Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
POOPTTIQXTUHMQ 7.2 IC50 2 Yes
FEOAQCGOOODCEB 7.2 Ki 2
FPVZBTVLTPLRDX 7.2 Ki 2 Yes
KGFIYGFYTIJLRJ 7.2 IC50 2 Yes
AWJDNWMDTDIGNU 7.1 Ki 2
GMAIGIQFMVFLBZ 7.1 Ki 2 Yes
MIUNVYQVNGDVKG 7.1 IC50 2 Yes
DEOUZOCNOYBARB 7.1 Ki 2 Yes
HBSCTWOGVRBGQM 7.1 IC50 2 Yes
LWLWLSWDXYMACR 7.1 IC50 2
RGFJPHVCLXSEHE 7.1 Ki 2 Yes
XQSCLQLQGFXSLK 7.1 IC50 2 Yes
IHTFQIMRRQEUKB 7.0 Ki 2
SLBLGMBJPJLBTA 7.0 Ki 2 Yes
QHXBSJRCFQZXTO 7.0 IC50 2 Yes
SNYZWGJVKSJMGZ 7.0 IC50 2 Yes
VNIAHKVXCCCDOZ 7.0 IC50 2 Yes
AHRZYQWKXXBNHK 7.0 Ki 4 Yes
FSEWRHPBSMPGFF 7.0 Ki 2
TVINVHGLLFLSBP 7.0 IC50 4 Yes
BJABGWNNTUGRHH 6.9 Ki 2 Yes
QPEUEORJEDJUHX 6.9 IC50 2
RTYGUEPUOWLIME 6.9 IC50 2 Yes
ATZKJWWUDVCPPQ 6.9 IC50 2 Yes
BYSPJTKARHNTCE 6.9 IC50 2 Yes
KSEULEJGJDECHB 6.9 IC50 2 Yes
PDWDMFQEOPBNJU 6.9 IC50 2
ZJGPYSQTJSMQNL 6.9 IC50 2
ZZVLKHHSRQKCEV 6.9 Ki 4 Yes
BVUCMLHZVCAVLT 6.9 Ki 2
KSEULEJGJDECHB 6.9 IC50 2 Yes
LQEROZJFLGEKCE 6.9 IC50 2
DDMOESJKCONAST 6.9 Ki 2 Yes
GWSFJWULDCAOKV 6.9 IC50 2 Yes
DXRCYRRBLUBBSH 6.8 IC50 2 Yes
IHNBBRXFWBWHAP 6.8 IC50 2
UBNMGTSDHSQBEL 6.8 IC50 2
WVNNVFIQARDNCG 6.8 IC50 2
LTNSZIYAGMZDDY 6.8 Ki 3 Yes
HSPFWSJPWOITQE 6.8 IC50 2 Yes
DZACSGLWVJJFJL 6.8 IC50 2 Yes
IBEXWSKBKHNHHX 6.8 IC50 2 Yes
OIXQINQYMGNCII 6.8 IC50 2 Yes
ZCLCUGHPNSTPGZ 6.8 IC50 2 Yes
MLJPZDPDIBXWNY 6.8 IC50 2
PKHVPLITWFVWGV 6.8 IC50 2
CFAMCNLQPGYLTL 6.7 Ki 2 Yes
CLFXXEFAURLAMH 6.7 IC50 2 Yes
JMDKMESJXNSGPX 6.7 Ki 4 Yes
NUPMWKNZJMFJQO 6.7 IC50 2 Yes
2D structure