Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DDROKKYSSQPXQO
|
7.6 | IC50 | 2 | Yes | |
ITMJPTIFWLPIOL
|
7.6 | IC50 | 2 | Yes | |
VTMQSICVVWNLPW
|
7.6 | Ki | 2 | — | |
DWHRPZRXNRDAQF
|
7.6 | Ki | 3 | Yes | |
IZIFZVHACKDILP
|
7.6 | Ki | 2 | Yes | |
SDJPEEZPMPFEON
|
7.6 | IC50 | 2 | Yes | |
GQFWYWXTSTVXPK
|
7.5 | IC50 | 2 | Yes | |
NIQAYAGJQYCQNK
|
7.5 | IC50 | 2 | Yes | |
PKNBIEKWQLWZNJ
|
7.5 | IC50 | 2 | Yes | |
VHAAOROZSHMZRJ
|
7.5 | IC50 | 2 | Yes | |
VNIAHKVXCCCDOZ
|
7.5 | IC50 | 2 | Yes | |
XNUGDRMOEPOBFR
|
7.5 | IC50 | 2 | Yes | |
YYUMVSJDMJRIKE
|
7.5 | IC50 | 2 | Yes | |
CHYXBVRNXVPDAR
|
7.5 | IC50 | 2 | Yes | |
MPLZTZIWSHXYGD
|
7.5 | IC50 | 2 | Yes | |
OGHIDHUMQVCJLH
|
7.5 | IC50 | 2 | — | |
OULXGYXKPKVJPL
|
7.5 | IC50 | 2 | Yes | |
XSHMFCLLINAWBH
|
7.5 | IC50 | 2 | — | |
YRULVPAVSSLIEL
|
7.5 | IC50 | 2 | Yes | |
YLANCCITSFOFMP
|
7.5 | Ki | 2 | — | |
CHEUONHPKBJUCB
|
7.5 | IC50 | 2 | Yes | |
PFDXGRUVVNQAQW
|
7.5 | IC50 | 2 | Yes | |
UXSCCYZDWXCQRW
|
7.5 | IC50 | 2 | Yes | |
NACOKSRFWNZWTN
|
7.5 | IC50 | 2 | Yes | |
MUNNAUUHDXISAJ
|
7.4 | Ki | 2 | Yes | |
RUXGBVNMEPICAJ
|
7.4 | IC50 | 2 | Yes | |
KTIVKLXXTDQNMF
|
7.4 | Ki | 2 | Yes | |
DPTKJTLNHCGWTH
|
7.4 | Ki | 2 | Yes | |
IRRPCAFDQVDMNP
|
7.4 | Ki | 2 | — | |
NCXFVQVUXTYYEG
|
7.4 | Ki | 2 | Yes | |
VLKJKVMACAESPP
|
7.4 | Kd | 2 | Yes | |
XWNQRVQSRVNMGY
|
7.4 | IC50 | 2 | Yes | |
INPUMSDGOIKULR
|
7.4 | IC50 | 2 | Yes | |
GKKCSRUSTYGKFF
|
7.4 | IC50 | 2 | Yes | |
FAQSZDGODZYSIN
|
7.4 | IC50 | 2 | Yes | |
LJOCWELELLFJSQ
|
7.4 | Ki | 2 | — | |
VQXCMRAQZMSGPR
|
7.4 | Ki | 2 | — | |
GAUFCDPHSYEFLM
|
7.3 | IC50 | 2 | — | |
HMGDEYJMBGQTPV
|
7.3 | Ki | 2 | Yes | |
USWDPRRJNGKNQG
|
7.3 | IC50 | 2 | Yes | |
JZBWOSXHOVOLBT
|
7.3 | Ki | 2 | Yes | |
PWEFAKIGTKFZQK
|
7.3 | Ki | 2 | Yes | |
HRFMJPIGMOWHLL
|
7.3 | IC50 | 2 | Yes | |
BERNHFOYDVXQGI
|
7.3 | IC50 | 2 | Yes | |
ZMTRGKKPVWRAII
|
7.3 | IC50 | 2 | Yes | |
XLQIEICIMTUDOM
|
7.2 | Ki | 2 | — | |
PIHWDFKUEPTNFH
|
7.2 | IC50 | 2 | Yes | |
HSPTWXGPKMKONJ
|
7.2 | IC50 | 2 | Yes | |
ZMTXZNHONYLRJA
|
7.2 | IC50 | 2 | Yes | |
BFIXTZFVFDMGQQ
|
7.2 | IC50 | 2 | — |