Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LZZPPPZINPSHEI
|
8.2 | Ki | 2 | Yes | |
RGJCMCCPAYOLOE
|
8.2 | Ki | 2 | Yes | |
PIYVAPZSWIDNTQ
|
8.2 | IC50 | 2 | Yes | |
VLKJKVMACAESPP
|
8.2 | IC50 | 2 | — | |
STXYGGMUUHCKOP
|
8.1 | Ki | 2 | — | |
UWZVTINXEBCDPO
|
8.1 | IC50 | 2 | Yes | |
ORTWASXZYRMKIJ
|
8.1 | IC50 | 2 | Yes | |
SJDGAPPCMGPKLY
|
8.1 | IC50 | 2 | Yes | |
CSNNJXSLJWKSCD
|
8.1 | IC50 | 2 | Yes | |
WLTSODCLBUFUDX
|
8.1 | IC50 | 2 | Yes | |
AHYNKYYQUAOMCJ
|
8.1 | Ki | 2 | — | |
QOSWNOTZBYMOLA
|
8.1 | IC50 | 2 | Yes | |
MYKVVXCIFKAFIQ
|
8.1 | IC50 | 2 | Yes | |
SYGCFCSEEIGJCO
|
8.1 | IC50 | 2 | Yes | |
ALSNOSFKYCYLJH
|
8.0 | IC50 | 2 | Yes | |
CABBMMXFOOZVMS
|
8.0 | IC50 | 2 | — | |
RAYLDYGVHMTPSI
|
8.0 | Ki | 2 | Yes | |
SBMRIYCGYSYWIJ
|
8.0 | IC50 | 2 | Yes | |
WGLBHEKCPCUEDT
|
8.0 | Ki | 2 | Yes | |
ZANFFYJCTUAWAK
|
8.0 | IC50 | 2 | Yes | |
DVASHPOLPKOKGD
|
8.0 | IC50 | 2 | Yes | |
GDFLLWZJUDPZMX
|
8.0 | Ki | 2 | — | |
HPZJMUBDEAMBFI
|
8.0 | Ki | 5 | — | |
UIISAWYHPZCXHX
|
7.9 | Ki | 2 | Yes | |
HEEJTBJFKMOMFO
|
7.9 | Ki | 2 | — | |
HLUCCSPJVQTJTM
|
7.9 | Ki | 2 | — | |
NFNSLUVCTGTZGY
|
7.9 | Ki | 2 | — | |
DQWCJWUIFIKCRT
|
7.9 | Ki | 2 | — | |
NCCODGOBVZOLFU
|
7.8 | Ki | 2 | Yes | |
RYNRWNJFDSYFLB
|
7.8 | Ki | 2 | Yes | |
YXAVZKKJFIOGEL
|
7.8 | Ki | 2 | — | |
BDKLOKRNGDIZTO
|
7.8 | Ki | 2 | Yes | |
KKPFQTRKARZYLE
|
7.8 | Ki | 3 | Yes | |
WDLOTEQZLXZCSI
|
7.8 | IC50 | 2 | Yes | |
YVOYRMXNVINXII
|
7.8 | Ki | 3 | Yes | |
HVCMNKCXHIIFDJ
|
7.8 | IC50 | 2 | Yes | |
JPSKDACFMPXNMN
|
7.8 | IC50 | 2 | — | |
NAYWENBSENWRRT
|
7.8 | IC50 | 2 | Yes | |
STEAMACHIRWBBH
|
7.8 | IC50 | 3 | — | |
DYFJGOOJNUUTLF
|
7.8 | Ki | 2 | — | |
NDMKAESGNQHGID
|
7.8 | Ki | 2 | — | |
ZUUGDHAKGUQZKD
|
7.7 | Ki | 3 | Yes | |
MLJPZDPDIBXWNY
|
7.7 | IC50 | 2 | — | |
AHKXHAMSXLISEI
|
7.7 | Ki | 2 | — | |
RLKUXRWOAPPZQB
|
7.7 | Ki | 2 | — | |
RSSCBKHOJPGYIW
|
7.6 | Ki | 2 | — | |
ALPLVUYDOOIUAE
|
7.6 | IC50 | 2 | Yes | |
BUDVFFOVUFVRER
|
7.6 | IC50 | 2 | Yes | |
ZJQCLCIESPIJML
|
7.6 | Ki | 2 | — | |
AKHKIVGBTDKSGG
|
7.6 | IC50 | 2 | Yes |