Target Details
UniProt ACP32245
Gene SymbolMC4R
Protein NameMelanocortin receptor 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 771
  • Clinical molecules 6
  • Avg pChEMBL 7.82
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (771)
InChIKey pChEMBL Type Targets Clinical
YIYFGSBFHVAQLI 10.6 Ki 2
JPHOERRRWXXXOC 10.3 Ki 2
VSGQPYQAGHZCFG 10.3 Ki 2
GGYWLZFXFKFWKL 10.2 Ki 3
SSZDAFBCWHVROA 10.2 Ki 3
WPNVZVWZWSOGOI 10.1 Ki 2
XPWIQGFRIVVHRC 10.1 Ki 4
JNEKRCCXHUFBPL 10.1 IC50 3
JMFDAPXKXHNPIL 10.0 Ki 3
UCISBBYZNLQVGP 10.0 Ki 2
CDHOQEHTFUNKKJ 10.0 Ki 3
SNEMRJZDOOLWPZ 10.0 Ki 4
XTFWFFODDNNYFQ 9.9 Ki 4
JMNUTDPHHUFMOG 9.9 Ki 4
KIFNALNSUOJQPJ 9.8 Ki 4
XQQIIPUPHPWBDF 9.8 Ki 3
CSIVLBODDQFIPR 9.8 Ki 2
YBKZXQIAHZXKIW 9.8 Ki 3
KHGZKFBKKYRZCD 9.8 IC50 3
GVLRCXVPKHTHFV 9.8 Ki 3
JGBGNKDRAKSUHZ 9.8 Ki 4
LKIXKBAXFLOUEW 9.8 Ki 4
QXDWLOZJHHTTCF 9.7 IC50 3
NVIBFTUPAARCBA 9.7 Kd 2
QBPUPEUBMHTUDK 9.7 Ki 3
JNEKRCCXHUFBPL 9.7 IC50 3
KYIGOCCCBXRHNJ 9.7 IC50 43
QXDWLOZJHHTTCF 9.6 IC50 3
QDKRFZOIHJPTRE 9.6 Ki 3
CNWHTMNTHKVVEV 9.6 Ki 2
UWUHDNLMNSCQPX 9.6 Ki 2
VPWMVGOTLXHAFL 9.6 Ki 2
BEGFBZSFSWOZDK 9.6 Ki 4
UTARRQKZBUCQBR 9.6 Ki 3
XDLJELQQEILLFZ 9.6 Ki 4
CHBTZNAADZTZLP 9.6 Ki 4
KYRVGEKZJIYJKZ 9.6 Ki 3
ANTVHWLGFDSXEN 9.5 Ki 2
LZYYGZAXFMYSBE 9.5 Ki 4
BUVGQEXSQXRZQG 9.5 Ki 4
BINHUIMAVHQSOM 9.5 Ki 4
HGBJQFBJSTUQOF 9.5 Ki 3
BPRBXYIGPSSVII 9.5 Ki 2
FWQGDGPDBUUACD 9.4 Ki 3
IFDBWKFSUPQKCA 9.4 IC50 4
UBKGFMZTCLCOLM 9.4 Ki 4
AXYNQPYLILCAPC 9.4 Ki 3
CBZNNNCTDMTAGU 9.4 Ki 3
RDCIPOBDQMOUKD 9.4 IC50 4
UNXFCHHFXJFRRB 9.4 Ki 3
2D structure