Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
TUEXZDIGHDGDGO 8.5 IC50 3
YMEXHIACKAXZLZ 8.5 IC50 3
UVUOMESIOOEXGA 8.4 IC50 3
HNVXASMBDVOKKN 8.4 IC50 2
ALUGMAFCICEWDO 8.4 IC50 3
BKDGLTMSFYSIAO 8.4 Ki 3
FSTDLRINZOKGRA 8.4 Ki 3
HIGBPTITEJOMDX 8.4 Ki 2
LQZTUMSSNFZEFV 8.4 Ki 2
MIAUOPQGTJQSKK 8.4 IC50 2
MMBHRGOCQSTXRS 8.4 Ki 2
MWOCTFMMKHRPCY 8.4 IC50 2
NSBYFZXDVSHNEF 8.4 Ki 3
NTMXDNFEFWCVSA 8.4 IC50 3
OLKZRPFXLZQEOU 8.4 Ki 2
REGPMQLCJMICLA 8.4 Ki 2
RNCVEEUMKRRHLC 8.4 IC50 4
SOCBNUUFEBTEOP 8.4 IC50 3
UKMQKNTZNHDSPD 8.4 IC50 4
WMMWJBFBADMJIK 8.4 Ki 3
XMQSVPKHHVWBGS 8.4 IC50 4
MIAUOPQGTJQSKK 8.4 IC50 2
HDHDTKMUACZDAA 8.4 Ki 3
SDXNKLFMLKIOBP 8.4 Ki 2
OBNLGUMWGVRYJW 8.4 IC50 3
OQIKSFAMWBMLCU 8.4 Ki 3
RQZHKEFEFWSLOK 8.4 Ki 3
CGANDSYNDFLFKG 8.4 IC50 4
DIWJBUBBVDFSOS 8.4 IC50 3
DQDUAZXNONBSMT 8.4 Ki 3
GUUMVPUVSBGKBI 8.3 IC50 3
JTEJZABLGYDSAQ 8.3 IC50 3
VOVCAFWIQXNUIB 8.3 Ki 2
YXPCHDOWVWAKKP 8.3 Ki 3
AMDDROJLTSPHMK 8.3 Ki 2
LDHOENQCWMSQTE 8.3 IC50 3
LMTCYYTZYVZVDJ 8.3 Ki 4
MTHZQNMVJGFKRT 8.3 Ki 2
ZQDYFCAQLYEQJM 8.3 IC50 3
BBYTXRAQNPWSMC 8.3 IC50 3
IVOZSKOYXPHCOQ 8.3 IC50 3
LNVJOUMPGCMIDQ 8.3 IC50 3
QOZPHXSKYHWXNY 8.3 IC50 4
AUPOJQYWSLXSAP 8.3 Ki 3
CZCIDYFBUVIGBB 8.3 IC50 3
DEMSFZJYAYNEHZ 8.3 Ki 3
DIWJBUBBVDFSOS 8.3 IC50 3
DPQPIDRPGTZJFK 8.3 Ki 2
FLJXXBKEOMUWAG 8.3 Ki 2
GTMASPVXPKDKOK 8.3 Ki 3
2D structure