Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
DTPYMOHNIPTAGK 7.1 Ki 3
FBIBREHNRFMLIZ 7.1 Ki 2
GWQJQMUYAJRYAV 7.1 IC50 2
VSVABBLUDNGFCZ 7.1 Ki 2
WZIILWAZGXRRFZ 7.1 IC50 3
UHCXNXMBPAFWDS 7.1 IC50 3
YVHWYCKBKQBQLH 7.1 IC50 2
CSQOOKHGXFRBEQ 7.1 Ki 2
PGJYWMVUWDKZMU 7.1 IC50 2
DZOXHHUQYQUKJB 7.1 Ki 4
KXWAHHUIDLURNT 7.1 Ki 4
ONUUGLJKQIIBGJ 7.1 IC50 3
SFVVQRJOGUKCEG 7.1 Ki 3
HAIHKNYZIMVIIW 7.1 Ki 3
PEOUPURBSIPXLE 7.1 Ki 3
WIUGVXOSBXINHH 7.0 Ki 3
XJMJZYGMMSEXNX 7.0 Ki 3
KBLNYXZHILRCGF 7.0 Ki 4
OHFHKCOOPQLGKC 7.0 Ki 3
WZIILWAZGXRRFZ 7.0 IC50 2
DYLFBHOZQPVNMC 7.0 Ki 2
OFPOZEFXTIZAHE 7.0 Ki 4
CATZYTHJWOAGOB 7.0 Ki 2
RBLCKVWSBGCRJN 7.0 Ki 2
GBTCAHLJDYHAKJ 7.0 Ki 3
JXWMBIOMMZLSIR 7.0 Ki 2
KKGFKAITEKCBRV 7.0 IC50 2
KRKYTJXTDCSSJS 7.0 IC50 4
LWRUHFMBKCOVAZ 7.0 Ki 3
NYBMXOVCJILSIJ 7.0 Ki 2
RHVBMPAJVRQKPF 7.0 Ki 3
AYKQERUAGGPJLP 7.0 IC50 3
AYRYPORYMTYECQ 7.0 IC50 2
DKHPVUADMFUYGQ 7.0 IC50 2
DOAQTQYFNKQPTO 7.0 IC50 2
LGJDLKCHZMGHIM 7.0 IC50 2
ODSFZEXVNOIJHI 7.0 IC50 3
RQIFYTAAHPOYSP 7.0 Ki 3
UJXZIZJAELMUHW 7.0 Ki 2
VLXDEFRTAJLNNA 7.0 Ki 3
WCVJJQCPIDBNFM 7.0 IC50 4
XNPPTTUWPBNRFQ 7.0 Ki 2
BVTKLQRLIKZFNA 7.0 Ki 2
IARGQFSHIKWWJL 7.0 Ki 2
IJVUOKFOZUYPMK 7.0 Ki 2
UYKWHGIEHONMDL 7.0 IC50 4
ZDRWLGHFJFKMFH 7.0 Ki 3
ZOFPYCCSYGWTCN 7.0 Ki 2
RCULCPVSLOFQPR 6.9 Ki 4
VOCXANHYYBVTET 6.9 Ki 4
2D structure