Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TVNLSGMCRJXNND
|
9.0 | IC50 | 2 | Yes | |
CMYDNIJMVCZZQK
|
9.0 | IC50 | 2 | Yes | |
KKPFQTRKARZYLE
|
9.0 | Ki | 3 | Yes | |
AIQFACLFKVFQQI
|
8.9 | Ki | 2 | — | |
LXFPQYIZOTVJFQ
|
8.9 | Ki | 2 | — | |
IEJRYJFWTCKXSD
|
8.8 | IC50 | 2 | Yes | |
ZYFZAOVAALGAJO
|
8.8 | IC50 | 2 | Yes | |
LFIFGNCFEBAIHA
|
8.8 | Ki | 4 | Yes | |
UGINDELNLJSTRU
|
8.8 | IC50 | 2 | Yes | |
KKPFQTRKARZYLE
|
8.8 | Ki | 4 | Yes | |
LFIFGNCFEBAIHA
|
8.8 | Ki | 3 | Yes | |
WFEXFFRNIOUBQX
|
8.8 | Ki | 2 | — | |
WYYQDZXURPONSW
|
8.8 | Ki | 2 | — | |
OFQAQYAFHZCAOX
|
8.8 | IC50 | 2 | Yes | |
JVCLXDNXAUQCLR
|
8.7 | IC50 | 2 | — | |
OGWBASUUCLOVLN
|
8.7 | IC50 | 2 | Yes | |
FVTWFHUCJJXREC
|
8.7 | IC50 | 2 | Yes | |
OCVIYTKLKRGXCI
|
8.7 | IC50 | 2 | — | |
QRYOMNSPKSJSKG
|
8.7 | IC50 | 2 | Yes | |
ZANGNFNVUAPKGY
|
8.7 | IC50 | 2 | Yes | |
IJHCWGDIGBABKC
|
8.7 | IC50 | 3 | Yes | |
IJHCWGDIGBABKC
|
8.7 | Ki | 3 | Yes | |
LGRKVVHGUJOXEN
|
8.7 | Ki | 4 | Yes | |
ZINWBFHVGIYPGZ
|
8.7 | IC50 | 2 | — | |
JHFTVYNYYKDISE
|
8.7 | IC50 | 2 | Yes | |
JJAYAAFBSRHMID
|
8.7 | IC50 | 2 | Yes | |
CLMCTKVZMVJCQP
|
8.6 | IC50 | 2 | Yes | |
URMOKEJAUAGZGV
|
8.6 | Ki | 2 | — | |
BFSMHEBYNOKMKU
|
8.6 | IC50 | 2 | Yes | |
XMLJSDGQSNTHPG
|
8.6 | Ki | 2 | — | |
KDFQABSFVYLGPM
|
8.5 | IC50 | 2 | Yes | |
CXNFPROZKYIEPE
|
8.5 | IC50 | 2 | Yes | |
DZFMLNMPSVVWNC
|
8.5 | IC50 | 2 | Yes | |
JMFXHOKUYGTFJU
|
8.5 | IC50 | 2 | Yes | |
KONMZUWCOVKBMG
|
8.4 | IC50 | 2 | — | |
KJQHRGYUFQCLJG
|
8.4 | Ki | 2 | — | |
RKKAWDULAQHRCY
|
8.4 | IC50 | 2 | Yes | |
QWOAONQRBDJQTC
|
8.4 | IC50 | 2 | Yes | |
GKDWRERMBNGKCZ
|
8.4 | IC50 | 2 | — | |
LJAZTWRBCMHLKX
|
8.4 | IC50 | 2 | Yes | |
IBOMYHWWSMSHBV
|
8.4 | IC50 | 2 | Yes | |
NXHWDEQNHXTHJU
|
8.3 | IC50 | 3 | Yes | |
DAZGMBOFHKYQHK
|
8.3 | IC50 | 2 | Yes | |
KSAGKPZDJHLHBS
|
8.3 | Ki | 4 | Yes | |
PFOLRJQYZKGBLP
|
8.3 | IC50 | 2 | Yes | |
QAZGXXFYHAMXIB
|
8.3 | Ki | 2 | Yes | |
MPQWSQLPSQOSKO
|
8.3 | IC50 | 2 | Yes | |
CABBMMXFOOZVMS
|
8.2 | IC50 | 2 | — | |
VMFFXQXFIYFZKK
|
8.2 | IC50 | 2 | — | |
BZVZYXCWVJJFDH
|
8.2 | Ki | 2 | Yes |