Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BMZYXLWLLWZVBA
|
6.2 | IC50 | 2 | — | |
OZUSVSPHYKYLAS
|
6.2 | IC50 | 2 | Yes | |
CTAHPXXZSACISG
|
6.2 | IC50 | 2 | Yes | |
UUNNSNYSEQPCKO
|
6.2 | Ki | 2 | — | |
ARRVGGQZILZZEJ
|
6.2 | IC50 | 2 | Yes | |
DDUAFEYIPWOELY
|
6.2 | IC50 | 2 | Yes | |
BMWKQHPGKPJLPG
|
6.2 | IC50 | 2 | Yes | |
GFMBISIECXFEJK
|
6.2 | IC50 | 2 | Yes | |
BERNHFOYDVXQGI
|
6.2 | IC50 | 2 | Yes | |
HQDSSVWRHVHJGQ
|
6.1 | Ki | 2 | — | |
NFHRQQKPEBFUJK
|
6.1 | IC50 | 2 | Yes | |
RPNVENCCLVKRAM
|
6.1 | IC50 | 2 | Yes | |
PSNAHSRRFJSWQU
|
6.1 | IC50 | 2 | Yes | |
XYEJNVLBRMQKPD
|
6.1 | IC50 | 2 | — | |
QNCFQRIXQDHLMN
|
6.1 | IC50 | 2 | Yes | |
ZKEBGVDIRJCKNA
|
6.1 | Ki | 2 | — | |
IRUDQSQIPJJXFZ
|
6.1 | IC50 | 2 | Yes | |
SXXOCXCOHMDHPD
|
6.1 | IC50 | 2 | — | |
DOABBONQBBUCRN
|
6.1 | IC50 | 2 | Yes | |
YGVMCMZWGQEBFU
|
6.1 | IC50 | 2 | Yes | |
ACWHYMXOCYJYPG
|
6.1 | IC50 | 2 | Yes | |
LNIOBOYWQUFRMI
|
6.1 | IC50 | 2 | — | |
SPJCSYUKRLKAQT
|
6.1 | IC50 | 2 | Yes | |
DTSANQSRTBGPPK
|
6.1 | IC50 | 2 | Yes | |
DUPJRHKBDSHZPG
|
6.0 | IC50 | 2 | Yes | |
QZFBYNPTVXYUII
|
6.0 | Ki | 2 | — | |
ZOZPVKJSFYNWLP
|
6.0 | IC50 | 2 | Yes | |
VEGZKBKISJJLJC
|
6.0 | IC50 | 3 | Yes | |
YCEIOOXEUSAMIZ
|
6.0 | IC50 | 3 | Yes | |
FNRFRMQWGSYIMM
|
6.0 | IC50 | 2 | — | |
GSIXSVTVZDJDOC
|
6.0 | IC50 | 2 | Yes | |
HMXDWDSNPRNUKI
|
6.0 | Ki | 72 | — | |
IEAOMUBPJVXBAO
|
6.0 | IC50 | 2 | Yes | |
LGYKPDHARJMLQN
|
6.0 | IC50 | 2 | — | |
OIVTVLWHNZZBJN
|
6.0 | IC50 | 2 | Yes | |
QPEUEORJEDJUHX
|
6.0 | IC50 | 2 | — | |
RRZKRPHYMGDLBB
|
6.0 | IC50 | 2 | Yes | |
TXSXJYRAIUVBDO
|
6.0 | IC50 | 2 | Yes | |
XLWHWNHGNRPPBH
|
6.0 | Ki | 2 | Yes | |
XLWHWNHGNRPPBH
|
6.0 | Ki | 2 | Yes | |
YJMMQRORYCUFDF
|
6.0 | IC50 | 2 | Yes |