Target Details
UniProt ACP32238
Gene SymbolCCKAR
Protein NameCholecystokinin receptor type A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF09193 (CholecysA-Rec_N)
Summary
  • Multi-target molecules 343
  • Clinical molecules 242
  • Avg pChEMBL 7.65
Top Co-occurrence Targets
Active Molecules (343)
InChIKey pChEMBL Type Targets Clinical
HRFMJPIGMOWHLL 7.3 pIC50 2 Yes
ZMTRGKKPVWRAII 7.3 pIC50 2 Yes
DILLUBXISCIMIT 7.2 IC50 2
HSPTWXGPKMKONJ 7.2 pIC50 2 Yes
ZMTXZNHONYLRJA 7.2 pIC50 2 Yes
POOPTTIQXTUHMQ 7.2 pIC50 2 Yes
FPVZBTVLTPLRDX 7.2 pIC50 2 Yes
KGFIYGFYTIJLRJ 7.2 pIC50 2 Yes
RLKUXRWOAPPZQB 7.1 Ki 2
GAUFCDPHSYEFLM 7.1 IC50 2
GMAIGIQFMVFLBZ 7.1 pIC50 2 Yes
MIUNVYQVNGDVKG 7.1 pIC50 2 Yes
URMOKEJAUAGZGV 7.1 Ki 2
WYYQDZXURPONSW 7.1 Ki 2
DEOUZOCNOYBARB 7.1 pIC50 2 Yes
HBSCTWOGVRBGQM 7.1 pIC50 2 Yes
PKHVPLITWFVWGV 7.1 IC50 2
RGFJPHVCLXSEHE 7.1 pIC50 2 Yes
XQSCLQLQGFXSLK 7.1 pIC50 2 Yes
IHTFQIMRRQEUKB 7.0 IC50 2
SLBLGMBJPJLBTA 7.0 pIC50 2 Yes
OGHIDHUMQVCJLH 7.0 IC50 2
QHXBSJRCFQZXTO 7.0 pIC50 2 Yes
SNYZWGJVKSJMGZ 7.0 pIC50 2 Yes
VNIAHKVXCCCDOZ 7.0 pIC50 2 Yes
FSEWRHPBSMPGFF 7.0 IC50 2
BJABGWNNTUGRHH 6.9 pIC50 2 Yes
ZRTOSCLSAJLFLV 6.9 Ki 2
ATZKJWWUDVCPPQ 6.9 pIC50 2 Yes
BYSPJTKARHNTCE 6.9 pIC50 2 Yes
KSEULEJGJDECHB 6.9 pIC50 2 Yes
CABBMMXFOOZVMS 6.9 IC50 2
BVUCMLHZVCAVLT 6.9 IC50 2
CABBMMXFOOZVMS 6.9 IC50 2
FEOAQCGOOODCEB 6.9 pIC50 2 Yes
KSEULEJGJDECHB 6.9 pIC50 2 Yes
DDMOESJKCONAST 6.9 pIC50 2 Yes
GWSFJWULDCAOKV 6.9 pIC50 2 Yes
LOXHZBJMXMSEOS 6.9 IC50 2
DXRCYRRBLUBBSH 6.8 pIC50 2 Yes
LNIOBOYWQUFRMI 6.8 IC50 2
HSPFWSJPWOITQE 6.8 pIC50 2 Yes
PDWDMFQEOPBNJU 6.8 IC50 2
DZACSGLWVJJFJL 6.8 pIC50 2 Yes
IBEXWSKBKHNHHX 6.8 pIC50 2 Yes
NFHRQQKPEBFUJK 6.8 pIC50 2 Yes
OIXQINQYMGNCII 6.8 pIC50 2 Yes
ZCLCUGHPNSTPGZ 6.8 pIC50 2 Yes
VLKJKVMACAESPP 6.8 Ki 2
CFAMCNLQPGYLTL 6.7 pIC50 2 Yes
2D structure