Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
GBTCAHLJDYHAKJ 8.0 Ki 3
NBQIAPVXQDUVTH 8.0 IC50 3
OEGHHWSPXMTMEY 8.0 Ki 3
QECOLCQUUXFPQQ 8.0 Ki 2
TXGKEAHPJFCNKT 8.0 Ki 2
UICVQJGBBAMKDX 8.0 Ki 4
VXVQZXYFPLAEJW 8.0 Ki 3
XGLWBUKNYXLAFF 8.0 Ki 2
YAVZBTAEIGLTOG 8.0 Ki 3
NSFFFSYEDFVOOT 8.0 Ki 2
AVSQFQRBSIWIJE 8.0 Ki 2
BGNHNMCZDLGXJG 8.0 IC50 3
DPPBMHXXQRAKPB 8.0 Ki 4
DUSMRMPLECSLRG 8.0 Ki 3
IVOZSKOYXPHCOQ 8.0 IC50 2
JSSBJZNAQLSMID 8.0 Ki 2
KXJHWAIMDKIUMK 8.0 Ki 2
NCLQWDCIPKHQBS 8.0 IC50 2
OECQYHIMZCIJFT 8.0 Ki 2
WETYFBSRFBUFCI 8.0 IC50 3
XAHOMYQYMFNUJP 8.0 Ki 2
KHUSEOUYELGLMC 7.9 Ki 2
AVXIGOUSBQQJBP 7.9 Ki 2
IVOZSKOYXPHCOQ 7.9 IC50 2
RQHOEQDAYOKRHG 7.9 Ki 3
FLYJFSWZKPJYBP 7.9 IC50 2
FVGGQGIVDDOMKK 7.9 Ki 2
CMKWAAKJKOZNBH 7.9 Ki 4
BOAIJXQJMLWMSF 7.9 Ki 3
KMNARKQYUZICHM 7.9 IC50 3
RETXHZDMGJHDNV 7.9 Ki 3
VJHTXZAEBALHDW 7.9 IC50 3
XTGXCCGBTWVVAZ 7.9 Ki 3
YUWKIIAXKBDHDF 7.9 Ki 2
ZKTNTRAJYNNFHC 7.9 Ki 3
AZYKYQHQEWLRAS 7.9 IC50 3
KSMXNEYOFKPWFI 7.9 Ki 4
PWVUYOZSIWYFJW 7.9 Ki 4
NMMRTJBOGUWCEQ 7.9 Ki 4
HQACQGVVMYJUAG 7.8 Ki 3
KHTORJRLHSSEND 7.8 IC50 2
SPKUFMODEUMWTR 7.8 Ki 2
VTKKYXSRNMKYHV 7.8 Ki 3
WOWDZBDFXRWMIV 7.8 Ki 3
HJMAXNXTRYYRCZ 7.8 Ki 4
ISVIJWUBKQJSNC 7.8 Ki 2
JVZABOZWHGLGBV 7.8 Ki 2
VWCDOUQYWQELEV 7.8 Ki 2
JMZSDACYKDRROH 7.8 IC50 2
KHTORJRLHSSEND 7.8 IC50 3
2D structure