Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
DDROKKYSSQPXQO 7.6 IC50 2 Yes
ITMJPTIFWLPIOL 7.6 IC50 2 Yes
VTMQSICVVWNLPW 7.6 Ki 2
DWHRPZRXNRDAQF 7.6 Ki 3 Yes
IZIFZVHACKDILP 7.6 Ki 2 Yes
SDJPEEZPMPFEON 7.6 IC50 2 Yes
GQFWYWXTSTVXPK 7.5 IC50 2 Yes
NIQAYAGJQYCQNK 7.5 IC50 2 Yes
PKNBIEKWQLWZNJ 7.5 IC50 2 Yes
VHAAOROZSHMZRJ 7.5 IC50 2 Yes
VNIAHKVXCCCDOZ 7.5 IC50 2 Yes
XNUGDRMOEPOBFR 7.5 IC50 2 Yes
YYUMVSJDMJRIKE 7.5 IC50 2 Yes
CHYXBVRNXVPDAR 7.5 IC50 2 Yes
MPLZTZIWSHXYGD 7.5 IC50 2 Yes
OGHIDHUMQVCJLH 7.5 IC50 2
OULXGYXKPKVJPL 7.5 IC50 2 Yes
XSHMFCLLINAWBH 7.5 IC50 2
YRULVPAVSSLIEL 7.5 IC50 2 Yes
YLANCCITSFOFMP 7.5 Ki 2
CHEUONHPKBJUCB 7.5 IC50 2 Yes
PFDXGRUVVNQAQW 7.5 IC50 2 Yes
UXSCCYZDWXCQRW 7.5 IC50 2 Yes
NACOKSRFWNZWTN 7.5 IC50 2 Yes
MUNNAUUHDXISAJ 7.4 Ki 2 Yes
RUXGBVNMEPICAJ 7.4 IC50 2 Yes
KTIVKLXXTDQNMF 7.4 Ki 2 Yes
DPTKJTLNHCGWTH 7.4 Ki 2 Yes
IRRPCAFDQVDMNP 7.4 Ki 2
NCXFVQVUXTYYEG 7.4 Ki 2 Yes
VLKJKVMACAESPP 7.4 Kd 2 Yes
XWNQRVQSRVNMGY 7.4 IC50 2 Yes
INPUMSDGOIKULR 7.4 IC50 2 Yes
GKKCSRUSTYGKFF 7.4 IC50 2 Yes
FAQSZDGODZYSIN 7.4 IC50 2 Yes
LJOCWELELLFJSQ 7.4 Ki 2
VQXCMRAQZMSGPR 7.4 Ki 2
GAUFCDPHSYEFLM 7.3 IC50 2
HMGDEYJMBGQTPV 7.3 Ki 2 Yes
USWDPRRJNGKNQG 7.3 IC50 2 Yes
JZBWOSXHOVOLBT 7.3 Ki 2 Yes
PWEFAKIGTKFZQK 7.3 Ki 2 Yes
HRFMJPIGMOWHLL 7.3 IC50 2 Yes
BERNHFOYDVXQGI 7.3 IC50 2 Yes
ZMTRGKKPVWRAII 7.3 IC50 2 Yes
XLQIEICIMTUDOM 7.2 Ki 2
PIHWDFKUEPTNFH 7.2 IC50 2 Yes
HSPTWXGPKMKONJ 7.2 IC50 2 Yes
ZMTXZNHONYLRJA 7.2 IC50 2 Yes
BFIXTZFVFDMGQQ 7.2 IC50 2
2D structure