Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
AIBOPTDBFGOAQA 6.9 Ki 2
FZMMHTRNAWCOMM 6.9 Ki 3
MTINEKLBSHMHSP 6.9 Ki 2
QALQZIUEBLVALT 6.9 IC50 2
RZLPZBLBQNNVLZ 6.9 IC50 2
KRZXMSMNMZEKGP 6.9 Ki 3
NMXSKMOZDYUBHU 6.9 IC50 2
IXQMIHWLSWEYPU 6.9 IC50 4
XMCIIUVWOCNDSA 6.9 IC50 2
VGBVAARMQYYITG 6.9 Ki 3
CQUKLRIOLMQYDE 6.9 IC50 4
AEBQLEXRXNCRKU 6.9 Ki 3
CRLGCHNGOJRZNC 6.9 Ki 3
DZEMZHXEKMDTDY 6.9 Ki 2
MMJANTAPAJRPCT 6.9 Ki 3
CZLALGVBUDRCJM 6.8 Ki 3
KBBHXCZBVZTXQH 6.8 Ki 2
LVACOVVOTCZAIW 6.8 IC50 2
LVACOVVOTCZAIW 6.8 IC50 2
NAEZHDBXDQXCIQ 6.8 Ki 3
AHRZYQWKXXBNHK 6.8 IC50 4 Yes
CHNMWUKSZIMHIX 6.8 Ki 3
GJRWWAJUJBKGQU 6.8 IC50 2
GKWBRFGCZAYVJV 6.8 IC50 2
HIYNTZOLQGBWSI 6.8 IC50 2
HIYNTZOLQGBWSI 6.8 IC50 2
PJDCKQFLLOIVHJ 6.8 Ki 3
RLWOSGQNOKLOKP 6.8 Ki 3
TVINVHGLLFLSBP 6.8 IC50 4 Yes
VNKGTZHAAMHYKK 6.8 Ki 3
XCXOPMSFLOPCFL 6.8 Ki 3
YUKODIVVRQEHLF 6.8 IC50 3
CAXNNMYXBQZZIP 6.8 Ki 2
WBTHAPYEEKFPSX 6.8 Ki 4
IGSPGKUFVFMXQE 6.8 Ki 2
JWVUTJWCWBNVDW 6.8 IC50 3
PRCMOLNMVBSDRO 6.8 Ki 3
ULKFOTUQRDIPQX 6.8 Ki 4
VKDMHINLWUJYEZ 6.8 IC50 3
NHBSWHPBPMPVCZ 6.8 IC50 2
GVZTZLFKKLVBJF 6.7 IC50 3
OVIZBCMXCJAPHP 6.7 Ki 3
YBCXRFXRMKTZQS 6.7 Ki 2
IENZGWYSQBAEDX 6.7 Ki 3
JQDBJPQYLBLUNL 6.7 Ki 2
MNJTTYMJKZNPFK 6.7 Ki 3
OMSSRUBSGSKAFS 6.7 IC50 3
RSZGGZUMSYSTES 6.7 Ki 3
RSZGGZUMSYSTES 6.7 Ki 3
BVHVEJVRGYHQTC 6.7 IC50 3
2D structure