Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
BMZYXLWLLWZVBA 6.2 IC50 2
OZUSVSPHYKYLAS 6.2 IC50 2 Yes
CTAHPXXZSACISG 6.2 IC50 2 Yes
UUNNSNYSEQPCKO 6.2 Ki 2
ARRVGGQZILZZEJ 6.2 IC50 2 Yes
DDUAFEYIPWOELY 6.2 IC50 2 Yes
BMWKQHPGKPJLPG 6.2 IC50 2 Yes
GFMBISIECXFEJK 6.2 IC50 2 Yes
BERNHFOYDVXQGI 6.2 IC50 2 Yes
HQDSSVWRHVHJGQ 6.1 Ki 2
NFHRQQKPEBFUJK 6.1 IC50 2 Yes
RPNVENCCLVKRAM 6.1 IC50 2 Yes
PSNAHSRRFJSWQU 6.1 IC50 2 Yes
XYEJNVLBRMQKPD 6.1 IC50 2
QNCFQRIXQDHLMN 6.1 IC50 2 Yes
ZKEBGVDIRJCKNA 6.1 Ki 2
IRUDQSQIPJJXFZ 6.1 IC50 2 Yes
SXXOCXCOHMDHPD 6.1 IC50 2
DOABBONQBBUCRN 6.1 IC50 2 Yes
YGVMCMZWGQEBFU 6.1 IC50 2 Yes
ACWHYMXOCYJYPG 6.1 IC50 2 Yes
LNIOBOYWQUFRMI 6.1 IC50 2
SPJCSYUKRLKAQT 6.1 IC50 2 Yes
DTSANQSRTBGPPK 6.1 IC50 2 Yes
DUPJRHKBDSHZPG 6.0 IC50 2 Yes
QZFBYNPTVXYUII 6.0 Ki 2
ZOZPVKJSFYNWLP 6.0 IC50 2 Yes
VEGZKBKISJJLJC 6.0 IC50 3 Yes
YCEIOOXEUSAMIZ 6.0 IC50 3 Yes
FNRFRMQWGSYIMM 6.0 IC50 2
GSIXSVTVZDJDOC 6.0 IC50 2 Yes
HMXDWDSNPRNUKI 6.0 Ki 72
IEAOMUBPJVXBAO 6.0 IC50 2 Yes
LGYKPDHARJMLQN 6.0 IC50 2
OIVTVLWHNZZBJN 6.0 IC50 2 Yes
QPEUEORJEDJUHX 6.0 IC50 2
RRZKRPHYMGDLBB 6.0 IC50 2 Yes
TXSXJYRAIUVBDO 6.0 IC50 2 Yes
XLWHWNHGNRPPBH 6.0 Ki 2 Yes
XLWHWNHGNRPPBH 6.0 Ki 2 Yes
YJMMQRORYCUFDF 6.0 IC50 2 Yes
2D structure