Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
KHGZKFBKKYRZCD 9.3 IC50 3
AFDFLEMNTOCMSC 9.3 Ki 2
GDRJSPPVRGELGB 9.3 Ki 3
RHDRZFXISWDZNM 9.3 Ki 3
FDLHDUZIGJCBAK 9.3 IC50 3
RVVLJWZWXHPMLS 9.3 IC50 4
RXAACDRLBPKKHH 9.3 IC50 3
SVNSNKFQLBXSEH 9.3 Ki 3
XATASKINOVYSLA 9.3 IC50 3
GJFLVESIDOAAJH 9.3 IC50 2
PPKIGEMCDOLKEY 9.3 Ki 3
PPKIGEMCDOLKEY 9.3 Ki 3
UNXFCHHFXJFRRB 9.3 Ki 3
VPORMYBONMHESW 9.3 Ki 2
ZSONGANRJTVTCP 9.3 Ki 4
XLDGDUSCVKLZIR 9.2 IC50 4
BGQGGVJRXUWNNU 9.2 Ki 3
XFQWSJOXRAVFGY 9.2 Ki 3
XUCSIJVANOTEDW 9.2 Ki 3
FWYIDGAEHPOSEJ 9.2 Ki 2
GGYWLZFXFKFWKL 9.2 IC50 4
KYOVLZCJSUXUJI 9.2 Ki 3
OBKWMOSDTIUARN 9.2 Ki 2
SVSUFMZEUZIVDX 9.2 Ki 2
UMHVNRYGRKBTCG 9.2 IC50 4
ZSAXEKUGMLDFHT 9.2 Ki 3
UHMCIGUGJPINOI 9.2 IC50 3
UCFQPBRLCMKTJY 9.2 Ki 2
LEURJYAAAHRVRF 9.2 Ki 2
NVIBFTUPAARCBA 9.2 IC50 3
AKHYEKNKKQDKLB 9.1 IC50 2
UAHFGYDRQSXQEB 9.1 IC50 5
DLOGSFRUKCUWHC 9.1 Ki 2
WSDYWWDQJYPQDS 9.1 Ki 3
ZSRGOYOFHLLWGA 9.1 Ki 2
AETQUGIIFBPWMW 9.1 Ki 2
AOMUTEUZPCRNFD 9.1 Ki 3
FEKXKTLLBDRSQH 9.1 Ki 3
IFDBWKFSUPQKCA 9.1 IC50 4
SZGSXARYIZZWDD 9.1 IC50 3
AEZCRBIFPKXUGD 9.1 Ki 3
FJSKRKLUQFIKJP 9.1 Ki 3
JOWUFLPXVQKTNW 9.1 Ki 3
UCOANIAEMBZDQE 9.1 IC50 2
YHYBBOPOIUAVHY 9.1 IC50 3
UAHFGYDRQSXQEB 9.1 Ki 3
DYRPZKYWKBUEOV 9.1 IC50 2
WRKBOTGDFLBBDK 9.1 Ki 2
QVLFTJGCGVDBFK 9.1 Ki 3
HAIHKNYZIMVIIW 9.1 Ki 3
2D structure