Target Details
UniProt ACP32239
Gene SymbolCCKBR
Protein NameGastrin/cholecystokinin type B receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 341
  • Clinical molecules 233
  • Avg pChEMBL 7.59
Top Co-occurrence Targets
Active Molecules (341)
InChIKey pChEMBL Type Targets Clinical
ZFTPEIAEGCLUII 10.2 Ki 2 Yes
IUSFSIDKWAJIKQ 10.0 IC50 2
VKDAZGQQWPSRFA 10.0 IC50 2 Yes
DGKMBNVRIZTNTK 10.0 Ki 2
CYCOQCORURTMQB 9.9 IC50 2
FCDAJLCDHWZLKC 9.9 IC50 2
YDZYKNJZCVIKPP 9.9 Ki 2
ADFBVAUNEXEYJP 9.8 Ki 2 Yes
CSXIDZJPJYRGSK 9.8 Ki 2 Yes
ROJMLIUODNIIEZ 9.8 IC50 2
LXWCNCKGNPJZAA 9.8 IC50 2
VLYZWOUEQOSDIN 9.7 Ki 2
UDFKASJOSSYSOL 9.7 IC50 2
DNKPXDLQYBBMPC 9.7 IC50 2 Yes
CNWXJSZWVGJITL 9.6 IC50 2 Yes
VCBHARIFOKYMTC 9.6 Ki 2
SFJVTILNSUYYFI 9.6 IC50 2 Yes
QUSCQANKQSFCGJ 9.6 Ki 2 Yes
CSXIDZJPJYRGSK 9.5 IC50 2 Yes
IFELUJVLOCAXCD 9.5 IC50 2
NMRHHKUTBQFJAA 9.5 Ki 2
PBVOPXCIKKBKIX 9.5 IC50 2 Yes
IZTQOLKUZKXIRV 9.5 IC50 2 Yes
ZAYFSWRWHALHQG 9.4 Ki 2
VDNWZTJUPNHYID 9.4 Ki 2
VNDOMFNPSJBMRV 9.4 IC50 2
ZRTOSCLSAJLFLV 9.4 Ki 2
QPRHQFFOOJJWON 9.3 Ki 2 Yes
DLRAUJSCRJKHJV 9.3 IC50 2 Yes
WLTSODCLBUFUDX 9.3 IC50 2 Yes
GUXRAKLYIXOIFQ 9.2 IC50 2 Yes
JVXUNHXYBLGVPM 9.2 IC50 2
KJQHRGYUFQCLJG 9.2 Ki 4 Yes
LWZREZWAQQSATC 9.2 IC50 2 Yes
OGBLGSTXVFINII 9.2 IC50 2 Yes
WSTOKXRJTCQBGW 9.2 IC50 2 Yes
HUOIRVSSWJKCQP 9.2 Ki 2
NACOKSRFWNZWTN 9.2 IC50 2 Yes
NLKGFOOGBGCDAL 9.2 IC50 2 Yes
NNMKTACSCZBLRL 9.2 Ki 2
YJPQVTKXGCBSPW 9.1 Ki 2 Yes
MQIOWUHVKXZQPM 9.1 IC50 2 Yes
IRCIITOKKBCNGO 9.1 IC50 2 Yes
NWLBBDKAIZNTHK 9.1 IC50 2 Yes
GHEUKVOXUQUGLZ 9.1 IC50 2
ODMAYKFSTPTMKE 9.1 Ki 2
AGBJVABYWAWOKN 9.0 IC50 2 Yes
ARYXAMNDWNZMBO 9.0 IC50 2 Yes
VLKJKVMACAESPP 9.0 Ki 2 Yes
VLKJKVMACAESPP 9.0 Ki 2
2D structure