Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UFHHKCDGLUBGJY
|
6.2 | pIC50 | 2 | Yes | |
VEGZKBKISJJLJC
|
6.2 | IC50 | 3 | Yes | |
VLYZWOUEQOSDIN
|
6.2 | Ki | 2 | — | |
OZUSVSPHYKYLAS
|
6.2 | pIC50 | 2 | Yes | |
RSSCBKHOJPGYIW
|
6.2 | Ki | 2 | — | |
CTAHPXXZSACISG
|
6.2 | pIC50 | 2 | Yes | |
HUOIRVSSWJKCQP
|
6.2 | Ki | 2 | — | |
UUNNSNYSEQPCKO
|
6.2 | IC50 | 2 | — | |
ZAYFSWRWHALHQG
|
6.2 | Ki | 2 | — | |
ARRVGGQZILZZEJ
|
6.2 | pIC50 | 2 | Yes | |
DDUAFEYIPWOELY
|
6.2 | pIC50 | 2 | Yes | |
BMWKQHPGKPJLPG
|
6.2 | pIC50 | 2 | Yes | |
BERNHFOYDVXQGI
|
6.2 | pIC50 | 2 | Yes | |
GFMBISIECXFEJK
|
6.2 | pIC50 | 2 | Yes | |
NFNSLUVCTGTZGY
|
6.1 | Ki | 2 | — | |
RPNVENCCLVKRAM
|
6.1 | pIC50 | 2 | Yes | |
PSNAHSRRFJSWQU
|
6.1 | pIC50 | 2 | Yes | |
QNCFQRIXQDHLMN
|
6.1 | pIC50 | 2 | Yes | |
IRUDQSQIPJJXFZ
|
6.1 | pIC50 | 2 | Yes | |
DOABBONQBBUCRN
|
6.1 | pIC50 | 2 | Yes | |
YGVMCMZWGQEBFU
|
6.1 | pIC50 | 2 | Yes | |
ACWHYMXOCYJYPG
|
6.1 | pIC50 | 2 | Yes | |
SPJCSYUKRLKAQT
|
6.1 | pIC50 | 2 | Yes | |
VMFFXQXFIYFZKK
|
6.1 | IC50 | 2 | — | |
DTSANQSRTBGPPK
|
6.1 | pIC50 | 2 | Yes | |
GKDWRERMBNGKCZ
|
6.1 | IC50 | 2 | — | |
DUPJRHKBDSHZPG
|
6.0 | pIC50 | 2 | Yes | |
QZFBYNPTVXYUII
|
6.0 | IC50 | 2 | — | |
KJQHRGYUFQCLJG
|
6.0 | pIC50 | 2 | Yes | |
ZOZPVKJSFYNWLP
|
6.0 | pIC50 | 2 | Yes | |
JVXUNHXYBLGVPM
|
6.0 | IC50 | 2 | — | |
XLWHWNHGNRPPBH
|
6.0 | Ki | 2 | Yes | |
GSIXSVTVZDJDOC
|
6.0 | pIC50 | 2 | Yes | |
IEAOMUBPJVXBAO
|
6.0 | pIC50 | 2 | Yes | |
OIVTVLWHNZZBJN
|
6.0 | pIC50 | 2 | Yes | |
RRZKRPHYMGDLBB
|
6.0 | pIC50 | 2 | Yes | |
TXSXJYRAIUVBDO
|
6.0 | pIC50 | 2 | Yes | |
YJMMQRORYCUFDF
|
6.0 | pIC50 | 2 | Yes | |
ZICGXQSIIFWORG
|
6.0 | pIC50 | 2 | Yes | |
CHVZZDMXXHMJNM
|
Clinical | TTD_MultiTarget | 2 | Yes | |
DWHRPZRXNRDAQF
|
Clinical | TTD_MultiTarget | 2 | Yes | |
IYNMVGGOTRCWGJ
|
Clinical | TTD_MultiTarget | 2 | Yes | |
LHFDBKUCTFELLO
|
Clinical | TTD_MultiTarget | 2 | Yes |