Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
TVNLSGMCRJXNND 9.0 IC50 2 Yes
CMYDNIJMVCZZQK 9.0 IC50 2 Yes
KKPFQTRKARZYLE 9.0 Ki 3 Yes
AIQFACLFKVFQQI 8.9 Ki 2
LXFPQYIZOTVJFQ 8.9 Ki 2
IEJRYJFWTCKXSD 8.8 IC50 2 Yes
ZYFZAOVAALGAJO 8.8 IC50 2 Yes
LFIFGNCFEBAIHA 8.8 Ki 4 Yes
UGINDELNLJSTRU 8.8 IC50 2 Yes
KKPFQTRKARZYLE 8.8 Ki 4 Yes
LFIFGNCFEBAIHA 8.8 Ki 3 Yes
WFEXFFRNIOUBQX 8.8 Ki 2
WYYQDZXURPONSW 8.8 Ki 2
OFQAQYAFHZCAOX 8.8 IC50 2 Yes
JVCLXDNXAUQCLR 8.7 IC50 2
OGWBASUUCLOVLN 8.7 IC50 2 Yes
FVTWFHUCJJXREC 8.7 IC50 2 Yes
OCVIYTKLKRGXCI 8.7 IC50 2
QRYOMNSPKSJSKG 8.7 IC50 2 Yes
ZANGNFNVUAPKGY 8.7 IC50 2 Yes
IJHCWGDIGBABKC 8.7 IC50 3 Yes
IJHCWGDIGBABKC 8.7 Ki 3 Yes
LGRKVVHGUJOXEN 8.7 Ki 4 Yes
ZINWBFHVGIYPGZ 8.7 IC50 2
JHFTVYNYYKDISE 8.7 IC50 2 Yes
JJAYAAFBSRHMID 8.7 IC50 2 Yes
CLMCTKVZMVJCQP 8.6 IC50 2 Yes
URMOKEJAUAGZGV 8.6 Ki 2
BFSMHEBYNOKMKU 8.6 IC50 2 Yes
XMLJSDGQSNTHPG 8.6 Ki 2
KDFQABSFVYLGPM 8.5 IC50 2 Yes
CXNFPROZKYIEPE 8.5 IC50 2 Yes
DZFMLNMPSVVWNC 8.5 IC50 2 Yes
JMFXHOKUYGTFJU 8.5 IC50 2 Yes
KONMZUWCOVKBMG 8.4 IC50 2
KJQHRGYUFQCLJG 8.4 Ki 2
RKKAWDULAQHRCY 8.4 IC50 2 Yes
QWOAONQRBDJQTC 8.4 IC50 2 Yes
GKDWRERMBNGKCZ 8.4 IC50 2
LJAZTWRBCMHLKX 8.4 IC50 2 Yes
IBOMYHWWSMSHBV 8.4 IC50 2 Yes
NXHWDEQNHXTHJU 8.3 IC50 3 Yes
DAZGMBOFHKYQHK 8.3 IC50 2 Yes
KSAGKPZDJHLHBS 8.3 Ki 4 Yes
PFOLRJQYZKGBLP 8.3 IC50 2 Yes
QAZGXXFYHAMXIB 8.3 Ki 2 Yes
MPQWSQLPSQOSKO 8.3 IC50 2 Yes
CABBMMXFOOZVMS 8.2 IC50 2
VMFFXQXFIYFZKK 8.2 IC50 2
BZVZYXCWVJJFDH 8.2 Ki 2 Yes
2D structure