Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
VKOORZDCJQQHKM 6.7 Ki 2 Yes
DTSANQSRTBGPPK 6.7 IC50 2 Yes
NENKRICCIWXRGU 6.7 Ki 4 Yes
NIQAYAGJQYCQNK 6.7 IC50 2 Yes
RSXHCVGPXZSMBO 6.7 IC50 2 Yes
ZEDOJUJFHGOAOS 6.7 Ki 2
BETHSQILIUBHDZ 6.7 IC50 2 Yes
HHYKRIBHFNFXEL 6.7 IC50 2 Yes
LTBDUUVNJFIMTM 6.7 IC50 2
SNVSYPLFUFXAES 6.7 IC50 2
TVINVHGLLFLSBP 6.7 Ki 4
IIYXZVJGZRIIKG 6.7 IC50 2 Yes
CVCDJFWPDDHHOS 6.7 IC50 2
KWQBJVBPMDEZRS 6.7 Ki 2
DILLUBXISCIMIT 6.7 IC50 2
WFRCVVPACDUWGD 6.7 Ki 2 Yes
GEOWQTGMJLRVOC 6.6 IC50 2 Yes
SKGADOFSECCZFC 6.6 Ki 2 Yes
NFHRQQKPEBFUJK 6.6 IC50 2 Yes
WNWLMMMHXDFXKP 6.6 IC50 2
AICFYCNTUWZWAG 6.6 Ki 2 Yes
HYWPVMQNTSVAPF 6.5 IC50 2 Yes
ZKCCHRIGDWWTRL 6.5 IC50 2 Yes
KLTPQGIBPCHXAQ 6.5 IC50 2
WCLONOKYROXQCI 6.5 IC50 2 Yes
WKUGDHYDAPFFHF 6.5 Ki 2
IAYFRXOMWAZQGV 6.5 IC50 2
SEIABTQHADRMGY 6.4 IC50 2 Yes
VZSPHGCBTKXLMY 6.4 IC50 2 Yes
YBJYGPHLNAJPTE 6.4 IC50 2 Yes
NBOSZKXBNZIDBS 6.4 Ki 2 Yes
CMYMFJIRDMYHDJ 6.4 IC50 2 Yes
WINOYNIKWSTXQD 6.4 Ki 2 Yes
OROBBIIDFVAOPI 6.4 IC50 2 Yes
NQWFBQBJSJTMCW 6.4 IC50 2 Yes
VJHDZLBKGPSGON 6.4 IC50 2 Yes
BAWQUHWZYDWDIH 6.4 IC50 2 Yes
XKDCRXFJHGOCJK 6.4 IC50 2 Yes
NAYWENBSENWRRT 6.3 IC50 2 Yes
OROBBIIDFVAOPI 6.3 IC50 2 Yes
GCLKVXOCZDHVEF 6.3 IC50 2
LOXHZBJMXMSEOS 6.3 Ki 2
KWYHFHAIKHYSHF 6.3 IC50 2 Yes
FMPRFCINNRGLNV 6.3 IC50 2 Yes
IHRCGSOFHCURCS 6.2 IC50 2 Yes
VVKBKPBAKDXLOT 6.2 IC50 3 Yes
UFHHKCDGLUBGJY 6.2 IC50 2 Yes
YJRSAZMDFOJHLB 6.2 IC50 2 Yes
YXNZPENQMVNHAZ 6.2 IC50 2
PRUIQGOHWDZVJD 6.2 Ki 2
2D structure