Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
PYANSLUAUZKUFT 6.7 Ki 2
UAISFSHHKXHKOI 6.7 IC50 4
CVFGCUVAZVPTRO 6.7 IC50 2
VDEUVZJQPRWULE 6.7 Ki 3
JKPIUTPQBDXSRH 6.7 Ki 3
MNSNXOUQPSOGHN 6.7 IC50 3
HJEMTEIBBSGTRL 6.7 Ki 2
BLUHVPTUPSCCBC 6.6 IC50 2
OJPUSZQXDWHXOL 6.6 Ki 3
YPMWOWLUDWNQOB 6.6 Ki 3
APASEPBZJFOHSF 6.6 IC50 2
QIKIYIZHGOCQOO 6.6 Ki 3
TVINVHGLLFLSBP 6.6 IC50 4
ZZVLKHHSRQKCEV 6.6 IC50 4 Yes
ZZWLTZIHMIAAFS 6.6 Ki 2
FYBQSBASELLFTJ 6.6 Ki 2
CAPRWXCJSDCJMN 6.6 Ki 2
DFCJPPDAOZROBS 6.6 Ki 3
MXAUIAYYRYRHPY 6.6 Ki 2
QCXXYYAQEUNASC 6.6 Ki 3
VILSSUAARNTCPC 6.6 IC50 3
NEVVXMYOTHZJES 6.6 IC50 3
OVCXMKITXFVUSL 6.6 IC50 3
PKHOEKKVDQTOOR 6.6 Ki 2
VNTJATGNGDRIFN 6.6 IC50 2
NEVVXMYOTHZJES 6.5 IC50 3
UNGLYFOZRWHRKE 6.5 Ki 2
MLXMTZDTPIINBF 6.5 Ki 2
MWUXCBIVLGSGOO 6.5 Ki 2
KDTZLQMUHBEBMZ 6.5 IC50 3
PNUQGRIALHGKEH 6.5 Ki 3
UHAQQQFLDCOOEA 6.5 Ki 2
ZPOQUKYSTRZAFA 6.5 Ki 2
JHIRSHLLKDOJGA 6.5 Ki 2
PBHKXVJFSKYMRO 6.5 Ki 2
ZWTUZOQCWSYYNO 6.5 IC50 3
DVRRTOIJYURKKI 6.5 Ki 2
OYRRSSXMTFYBBG 6.5 Ki 2
YUUZCRILYWDWPO 6.5 IC50 3
BZFJGKHIEZMTSV 6.5 Ki 2
KWPBFXVTEVUNPD 6.5 IC50 4
SGKSNHUSKUVYHG 6.5 Ki 2
SGKSNHUSKUVYHG 6.5 Ki 2
SOPYHFQNBMKJEU 6.5 Ki 3
YJCDHAJJLSUBDS 6.5 IC50 4
CADNRYGCBMLNJN 6.5 Ki 3
DFCJPPDAOZROBS 6.5 IC50 4
KPDWCDURFGPKLY 6.5 Ki 2
JUOGFOXGQYCMTJ 6.4 Ki 2
SFGAMHAXMGIWOF 6.4 IC50 3
2D structure