Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
FEKXKTLLBDRSQH 7.5 Ki 2
IXLVDOBKTIIMBE 7.5 Ki 4
KZZQDCIGVAXNMN 7.5 IC50 3
PVVLKBSYHAGXBD 7.5 Ki 4
AIBOPTDBFGOAQA 7.5 Ki 3
APAIPJOPPUMQFD 7.5 Ki 4
AWZTZSDCMJPFJF 7.5 Ki 3
YCEIOOXEUSAMIZ 7.5 IC50 3 Yes
WLYFDIRUCOZYRB 7.5 IC50 3
FIPGSBWOMGALGM 7.5 Ki 4
IJVUOKFOZUYPMK 7.5 Ki 2
JLMVHMLMBIPZSW 7.5 Ki 4
NUEQNUVEEKTGQM 7.5 IC50 2
YYXKYIYEADPIBB 7.5 Ki 2
LAHUDBCXWRATGM 7.5 IC50 3
PAILFUNFWZLMMN 7.5 IC50 3
ZKFHMXVIVJCDFY 7.5 Ki 4
BUTABXHVJVEFTF 7.5 Ki 3
NOLFWMRTIVNJFP 7.5 Ki 4
QSMNQYOEIKDHHC 7.5 Ki 2
TVCZNUJSXSNMJP 7.5 IC50 3
CQIHYFQHPBTXLQ 7.4 Ki 2
IPSFANQKYGITFT 7.4 IC50 3
NOMHNUFAKKUFFP 7.4 Ki 2
PCKSOAZIMLQBHU 7.4 Ki 4
NHZYDUWLLZYUEJ 7.4 IC50 3
WHNFPRLDDSXQCL 7.4 IC50 4
KCOGRZRTHYZEQU 7.4 Ki 2
SSCJBDJJWLFQLZ 7.4 IC50 3
VJUGSZWVYVMRBR 7.4 IC50 2
HICQRDPLMADMBD 7.4 Ki 4
QEQUHVRIJFFOKD 7.4 IC50 4
WWDUVSWFUPRTGG 7.4 Ki 4
YEUMEJHOKABUMX 7.4 Ki 2
BHDPSUNZDKCRLI 7.3 Ki 2
FEFWDDKHEOVPCG 7.3 IC50 4
FLQGGHIOZAPIQO 7.3 IC50 4
HJERQRDKWIWHPW 7.3 Ki 4
QQVWMYDNTPWWPW 7.3 Ki 2
VOSIMUPSRJWOJN 7.3 Ki 2
DEQSFWKJAFMEST 7.3 Ki 3
IKTNZHMAWQNOLP 7.3 IC50 2
KWTLWMHGSUOSHU 7.3 Ki 4
ROSDSGGMKIYLIM 7.3 IC50 3
SZCLBSHELXLOEC 7.3 Ki 4
YRPCDHHSQYGEDU 7.3 IC50 4
ZTBIYCCYYNUCCA 7.3 Ki 3
IDDVSLRYKLDACE 7.3 Ki 4
IVQPGYKGSXUDKV 7.3 IC50 4
JPRKCJZGKZFHOW 7.3 IC50 3
2D structure