Target Details
UniProt ACP32238
Gene SymbolCCKAR
Protein NameCholecystokinin receptor type A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF09193 (CholecysA-Rec_N)
Summary
  • Multi-target molecules 343
  • Clinical molecules 242
  • Avg pChEMBL 7.65
Top Co-occurrence Targets
Active Molecules (343)
InChIKey pChEMBL Type Targets Clinical
UFHHKCDGLUBGJY 6.2 pIC50 2 Yes
VEGZKBKISJJLJC 6.2 IC50 3 Yes
VLYZWOUEQOSDIN 6.2 Ki 2
OZUSVSPHYKYLAS 6.2 pIC50 2 Yes
RSSCBKHOJPGYIW 6.2 Ki 2
CTAHPXXZSACISG 6.2 pIC50 2 Yes
HUOIRVSSWJKCQP 6.2 Ki 2
UUNNSNYSEQPCKO 6.2 IC50 2
ZAYFSWRWHALHQG 6.2 Ki 2
ARRVGGQZILZZEJ 6.2 pIC50 2 Yes
DDUAFEYIPWOELY 6.2 pIC50 2 Yes
BMWKQHPGKPJLPG 6.2 pIC50 2 Yes
BERNHFOYDVXQGI 6.2 pIC50 2 Yes
GFMBISIECXFEJK 6.2 pIC50 2 Yes
NFNSLUVCTGTZGY 6.1 Ki 2
RPNVENCCLVKRAM 6.1 pIC50 2 Yes
PSNAHSRRFJSWQU 6.1 pIC50 2 Yes
QNCFQRIXQDHLMN 6.1 pIC50 2 Yes
IRUDQSQIPJJXFZ 6.1 pIC50 2 Yes
DOABBONQBBUCRN 6.1 pIC50 2 Yes
YGVMCMZWGQEBFU 6.1 pIC50 2 Yes
ACWHYMXOCYJYPG 6.1 pIC50 2 Yes
SPJCSYUKRLKAQT 6.1 pIC50 2 Yes
VMFFXQXFIYFZKK 6.1 IC50 2
DTSANQSRTBGPPK 6.1 pIC50 2 Yes
GKDWRERMBNGKCZ 6.1 IC50 2
DUPJRHKBDSHZPG 6.0 pIC50 2 Yes
QZFBYNPTVXYUII 6.0 IC50 2
KJQHRGYUFQCLJG 6.0 pIC50 2 Yes
ZOZPVKJSFYNWLP 6.0 pIC50 2 Yes
JVXUNHXYBLGVPM 6.0 IC50 2
XLWHWNHGNRPPBH 6.0 Ki 2 Yes
GSIXSVTVZDJDOC 6.0 pIC50 2 Yes
IEAOMUBPJVXBAO 6.0 pIC50 2 Yes
OIVTVLWHNZZBJN 6.0 pIC50 2 Yes
RRZKRPHYMGDLBB 6.0 pIC50 2 Yes
TXSXJYRAIUVBDO 6.0 pIC50 2 Yes
YJMMQRORYCUFDF 6.0 pIC50 2 Yes
ZICGXQSIIFWORG 6.0 pIC50 2 Yes
CHVZZDMXXHMJNM Clinical TTD_MultiTarget 2 Yes
DWHRPZRXNRDAQF Clinical TTD_MultiTarget 2 Yes
IYNMVGGOTRCWGJ Clinical TTD_MultiTarget 2 Yes
LHFDBKUCTFELLO Clinical TTD_MultiTarget 2 Yes
2D structure