Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MPQWSQLPSQOSKO
|
8.3 | pIC50 | 2 | Yes | |
KYWMQIRORZGHDH
|
8.2 | IC50 | 2 | — | |
LZZPPPZINPSHEI
|
8.2 | pIC50 | 2 | Yes | |
BZVZYXCWVJJFDH
|
8.2 | pIC50 | 2 | Yes | |
RGJCMCCPAYOLOE
|
8.2 | pIC50 | 2 | Yes | |
PIHWDFKUEPTNFH
|
8.2 | pIC50 | 2 | Yes | |
PIYVAPZSWIDNTQ
|
8.2 | pIC50 | 2 | Yes | |
UWZVTINXEBCDPO
|
8.1 | pIC50 | 2 | Yes | |
ORTWASXZYRMKIJ
|
8.1 | pIC50 | 2 | Yes | |
SJDGAPPCMGPKLY
|
8.1 | pIC50 | 2 | Yes | |
CSNNJXSLJWKSCD
|
8.1 | pIC50 | 2 | Yes | |
LTNSZIYAGMZDDY
|
8.1 | pIC50 | 3 | Yes | |
WLTSODCLBUFUDX
|
8.1 | pIC50 | 2 | Yes | |
AHYNKYYQUAOMCJ
|
8.1 | IC50 | 2 | — | |
MYKVVXCIFKAFIQ
|
8.1 | pIC50 | 2 | Yes | |
SYGCFCSEEIGJCO
|
8.1 | pIC50 | 2 | Yes | |
ZZVLKHHSRQKCEV
|
8.1 | Ki | 4 | Yes | |
FCDAJLCDHWZLKC
|
8.0 | IC50 | 2 | — | |
YVOYRMXNVINXII
|
8.0 | Ki | 3 | Yes | |
ALSNOSFKYCYLJH
|
8.0 | pIC50 | 2 | Yes | |
RAYLDYGVHMTPSI
|
8.0 | pIC50 | 2 | Yes | |
SBMRIYCGYSYWIJ
|
8.0 | pIC50 | 2 | Yes | |
SNVSYPLFUFXAES
|
8.0 | IC50 | 2 | — | |
VDNWZTJUPNHYID
|
8.0 | Ki | 2 | — | |
WGLBHEKCPCUEDT
|
8.0 | pIC50 | 2 | Yes | |
DVASHPOLPKOKGD
|
8.0 | pIC50 | 2 | Yes | |
GDFLLWZJUDPZMX
|
8.0 | IC50 | 2 | — | |
MLJPZDPDIBXWNY
|
7.9 | IC50 | 2 | — | |
UIISAWYHPZCXHX
|
7.9 | pIC50 | 2 | Yes | |
HLUCCSPJVQTJTM
|
7.9 | IC50 | 2 | — | |
DQWCJWUIFIKCRT
|
7.9 | IC50 | 2 | — | |
NCCODGOBVZOLFU
|
7.8 | pIC50 | 2 | Yes | |
RYNRWNJFDSYFLB
|
7.8 | pIC50 | 2 | Yes | |
YXAVZKKJFIOGEL
|
7.8 | IC50 | 2 | — | |
BDKLOKRNGDIZTO
|
7.8 | pIC50 | 2 | Yes | |
KKPFQTRKARZYLE
|
7.8 | pIC50 | 3 | Yes | |
TVINVHGLLFLSBP
|
7.8 | Ki | 4 | — | |
WDLOTEQZLXZCSI
|
7.8 | pIC50 | 2 | Yes | |
HVCMNKCXHIIFDJ
|
7.8 | pIC50 | 2 | Yes | |
IAYFRXOMWAZQGV
|
7.8 | IC50 | 2 | — | |
IHNBBRXFWBWHAP
|
7.8 | IC50 | 2 | — | |
NAYWENBSENWRRT
|
7.8 | pIC50 | 2 | Yes | |
ZKEBGVDIRJCKNA
|
7.8 | IC50 | 2 | — | |
DYFJGOOJNUUTLF
|
7.8 | IC50 | 2 | — | |
NDMKAESGNQHGID
|
7.8 | IC50 | 2 | — | |
AHRZYQWKXXBNHK
|
7.7 | Ki | 4 | Yes | |
RTYGUEPUOWLIME
|
7.7 | pIC50 | 2 | Yes | |
ZUUGDHAKGUQZKD
|
7.7 | pIC50 | 3 | Yes | |
KLTPQGIBPCHXAQ
|
7.7 | IC50 | 2 | — | |
AHKXHAMSXLISEI
|
7.7 | IC50 | 2 | — |