Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
KKBPPVVSQKSKNV 8.7 Ki 3
MRFZKAWUCKFKJV 8.7 IC50 3
CXGYZUHRSDOJIS 8.7 Ki 2
AWOIGQXOOIHLJT 8.7 Ki 2
BCFFSQJVHOEAAU 8.7 IC50 3
HSMWDLAIQGCRBD 8.7 Ki 3
LDKZCTCDXVIBCI 8.7 Ki 2
SHUMMQAOTPBZAQ 8.7 Ki 2
SSOJHWGDEMWTNO 8.7 Ki 2
VVNAQHKXBHSZIX 8.7 IC50 3
WMIJFYRFKZUVFF 8.7 Ki 2
ZSRGOYOFHLLWGA 8.7 Ki 2
RXVHNQJRLPWMJA 8.7 Ki 2
WRXWCWIFEFKMJL 8.7 IC50 3
KLOVFBFHFHKKJQ 8.7 IC50 3
KRZXMSMNMZEKGP 8.7 Ki 4
JKJKHYOUTNOITO 8.7 IC50 3
PIHBUAVCWXDWIB 8.7 Ki 3
DCRRHKOGXQUJTJ 8.6 Ki 3
KWBYYFKCXHSTPA 8.6 IC50 4
XATASKINOVYSLA 8.6 IC50 3
DHGVVSQOBPUMLY 8.6 Ki 3
GGYWLZFXFKFWKL 8.6 IC50 4
PPKCWGLTAGNYCP 8.6 Ki 2
OODHJMPCOPKKSM 8.6 Ki 3
REMHNXQVRVXAGT 8.6 IC50 4
UKCAJRRGLXHDRO 8.6 Ki 3
WOSXQRHNBLCZBB 8.6 IC50 2
DPJAKAHREXIEPH 8.6 IC50 3
VRGPMQNQBPODPZ 8.6 Ki 2
YITJJGWDWIIORX 8.5 Ki 3
HOWXKXAJVJPQOI 8.5 IC50 3
CDHOQEHTFUNKKJ 8.5 Ki 3
JWBGVBLXXIKBCO 8.5 Ki 2
KLOVFBFHFHKKJQ 8.5 IC50 3
QECBRZQFCKLWKS 8.5 Ki 2
ROTIMMRQYLIORG 8.5 Ki 2
UCISBBYZNLQVGP 8.5 Ki 2
VVUGZLZXEFCSGI 8.5 Ki 2
XTNWQOXFVSNCOT 8.5 IC50 2
YPCZQXKWTSFFSU 8.5 Ki 2
ZSWPGAPVLVMTJG 8.5 Ki 2
KDEFFRZENHEKTD 8.5 Ki 4
KPFZSXDUVZTNAQ 8.5 IC50 3
AZYLFDYQQJPDQC 8.5 IC50 2
DADQHECQKQBHAW 8.5 Ki 3
GGYWLZFXFKFWKL 8.5 IC50 3
MZFOEDJULWOZIV 8.5 IC50 3
GFIRCBLJLBAPRI 8.5 IC50 3
OLLQZYNQBYGVCQ 8.5 IC50 3
2D structure