Target Details
UniProt ACP32238
Gene SymbolCCKAR
Protein NameCholecystokinin receptor type A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF09193 (CholecysA-Rec_N)
Summary
  • Multi-target molecules 343
  • Clinical molecules 242
  • Avg pChEMBL 7.65
Top Co-occurrence Targets
Active Molecules (343)
InChIKey pChEMBL Type Targets Clinical
CLFXXEFAURLAMH 6.7 pIC50 2 Yes
NUPMWKNZJMFJQO 6.7 pIC50 2 Yes
VKOORZDCJQQHKM 6.7 pIC50 2 Yes
DTSANQSRTBGPPK 6.7 pIC50 2 Yes
NIQAYAGJQYCQNK 6.7 pIC50 2 Yes
RSXHCVGPXZSMBO 6.7 pIC50 2 Yes
AICFYCNTUWZWAG 6.7 Ki 2 Yes
BETHSQILIUBHDZ 6.7 pIC50 2 Yes
HHYKRIBHFNFXEL 6.7 pIC50 2 Yes
IIYXZVJGZRIIKG 6.7 pIC50 2 Yes
VNDOMFNPSJBMRV 6.7 IC50 2
WFRCVVPACDUWGD 6.7 pIC50 2 Yes
GEOWQTGMJLRVOC 6.6 pIC50 2 Yes
MLJPZDPDIBXWNY 6.6 IC50 2
SKGADOFSECCZFC 6.6 pIC50 2 Yes
YCEIOOXEUSAMIZ 6.6 IC50 3 Yes
ODMAYKFSTPTMKE 6.5 Ki 2
HYWPVMQNTSVAPF 6.5 pIC50 2 Yes
ZKCCHRIGDWWTRL 6.5 pIC50 2 Yes
WCLONOKYROXQCI 6.5 pIC50 2 Yes
WKUGDHYDAPFFHF 6.5 IC50 2
AIQFACLFKVFQQI 6.5 Ki 2
LTNSZIYAGMZDDY 6.5 pIC50 2 Yes
HQDSSVWRHVHJGQ 6.5 IC50 2
ZJQCLCIESPIJML 6.4 Ki 2
NNMKTACSCZBLRL 6.4 Ki 2
SEIABTQHADRMGY 6.4 pIC50 2 Yes
VZSPHGCBTKXLMY 6.4 pIC50 2 Yes
YBJYGPHLNAJPTE 6.4 pIC50 2 Yes
NBOSZKXBNZIDBS 6.4 pIC50 2 Yes
CMYMFJIRDMYHDJ 6.4 pIC50 2 Yes
WINOYNIKWSTXQD 6.4 pIC50 2 Yes
OROBBIIDFVAOPI 6.4 pIC50 2 Yes
NQWFBQBJSJTMCW 6.4 pIC50 2 Yes
VJHDZLBKGPSGON 6.4 pIC50 2 Yes
BAWQUHWZYDWDIH 6.4 pIC50 2 Yes
XKDCRXFJHGOCJK 6.4 pIC50 2 Yes
NAYWENBSENWRRT 6.3 pIC50 2 Yes
OROBBIIDFVAOPI 6.3 pIC50 2 Yes
STXYGGMUUHCKOP 6.3 Ki 2
VCBHARIFOKYMTC 6.3 Ki 2
DGKMBNVRIZTNTK 6.3 Ki 2
ZEDOJUJFHGOAOS 6.3 IC50 2
KWYHFHAIKHYSHF 6.3 pIC50 2 Yes
VTMQSICVVWNLPW 6.3 IC50 2
FMPRFCINNRGLNV 6.3 pIC50 2 Yes
NMRHHKUTBQFJAA 6.3 Ki 2
WFEXFFRNIOUBQX 6.3 Ki 2
IHRCGSOFHCURCS 6.2 pIC50 2 Yes
VVKBKPBAKDXLOT 6.2 pIC50 3 Yes
2D structure