGLAXECQSDAPBR 9.4 IC50 3
AKHCKCPDLAYHDW 9.3 IC50 4
QAEMLNYVRDMVAV 9.3 IC50 3
JYBXLCIZWPNCMU 9.3 IC50 11
VPTXDMQKJHWYPV 9.3 IC50 4
PGTPXIBBHIHMQS 9.2 IC50 10
QYFZGNQKVGYCKF 9.2 IC50 4
VBQDZZHUUPHQGQ 9.2 IC50 11
ABPSWEJOHYDZDP 9.2 IC50 11
HCVVQYDWEUQYOH 9.2 IC50 4
MYNNHDMKXARIMJ 9.2 Ki 2
GDSORCYTZJIZHU 9.2 Ki 4
PREYWAJYVTVVPE 9.2 IC50 10
LPYOFVQCAYSFSJ 9.1 IC50 6
YPROVAPWLFJEAL 9.1 Ki 2
CDPZCHYPADBVMB 9.1 Ki 2
DZHHVCPMWMWVDW 9.1 Ki 2
LJIJFOCTKOLRPU 9.1 Ki 4
AZKMTKVSVYHHAA 9.0 IC50 4
VYJRBHHHDMICNS 9.0 IC50 4
DQKGYJNWJXXUPR 9.0 Ki 2
FVFPYWYYJOGROX 9.0 IC50 4
LKOFWOBOOSHEEE 9.0 Ki 2
BGMUZBOFMKWKCS 9.0 IC50 5
MQVIMBLKNBRZEH 9.0 Ki 2
FOBOXOHWDKQRAH 9.0 IC50 4
UCMCIMRDJCGRNT 9.0 IC50 4
WYGBFIPJEFIRLV 9.0 IC50 3
BJLKZFUZNNATGZ 8.9 IC50 7
XAJIUQJGEWGZBC 8.9 Ki 2
HXZFPBBYBMMKAQ 8.9 Ki 2
PHXYNFXNEHTNMS 8.9 Ki 2
GIDJZDYNVHMFAH 8.9 IC50 9
2D structure