Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLFXXEFAURLAMH
|
6.7 | pIC50 | 2 | Yes | |
NUPMWKNZJMFJQO
|
6.7 | pIC50 | 2 | Yes | |
VKOORZDCJQQHKM
|
6.7 | pIC50 | 2 | Yes | |
DTSANQSRTBGPPK
|
6.7 | pIC50 | 2 | Yes | |
NIQAYAGJQYCQNK
|
6.7 | pIC50 | 2 | Yes | |
RSXHCVGPXZSMBO
|
6.7 | pIC50 | 2 | Yes | |
AICFYCNTUWZWAG
|
6.7 | Ki | 2 | Yes | |
BETHSQILIUBHDZ
|
6.7 | pIC50 | 2 | Yes | |
HHYKRIBHFNFXEL
|
6.7 | pIC50 | 2 | Yes | |
IIYXZVJGZRIIKG
|
6.7 | pIC50 | 2 | Yes | |
VNDOMFNPSJBMRV
|
6.7 | IC50 | 2 | — | |
WFRCVVPACDUWGD
|
6.7 | pIC50 | 2 | Yes | |
GEOWQTGMJLRVOC
|
6.6 | pIC50 | 2 | Yes | |
MLJPZDPDIBXWNY
|
6.6 | IC50 | 2 | — | |
SKGADOFSECCZFC
|
6.6 | pIC50 | 2 | Yes | |
YCEIOOXEUSAMIZ
|
6.6 | IC50 | 3 | Yes | |
ODMAYKFSTPTMKE
|
6.5 | Ki | 2 | — | |
HYWPVMQNTSVAPF
|
6.5 | pIC50 | 2 | Yes | |
ZKCCHRIGDWWTRL
|
6.5 | pIC50 | 2 | Yes | |
WCLONOKYROXQCI
|
6.5 | pIC50 | 2 | Yes | |
WKUGDHYDAPFFHF
|
6.5 | IC50 | 2 | — | |
AIQFACLFKVFQQI
|
6.5 | Ki | 2 | — | |
LTNSZIYAGMZDDY
|
6.5 | pIC50 | 2 | Yes | |
HQDSSVWRHVHJGQ
|
6.5 | IC50 | 2 | — | |
ZJQCLCIESPIJML
|
6.4 | Ki | 2 | — | |
NNMKTACSCZBLRL
|
6.4 | Ki | 2 | — | |
SEIABTQHADRMGY
|
6.4 | pIC50 | 2 | Yes | |
VZSPHGCBTKXLMY
|
6.4 | pIC50 | 2 | Yes | |
YBJYGPHLNAJPTE
|
6.4 | pIC50 | 2 | Yes | |
NBOSZKXBNZIDBS
|
6.4 | pIC50 | 2 | Yes | |
CMYMFJIRDMYHDJ
|
6.4 | pIC50 | 2 | Yes | |
WINOYNIKWSTXQD
|
6.4 | pIC50 | 2 | Yes | |
OROBBIIDFVAOPI
|
6.4 | pIC50 | 2 | Yes | |
NQWFBQBJSJTMCW
|
6.4 | pIC50 | 2 | Yes | |
VJHDZLBKGPSGON
|
6.4 | pIC50 | 2 | Yes | |
BAWQUHWZYDWDIH
|
6.4 | pIC50 | 2 | Yes | |
XKDCRXFJHGOCJK
|
6.4 | pIC50 | 2 | Yes | |
NAYWENBSENWRRT
|
6.3 | pIC50 | 2 | Yes | |
OROBBIIDFVAOPI
|
6.3 | pIC50 | 2 | Yes | |
STXYGGMUUHCKOP
|
6.3 | Ki | 2 | — | |
VCBHARIFOKYMTC
|
6.3 | Ki | 2 | — | |
DGKMBNVRIZTNTK
|
6.3 | Ki | 2 | — | |
ZEDOJUJFHGOAOS
|
6.3 | IC50 | 2 | — | |
KWYHFHAIKHYSHF
|
6.3 | pIC50 | 2 | Yes | |
VTMQSICVVWNLPW
|
6.3 | IC50 | 2 | — | |
FMPRFCINNRGLNV
|
6.3 | pIC50 | 2 | Yes | |
NMRHHKUTBQFJAA
|
6.3 | Ki | 2 | — | |
WFEXFFRNIOUBQX
|
6.3 | Ki | 2 | — | |
IHRCGSOFHCURCS
|
6.2 | pIC50 | 2 | Yes | |
VVKBKPBAKDXLOT
|
6.2 | pIC50 | 3 | Yes |