Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HRFMJPIGMOWHLL
|
7.3 | pIC50 | 2 | Yes | |
ZMTRGKKPVWRAII
|
7.3 | pIC50 | 2 | Yes | |
DILLUBXISCIMIT
|
7.2 | IC50 | 2 | — | |
HSPTWXGPKMKONJ
|
7.2 | pIC50 | 2 | Yes | |
ZMTXZNHONYLRJA
|
7.2 | pIC50 | 2 | Yes | |
POOPTTIQXTUHMQ
|
7.2 | pIC50 | 2 | Yes | |
FPVZBTVLTPLRDX
|
7.2 | pIC50 | 2 | Yes | |
KGFIYGFYTIJLRJ
|
7.2 | pIC50 | 2 | Yes | |
RLKUXRWOAPPZQB
|
7.1 | Ki | 2 | — | |
GAUFCDPHSYEFLM
|
7.1 | IC50 | 2 | — | |
GMAIGIQFMVFLBZ
|
7.1 | pIC50 | 2 | Yes | |
MIUNVYQVNGDVKG
|
7.1 | pIC50 | 2 | Yes | |
URMOKEJAUAGZGV
|
7.1 | Ki | 2 | — | |
WYYQDZXURPONSW
|
7.1 | Ki | 2 | — | |
DEOUZOCNOYBARB
|
7.1 | pIC50 | 2 | Yes | |
HBSCTWOGVRBGQM
|
7.1 | pIC50 | 2 | Yes | |
PKHVPLITWFVWGV
|
7.1 | IC50 | 2 | — | |
RGFJPHVCLXSEHE
|
7.1 | pIC50 | 2 | Yes | |
XQSCLQLQGFXSLK
|
7.1 | pIC50 | 2 | Yes | |
IHTFQIMRRQEUKB
|
7.0 | IC50 | 2 | — | |
SLBLGMBJPJLBTA
|
7.0 | pIC50 | 2 | Yes | |
OGHIDHUMQVCJLH
|
7.0 | IC50 | 2 | — | |
QHXBSJRCFQZXTO
|
7.0 | pIC50 | 2 | Yes | |
SNYZWGJVKSJMGZ
|
7.0 | pIC50 | 2 | Yes | |
VNIAHKVXCCCDOZ
|
7.0 | pIC50 | 2 | Yes | |
FSEWRHPBSMPGFF
|
7.0 | IC50 | 2 | — | |
BJABGWNNTUGRHH
|
6.9 | pIC50 | 2 | Yes | |
ZRTOSCLSAJLFLV
|
6.9 | Ki | 2 | — | |
ATZKJWWUDVCPPQ
|
6.9 | pIC50 | 2 | Yes | |
BYSPJTKARHNTCE
|
6.9 | pIC50 | 2 | Yes | |
KSEULEJGJDECHB
|
6.9 | pIC50 | 2 | Yes | |
CABBMMXFOOZVMS
|
6.9 | IC50 | 2 | — | |
BVUCMLHZVCAVLT
|
6.9 | IC50 | 2 | — | |
CABBMMXFOOZVMS
|
6.9 | IC50 | 2 | — | |
FEOAQCGOOODCEB
|
6.9 | pIC50 | 2 | Yes | |
KSEULEJGJDECHB
|
6.9 | pIC50 | 2 | Yes | |
DDMOESJKCONAST
|
6.9 | pIC50 | 2 | Yes | |
GWSFJWULDCAOKV
|
6.9 | pIC50 | 2 | Yes | |
LOXHZBJMXMSEOS
|
6.9 | IC50 | 2 | — | |
DXRCYRRBLUBBSH
|
6.8 | pIC50 | 2 | Yes | |
LNIOBOYWQUFRMI
|
6.8 | IC50 | 2 | — | |
HSPFWSJPWOITQE
|
6.8 | pIC50 | 2 | Yes | |
PDWDMFQEOPBNJU
|
6.8 | IC50 | 2 | — | |
DZACSGLWVJJFJL
|
6.8 | pIC50 | 2 | Yes | |
IBEXWSKBKHNHHX
|
6.8 | pIC50 | 2 | Yes | |
NFHRQQKPEBFUJK
|
6.8 | pIC50 | 2 | Yes | |
OIXQINQYMGNCII
|
6.8 | pIC50 | 2 | Yes | |
ZCLCUGHPNSTPGZ
|
6.8 | pIC50 | 2 | Yes | |
VLKJKVMACAESPP
|
6.8 | Ki | 2 | — | |
CFAMCNLQPGYLTL
|
6.7 | pIC50 | 2 | Yes |