Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
HLCHESOMJVGDSJ 8.2 Ki 4
OFHSVORZHRSITE 8.2 IC50 2
SOCBNUUFEBTEOP 8.2 IC50 3
UDIAMBWWCWFAJW 8.2 IC50 3
OUFAADNZNCCMJZ 8.2 Ki 4
BACKPKKWDGBCRT 8.2 Ki 3
DCOSVJTYYUGOGC 8.2 Ki 2
DNYQDGRNDXYRDY 8.2 Ki 2
GVUXGBSAZGMQMX 8.2 Ki 2
MSXFGNGAAAPRSR 8.2 Ki 3
QHXULIILOQCKTQ 8.2 IC50 3
WBDPEYKQRJEOEW 8.2 Ki 2
XRFUQRXQTHWOJG 8.2 Ki 2
AODONYDDQNDROG 8.1 IC50 2
CHNMWUKSZIMHIX 8.1 Ki 3
ASZHCTOSSULQLD 8.1 IC50 3
HHHGGOMKUAYOJZ 8.1 Ki 3
HLCHESOMJVGDSJ 8.1 Ki 2
VTYFXSGVWVZOFL 8.1 Ki 3
LDCYRYGDVBLWLI 8.1 IC50 2
MCJFEKJJFCZAHM 8.1 Ki 3
PNFDTYPRKXTXAO 8.1 IC50 2
WFOFJUYRBUEJBI 8.1 IC50 2
ARFBDECCXOFCBN 8.1 IC50 3
FFAUSQSMDWHWML 8.1 Ki 2
HJSDVHQHZYTQEH 8.1 Ki 2
ITVFKSXIFRKUOS 8.1 Ki 2
KPAXZSMXFNRRAR 8.1 IC50 3
OGIIVLJDBHLNNQ 8.1 Ki 2
PQOAIQOLRRUAHF 8.1 Ki 2
QAXKNGODUAVCKD 8.1 Ki 4
VBLQHXVKCWZWRQ 8.1 Ki 2
ZLLOVWBBACAVIV 8.1 Ki 3
APHPBWUTFHDTLW 8.1 Ki 4
HXKRGRRDOBSQCO 8.1 IC50 3
XLLJFSCSXTYVTN 8.1 Ki 4
AWDCZSOETVHKLV 8.1 Ki 2
HNVXASMBDVOKKN 8.1 IC50 3
ROTHBSFMHAHRTG 8.1 IC50 4
DBZMYFPVMVRJJO 8.1 Ki 2
RDQOUEKWQGRDRJ 8.1 Ki 3
UEQVXEFRAIHLCM 8.1 IC50 3
UIMWAMYMWYXGRV 8.1 Ki 2
KYLMYZLCQJJVMF 8.0 IC50 4
YBWGYSWBATYFBD 8.0 IC50 4
NDRYSEKKAUQGGO 8.0 IC50 3
AMLJFTMENZUCBN 8.0 Ki 3
FRHBHVROLQSPMW 8.0 IC50 4
HSIYJWUPHNPTOY 8.0 Ki 2
DLPKFLGDHWMYLD 8.0 IC50 2
2D structure