Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKOORZDCJQQHKM
|
6.7 | Ki | 2 | Yes | |
DTSANQSRTBGPPK
|
6.7 | IC50 | 2 | Yes | |
NENKRICCIWXRGU
|
6.7 | Ki | 4 | Yes | |
NIQAYAGJQYCQNK
|
6.7 | IC50 | 2 | Yes | |
RSXHCVGPXZSMBO
|
6.7 | IC50 | 2 | Yes | |
ZEDOJUJFHGOAOS
|
6.7 | Ki | 2 | — | |
BETHSQILIUBHDZ
|
6.7 | IC50 | 2 | Yes | |
HHYKRIBHFNFXEL
|
6.7 | IC50 | 2 | Yes | |
LTBDUUVNJFIMTM
|
6.7 | IC50 | 2 | — | |
SNVSYPLFUFXAES
|
6.7 | IC50 | 2 | — | |
TVINVHGLLFLSBP
|
6.7 | Ki | 4 | — | |
IIYXZVJGZRIIKG
|
6.7 | IC50 | 2 | Yes | |
CVCDJFWPDDHHOS
|
6.7 | IC50 | 2 | — | |
KWQBJVBPMDEZRS
|
6.7 | Ki | 2 | — | |
DILLUBXISCIMIT
|
6.7 | IC50 | 2 | — | |
WFRCVVPACDUWGD
|
6.7 | Ki | 2 | Yes | |
GEOWQTGMJLRVOC
|
6.6 | IC50 | 2 | Yes | |
SKGADOFSECCZFC
|
6.6 | Ki | 2 | Yes | |
NFHRQQKPEBFUJK
|
6.6 | IC50 | 2 | Yes | |
WNWLMMMHXDFXKP
|
6.6 | IC50 | 2 | — | |
AICFYCNTUWZWAG
|
6.6 | Ki | 2 | Yes | |
HYWPVMQNTSVAPF
|
6.5 | IC50 | 2 | Yes | |
ZKCCHRIGDWWTRL
|
6.5 | IC50 | 2 | Yes | |
KLTPQGIBPCHXAQ
|
6.5 | IC50 | 2 | — | |
WCLONOKYROXQCI
|
6.5 | IC50 | 2 | Yes | |
WKUGDHYDAPFFHF
|
6.5 | Ki | 2 | — | |
IAYFRXOMWAZQGV
|
6.5 | IC50 | 2 | — | |
SEIABTQHADRMGY
|
6.4 | IC50 | 2 | Yes | |
VZSPHGCBTKXLMY
|
6.4 | IC50 | 2 | Yes | |
YBJYGPHLNAJPTE
|
6.4 | IC50 | 2 | Yes | |
NBOSZKXBNZIDBS
|
6.4 | Ki | 2 | Yes | |
CMYMFJIRDMYHDJ
|
6.4 | IC50 | 2 | Yes | |
WINOYNIKWSTXQD
|
6.4 | Ki | 2 | Yes | |
OROBBIIDFVAOPI
|
6.4 | IC50 | 2 | Yes | |
NQWFBQBJSJTMCW
|
6.4 | IC50 | 2 | Yes | |
VJHDZLBKGPSGON
|
6.4 | IC50 | 2 | Yes | |
BAWQUHWZYDWDIH
|
6.4 | IC50 | 2 | Yes | |
XKDCRXFJHGOCJK
|
6.4 | IC50 | 2 | Yes | |
NAYWENBSENWRRT
|
6.3 | IC50 | 2 | Yes | |
OROBBIIDFVAOPI
|
6.3 | IC50 | 2 | Yes | |
GCLKVXOCZDHVEF
|
6.3 | IC50 | 2 | — | |
LOXHZBJMXMSEOS
|
6.3 | Ki | 2 | — | |
KWYHFHAIKHYSHF
|
6.3 | IC50 | 2 | Yes | |
FMPRFCINNRGLNV
|
6.3 | IC50 | 2 | Yes | |
IHRCGSOFHCURCS
|
6.2 | IC50 | 2 | Yes | |
VVKBKPBAKDXLOT
|
6.2 | IC50 | 3 | Yes | |
UFHHKCDGLUBGJY
|
6.2 | IC50 | 2 | Yes | |
YJRSAZMDFOJHLB
|
6.2 | IC50 | 2 | Yes | |
YXNZPENQMVNHAZ
|
6.2 | IC50 | 2 | — | |
PRUIQGOHWDZVJD
|
6.2 | Ki | 2 | — |