Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
LZZPPPZINPSHEI 8.2 Ki 2 Yes
RGJCMCCPAYOLOE 8.2 Ki 2 Yes
PIYVAPZSWIDNTQ 8.2 IC50 2 Yes
VLKJKVMACAESPP 8.2 IC50 2
STXYGGMUUHCKOP 8.1 Ki 2
UWZVTINXEBCDPO 8.1 IC50 2 Yes
ORTWASXZYRMKIJ 8.1 IC50 2 Yes
SJDGAPPCMGPKLY 8.1 IC50 2 Yes
CSNNJXSLJWKSCD 8.1 IC50 2 Yes
WLTSODCLBUFUDX 8.1 IC50 2 Yes
AHYNKYYQUAOMCJ 8.1 Ki 2
QOSWNOTZBYMOLA 8.1 IC50 2 Yes
MYKVVXCIFKAFIQ 8.1 IC50 2 Yes
SYGCFCSEEIGJCO 8.1 IC50 2 Yes
ALSNOSFKYCYLJH 8.0 IC50 2 Yes
CABBMMXFOOZVMS 8.0 IC50 2
RAYLDYGVHMTPSI 8.0 Ki 2 Yes
SBMRIYCGYSYWIJ 8.0 IC50 2 Yes
WGLBHEKCPCUEDT 8.0 Ki 2 Yes
ZANFFYJCTUAWAK 8.0 IC50 2 Yes
DVASHPOLPKOKGD 8.0 IC50 2 Yes
GDFLLWZJUDPZMX 8.0 Ki 2
HPZJMUBDEAMBFI 8.0 Ki 5
UIISAWYHPZCXHX 7.9 Ki 2 Yes
HEEJTBJFKMOMFO 7.9 Ki 2
HLUCCSPJVQTJTM 7.9 Ki 2
NFNSLUVCTGTZGY 7.9 Ki 2
DQWCJWUIFIKCRT 7.9 Ki 2
NCCODGOBVZOLFU 7.8 Ki 2 Yes
RYNRWNJFDSYFLB 7.8 Ki 2 Yes
YXAVZKKJFIOGEL 7.8 Ki 2
BDKLOKRNGDIZTO 7.8 Ki 2 Yes
KKPFQTRKARZYLE 7.8 Ki 3 Yes
WDLOTEQZLXZCSI 7.8 IC50 2 Yes
YVOYRMXNVINXII 7.8 Ki 3 Yes
HVCMNKCXHIIFDJ 7.8 IC50 2 Yes
JPSKDACFMPXNMN 7.8 IC50 2
NAYWENBSENWRRT 7.8 IC50 2 Yes
STEAMACHIRWBBH 7.8 IC50 3
DYFJGOOJNUUTLF 7.8 Ki 2
NDMKAESGNQHGID 7.8 Ki 2
ZUUGDHAKGUQZKD 7.7 Ki 3 Yes
MLJPZDPDIBXWNY 7.7 IC50 2
AHKXHAMSXLISEI 7.7 Ki 2
RLKUXRWOAPPZQB 7.7 Ki 2
RSSCBKHOJPGYIW 7.6 Ki 2
ALPLVUYDOOIUAE 7.6 IC50 2 Yes
BUDVFFOVUFVRER 7.6 IC50 2 Yes
ZJQCLCIESPIJML 7.6 Ki 2
AKHKIVGBTDKSGG 7.6 IC50 2 Yes
2D structure