Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
MTFOEQYGYVFQPJ 9.1 Ki 3
WZIILWAZGXRRFZ 9.1 IC50 4
AUTMNYLYUILQAZ 9.0 Ki 2
DTYOAGHBUMBHBH 9.0 IC50 3
RANDNDRFMFBRFD 9.0 Ki 3
UHXVSCQTWQLUSR 9.0 IC50 2
ZTSQVRSYAGAZPG 9.0 IC50 4
RDLAZLIJEHHWIX 9.0 Ki 2
SXYITQIOONIMPP 9.0 Ki 2
UNUGBHUNONVSEZ 9.0 Ki 2
ILTSJNSAHXKVSQ 9.0 Ki 3
IVRFZQRHPFZUMZ 9.0 Ki 4
VVTLPZHJHVZUSC 9.0 Ki 2
WOQVIKOQMYEYTM 9.0 Ki 2
ZZZCDEAVWIKQBQ 9.0 Ki 2
JDKLPDJLXHXHNV 9.0 IC50 4
NMZQXNVSJCWFFD 9.0 IC50 4
ORPYCWJPNJKZIA 9.0 IC50 4
ZPANOUCVWZTSLE 9.0 IC50 4
ZRHYLFBORVIBEU 9.0 Ki 3
LBOGVWLKUREGLH 8.9 IC50 2
TXXMJHUJXUWXNR 8.9 IC50 2
QBYHLGIJWBFDGJ 8.9 IC50 4
QXRXXIKAVZAGHZ 8.9 IC50 3
RVKSMTBVJXMWFD 8.9 IC50 4
ASUAOIWGQADQOH 8.9 Ki 3
MTFOEQYGYVFQPJ 8.9 Ki 3
BZEWEHPSOMSRJV 8.9 Ki 3
CZCIDYFBUVIGBB 8.9 IC50 3
GUUMVPUVSBGKBI 8.9 IC50 3
JAOFTGJUMOHSQY 8.9 Ki 2
YZQBDVJPOXNSJR 8.9 Ki 3
FDLHDUZIGJCBAK 8.9 IC50 3
SLPDXDVCXNVEEV 8.9 Ki 2
DBDVRJVEKWLHPY 8.8 Ki 3
JKJSJPHXCRZLKD 8.8 Ki 2
MGPPGHOYFKVPCB 8.8 IC50 2
XJIWJTAALOWWFJ 8.8 Ki 3
ZYJYAZJJQYYWKW 8.8 Ki 3
YLVUKTHOPXMSDE 8.8 IC50 2
GSECRIQNUWHRKM 8.8 Ki 3
RBKDACLJKAMLFN 8.8 IC50 3
RBZTXCPXQHRLIB 8.8 Ki 3
REMHNXQVRVXAGT 8.8 IC50 4
VFJOTTZGMDRNPT 8.8 Ki 3
VESJJEZSWHFEGA 8.8 Ki 3
HVLGSWMYZPWZTD 8.8 IC50 2
FDPBRBMLLVILMV 8.8 Ki 3
VITHTUWCONJLQU 8.8 Ki 3
GGYWLZFXFKFWKL 8.7 IC50 3
2D structure