Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
POOPTTIQXTUHMQ
|
7.2 | IC50 | 2 | Yes | |
FEOAQCGOOODCEB
|
7.2 | Ki | 2 | — | |
FPVZBTVLTPLRDX
|
7.2 | Ki | 2 | Yes | |
KGFIYGFYTIJLRJ
|
7.2 | IC50 | 2 | Yes | |
AWJDNWMDTDIGNU
|
7.1 | Ki | 2 | — | |
GMAIGIQFMVFLBZ
|
7.1 | Ki | 2 | Yes | |
MIUNVYQVNGDVKG
|
7.1 | IC50 | 2 | Yes | |
DEOUZOCNOYBARB
|
7.1 | Ki | 2 | Yes | |
HBSCTWOGVRBGQM
|
7.1 | IC50 | 2 | Yes | |
LWLWLSWDXYMACR
|
7.1 | IC50 | 2 | — | |
RGFJPHVCLXSEHE
|
7.1 | Ki | 2 | Yes | |
XQSCLQLQGFXSLK
|
7.1 | IC50 | 2 | Yes | |
IHTFQIMRRQEUKB
|
7.0 | Ki | 2 | — | |
SLBLGMBJPJLBTA
|
7.0 | Ki | 2 | Yes | |
QHXBSJRCFQZXTO
|
7.0 | IC50 | 2 | Yes | |
SNYZWGJVKSJMGZ
|
7.0 | IC50 | 2 | Yes | |
VNIAHKVXCCCDOZ
|
7.0 | IC50 | 2 | Yes | |
AHRZYQWKXXBNHK
|
7.0 | Ki | 4 | Yes | |
FSEWRHPBSMPGFF
|
7.0 | Ki | 2 | — | |
TVINVHGLLFLSBP
|
7.0 | IC50 | 4 | Yes | |
BJABGWNNTUGRHH
|
6.9 | Ki | 2 | Yes | |
QPEUEORJEDJUHX
|
6.9 | IC50 | 2 | — | |
RTYGUEPUOWLIME
|
6.9 | IC50 | 2 | Yes | |
ATZKJWWUDVCPPQ
|
6.9 | IC50 | 2 | Yes | |
BYSPJTKARHNTCE
|
6.9 | IC50 | 2 | Yes | |
KSEULEJGJDECHB
|
6.9 | IC50 | 2 | Yes | |
PDWDMFQEOPBNJU
|
6.9 | IC50 | 2 | — | |
ZJGPYSQTJSMQNL
|
6.9 | IC50 | 2 | — | |
ZZVLKHHSRQKCEV
|
6.9 | Ki | 4 | Yes | |
BVUCMLHZVCAVLT
|
6.9 | Ki | 2 | — | |
KSEULEJGJDECHB
|
6.9 | IC50 | 2 | Yes | |
LQEROZJFLGEKCE
|
6.9 | IC50 | 2 | — | |
DDMOESJKCONAST
|
6.9 | Ki | 2 | Yes | |
GWSFJWULDCAOKV
|
6.9 | IC50 | 2 | Yes | |
DXRCYRRBLUBBSH
|
6.8 | IC50 | 2 | Yes | |
IHNBBRXFWBWHAP
|
6.8 | IC50 | 2 | — | |
UBNMGTSDHSQBEL
|
6.8 | IC50 | 2 | — | |
WVNNVFIQARDNCG
|
6.8 | IC50 | 2 | — | |
LTNSZIYAGMZDDY
|
6.8 | Ki | 3 | Yes | |
HSPFWSJPWOITQE
|
6.8 | IC50 | 2 | Yes | |
DZACSGLWVJJFJL
|
6.8 | IC50 | 2 | Yes | |
IBEXWSKBKHNHHX
|
6.8 | IC50 | 2 | Yes | |
OIXQINQYMGNCII
|
6.8 | IC50 | 2 | Yes | |
ZCLCUGHPNSTPGZ
|
6.8 | IC50 | 2 | Yes | |
MLJPZDPDIBXWNY
|
6.8 | IC50 | 2 | — | |
PKHVPLITWFVWGV
|
6.8 | IC50 | 2 | — | |
CFAMCNLQPGYLTL
|
6.7 | Ki | 2 | Yes | |
CLFXXEFAURLAMH
|
6.7 | IC50 | 2 | Yes | |
JMDKMESJXNSGPX
|
6.7 | Ki | 4 | Yes | |
NUPMWKNZJMFJQO
|
6.7 | IC50 | 2 | Yes |