Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LGYKPDHARJMLQN
|
7.6 | IC50 | 2 | — | |
ALPLVUYDOOIUAE
|
7.6 | pIC50 | 2 | Yes | |
BUDVFFOVUFVRER
|
7.6 | pIC50 | 2 | Yes | |
AKHKIVGBTDKSGG
|
7.6 | pIC50 | 2 | Yes | |
DDROKKYSSQPXQO
|
7.6 | pIC50 | 2 | Yes | |
DWHRPZRXNRDAQF
|
7.6 | pIC50 | 3 | Yes | |
IZIFZVHACKDILP
|
7.6 | pIC50 | 2 | Yes | |
SDJPEEZPMPFEON
|
7.6 | pIC50 | 2 | Yes | |
GQFWYWXTSTVXPK
|
7.5 | pIC50 | 2 | Yes | |
NIQAYAGJQYCQNK
|
7.5 | pIC50 | 2 | Yes | |
PKNBIEKWQLWZNJ
|
7.5 | pIC50 | 2 | Yes | |
VHAAOROZSHMZRJ
|
7.5 | pIC50 | 2 | Yes | |
PRUIQGOHWDZVJD
|
7.5 | IC50 | 2 | — | |
YDZYKNJZCVIKPP
|
7.5 | Ki | 2 | — | |
VNIAHKVXCCCDOZ
|
7.5 | pIC50 | 2 | Yes | |
XNUGDRMOEPOBFR
|
7.5 | pIC50 | 2 | Yes | |
YYUMVSJDMJRIKE
|
7.5 | pIC50 | 2 | Yes | |
CHYXBVRNXVPDAR
|
7.5 | pIC50 | 2 | Yes | |
TVINVHGLLFLSBP
|
7.5 | IC50 | 4 | Yes | |
YRULVPAVSSLIEL
|
7.5 | IC50 | 2 | Yes | |
MPLZTZIWSHXYGD
|
7.5 | pIC50 | 2 | Yes | |
OULXGYXKPKVJPL
|
7.5 | pIC50 | 2 | Yes | |
CHEUONHPKBJUCB
|
7.5 | pIC50 | 2 | Yes | |
PFDXGRUVVNQAQW
|
7.5 | pIC50 | 2 | Yes | |
UXSCCYZDWXCQRW
|
7.5 | pIC50 | 2 | Yes | |
NACOKSRFWNZWTN
|
7.5 | pIC50 | 2 | Yes | |
JVCLXDNXAUQCLR
|
7.4 | IC50 | 2 | — | |
MUNNAUUHDXISAJ
|
7.4 | pIC50 | 2 | Yes | |
RUXGBVNMEPICAJ
|
7.4 | pIC50 | 2 | Yes | |
SXXOCXCOHMDHPD
|
7.4 | IC50 | 2 | — | |
KTIVKLXXTDQNMF
|
7.4 | pIC50 | 2 | Yes | |
DPTKJTLNHCGWTH
|
7.4 | pIC50 | 2 | Yes | |
IRRPCAFDQVDMNP
|
7.4 | IC50 | 2 | — | |
NCXFVQVUXTYYEG
|
7.4 | pIC50 | 2 | Yes | |
JPSKDACFMPXNMN
|
7.4 | IC50 | 2 | — | |
XWNQRVQSRVNMGY
|
7.4 | pIC50 | 2 | Yes | |
INPUMSDGOIKULR
|
7.4 | pIC50 | 2 | Yes | |
GKKCSRUSTYGKFF
|
7.4 | pIC50 | 2 | Yes | |
UBNMGTSDHSQBEL
|
7.4 | IC50 | 2 | — | |
FAQSZDGODZYSIN
|
7.4 | pIC50 | 2 | Yes | |
LJOCWELELLFJSQ
|
7.4 | IC50 | 2 | — | |
VQXCMRAQZMSGPR
|
7.4 | IC50 | 2 | — | |
HEEJTBJFKMOMFO
|
7.3 | Ki | 2 | — | |
HMGDEYJMBGQTPV
|
7.3 | pIC50 | 2 | Yes | |
ITMJPTIFWLPIOL
|
7.3 | IC50 | 2 | Yes | |
USWDPRRJNGKNQG
|
7.3 | pIC50 | 2 | Yes | |
XSHMFCLLINAWBH
|
7.3 | IC50 | 2 | — | |
JZBWOSXHOVOLBT
|
7.3 | pIC50 | 2 | Yes | |
PWEFAKIGTKFZQK
|
7.3 | pIC50 | 2 | Yes | |
ZJGPYSQTJSMQNL
|
7.3 | IC50 | 2 | — |