Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
KUNGBRWETVSHKU 7.8 IC50 2
QTGLDSNZORTQEK 7.8 IC50 4
TYFFXNLNRYRUAU 7.8 IC50 3
XVPBPJWOKGRCPR 7.8 Ki 3
BAEZCMHLDJIEPF 7.8 IC50 2
FPYYFGFPTJRMBR 7.8 IC50 4
NSMUITYTUDRYSP 7.8 Ki 3
XJIWJTAALOWWFJ 7.8 IC50 3
CETOWTIWZXCWLA 7.8 IC50 3
HTSRDLNRKNCSLJ 7.8 Ki 3
UYOAPGITMAMCFT 7.8 IC50 4
JNEKRCCXHUFBPL 7.7 IC50 2
KZXNIFOXWZLCOK 7.7 IC50 4
SPSOCPFYUPNNCP 7.7 Ki 3
BXJJBQWOZVLBPK 7.7 IC50 3
JKCHNCUBXBYAJL 7.7 Ki 2
SCWYPKQWJXXMFD 7.7 Ki 3
GSOVKXCTSWIFEY 7.7 Ki 2
HYWBNHIBZICAAO 7.7 Ki 2
JKPCTIHGIAFIKV 7.7 IC50 2
NIGXYCDFYWYVQS 7.7 Ki 2
OHFMRHZLQMSCRN 7.7 IC50 4
UQYKJLAPTINKFZ 7.7 IC50 2
XANHKAKFNIWYOE 7.7 IC50 4
YXIBEMYOGWJEQC 7.7 Ki 4
FFHBJDQSGDNCIV 7.7 Ki 4
GRAFEEBFOIOLGS 7.7 Ki 3
OJPUSZQXDWHXOL 7.7 Ki 3
YPMWOWLUDWNQOB 7.7 Ki 3
DEKJJIFFJPAHRM 7.7 IC50 2
PHHQWWPLQKXGDH 7.7 Ki 4
SMAWMSUKCNWJNR 7.7 Ki 3
FISNMOAZOFAUNZ 7.7 IC50 3
XHASNPJPTJYEPD 7.7 IC50 3
AODONYDDQNDROG 7.6 IC50 2
KHUSEOUYELGLMC 7.6 IC50 2
WHNFPRLDDSXQCL 7.6 Ki 4
WVDXXZITSATFRU 7.6 IC50 2
KNWLOSLCTAQNSO 7.6 Ki 4
UVJBRYNBZSRMBZ 7.6 Ki 4
GEDCOLLODBJRNS 7.6 Ki 2
NUALMFMLNXDIHK 7.6 Ki 2
TXSUTEHZKIBGJG 7.6 Ki 3
BOAIJXQJMLWMSF 7.5 Ki 3
GVPVGDSXVWSVRJ 7.5 Ki 2
HQPISMGZXLHBTG 7.5 IC50 2
KXPKJVIQPPHENQ 7.5 Ki 2
PUBNSQFRKLLQSF 7.5 Ki 2
QVAVMOYDEXISTD 7.5 IC50 2
SYIWIZYUJLMOJX 7.5 IC50 3
2D structure