Target Details
| UniProt AC | P32239 |
|---|---|
| Gene Symbol | CCKBR |
| Protein Name | Gastrin/cholecystokinin type B receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 341
- Clinical molecules 233
- Avg pChEMBL 7.59
KEGG Pathways (4)
Active Molecules (341)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZFTPEIAEGCLUII
|
10.2 | Ki | 2 | Yes | |
IUSFSIDKWAJIKQ
|
10.0 | IC50 | 2 | — | |
VKDAZGQQWPSRFA
|
10.0 | IC50 | 2 | Yes | |
DGKMBNVRIZTNTK
|
10.0 | Ki | 2 | — | |
CYCOQCORURTMQB
|
9.9 | IC50 | 2 | — | |
FCDAJLCDHWZLKC
|
9.9 | IC50 | 2 | — | |
YDZYKNJZCVIKPP
|
9.9 | Ki | 2 | — | |
ADFBVAUNEXEYJP
|
9.8 | Ki | 2 | Yes | |
CSXIDZJPJYRGSK
|
9.8 | Ki | 2 | Yes | |
ROJMLIUODNIIEZ
|
9.8 | IC50 | 2 | — | |
LXWCNCKGNPJZAA
|
9.8 | IC50 | 2 | — | |
VLYZWOUEQOSDIN
|
9.7 | Ki | 2 | — | |
UDFKASJOSSYSOL
|
9.7 | IC50 | 2 | — | |
DNKPXDLQYBBMPC
|
9.7 | IC50 | 2 | Yes | |
CNWXJSZWVGJITL
|
9.6 | IC50 | 2 | Yes | |
VCBHARIFOKYMTC
|
9.6 | Ki | 2 | — | |
SFJVTILNSUYYFI
|
9.6 | IC50 | 2 | Yes | |
QUSCQANKQSFCGJ
|
9.6 | Ki | 2 | Yes | |
CSXIDZJPJYRGSK
|
9.5 | IC50 | 2 | Yes | |
IFELUJVLOCAXCD
|
9.5 | IC50 | 2 | — | |
NMRHHKUTBQFJAA
|
9.5 | Ki | 2 | — | |
PBVOPXCIKKBKIX
|
9.5 | IC50 | 2 | Yes | |
IZTQOLKUZKXIRV
|
9.5 | IC50 | 2 | Yes | |
ZAYFSWRWHALHQG
|
9.4 | Ki | 2 | — | |
VDNWZTJUPNHYID
|
9.4 | Ki | 2 | — | |
VNDOMFNPSJBMRV
|
9.4 | IC50 | 2 | — | |
ZRTOSCLSAJLFLV
|
9.4 | Ki | 2 | — | |
QPRHQFFOOJJWON
|
9.3 | Ki | 2 | Yes | |
DLRAUJSCRJKHJV
|
9.3 | IC50 | 2 | Yes | |
WLTSODCLBUFUDX
|
9.3 | IC50 | 2 | Yes | |
GUXRAKLYIXOIFQ
|
9.2 | IC50 | 2 | Yes | |
JVXUNHXYBLGVPM
|
9.2 | IC50 | 2 | — | |
KJQHRGYUFQCLJG
|
9.2 | Ki | 4 | Yes | |
LWZREZWAQQSATC
|
9.2 | IC50 | 2 | Yes | |
OGBLGSTXVFINII
|
9.2 | IC50 | 2 | Yes | |
WSTOKXRJTCQBGW
|
9.2 | IC50 | 2 | Yes | |
HUOIRVSSWJKCQP
|
9.2 | Ki | 2 | — | |
NACOKSRFWNZWTN
|
9.2 | IC50 | 2 | Yes | |
NLKGFOOGBGCDAL
|
9.2 | IC50 | 2 | Yes | |
NNMKTACSCZBLRL
|
9.2 | Ki | 2 | — | |
YJPQVTKXGCBSPW
|
9.1 | Ki | 2 | Yes | |
MQIOWUHVKXZQPM
|
9.1 | IC50 | 2 | Yes | |
IRCIITOKKBCNGO
|
9.1 | IC50 | 2 | Yes | |
NWLBBDKAIZNTHK
|
9.1 | IC50 | 2 | Yes | |
GHEUKVOXUQUGLZ
|
9.1 | IC50 | 2 | — | |
ODMAYKFSTPTMKE
|
9.1 | Ki | 2 | — | |
AGBJVABYWAWOKN
|
9.0 | IC50 | 2 | Yes | |
ARYXAMNDWNZMBO
|
9.0 | IC50 | 2 | Yes | |
VLKJKVMACAESPP
|
9.0 | Ki | 2 | Yes | |
VLKJKVMACAESPP
|
9.0 | Ki | 2 | — |