Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
JICSVJQEGDFDBH 8.3 Ki 3
KOMGNGDDTPNSKC 8.3 Ki 3
KOWZSZLHPBJHEB 8.3 Ki 3
PZVZJDCUPVOTTP 8.3 IC50 4
RLQHLELPSPEDPJ 8.3 Ki 2
RVEIEULWMVBMRD 8.3 IC50 4
SLZKONAGMRVCMC 8.3 Ki 2
STSKLVUCFFVQGJ 8.3 Ki 2
SUYDUGVDUFCDHQ 8.3 Ki 3
XFRXFJPUAKFDHC 8.3 Ki 2
ZQDYFCAQLYEQJM 8.3 IC50 2
CJCOTNMGGCNQIS 8.3 IC50 3
DZBWWVGXDVRUHV 8.3 Ki 3
QMJPEHNJEMTEMH 8.3 Ki 3
SJRCSWXLNHDZIX 8.3 Ki 3
XQMPAWYRHAOJTE 8.3 Ki 4
QKGLIQPAOWFWIE 8.3 IC50 3
BWVHAZIIKXCXDT 8.3 IC50 3
SYYCZXDFWBANLC 8.3 Ki 3
HEILVIDOVAHKRM 8.2 Ki 2
JHQJUSRZOBDPMK 8.2 Ki 3
KFZNXVCUWNNJMQ 8.2 Ki 3
UMHVNRYGRKBTCG 8.2 IC50 4
WSDYWWDQJYPQDS 8.2 IC50 4
YDQIBTSSHWCIEQ 8.2 Ki 3
AHYGIWNTGDKMRR 8.2 Ki 3
AIVKUJJDLDHLNN 8.2 Ki 3
ARFBDECCXOFCBN 8.2 IC50 2
AWKJUBFDTQDCHX 8.2 Ki 2
DLLIKIKBBRMHTJ 8.2 Ki 2
FHNLUGMXKXPEFR 8.2 IC50 4
HYNXKHHGAXLIEQ 8.2 Ki 3
NVXVBSBXBTZZNU 8.2 Ki 3
OKHXBJLIBJDJMV 8.2 IC50 4
RZFOKMNOCAQLCI 8.2 Ki 2
SUYDUGVDUFCDHQ 8.2 Ki 3
WUDKHRNOVXFNLO 8.2 Ki 2
YWRRNKAZKAJGFT 8.2 Ki 2
AGENZPFZMBQUPS 8.2 Ki 2
CFAHIOAXVOKBCK 8.2 IC50 3
HDBFFTYMERRCIX 8.2 IC50 3
LKGYQUQHVGIHMG 8.2 IC50 3
PWADIMGJQZHREF 8.2 IC50 2
UWUFZBBTPNPUEY 8.2 IC50 3
RUDWSQPLBXOLBE 8.2 IC50 3
UBWLAYRWNUNYHG 8.2 IC50 4
YOJWKJVHBTUFST 8.2 IC50 3
HAYIRZKTTMIXAL 8.2 Ki 2
NKVAOVHVGQNSIX 8.2 Ki 2
OFNOTFBPXMBPPC 8.2 Ki 2
2D structure