Target Details
UniProt ACP32238
Gene SymbolCCKAR
Protein NameCholecystokinin receptor type A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1) PF09193 (CholecysA-Rec_N)
Summary
  • Multi-target molecules 343
  • Clinical molecules 242
  • Avg pChEMBL 7.65
Top Co-occurrence Targets
Active Molecules (343)
InChIKey pChEMBL Type Targets Clinical
CQUWKHKELQQYRI 9.0 IC50 4
CQUWKHKELQQYRI 9.0 IC50 4
VLKJKVMACAESPP 9.0 pIC50 2 Yes
TVNLSGMCRJXNND 9.0 pIC50 2 Yes
CMYDNIJMVCZZQK 9.0 pIC50 2 Yes
KDFQABSFVYLGPM 9.0 pIC50 2 Yes
KKPFQTRKARZYLE 9.0 pIC50 3 Yes
ROJMLIUODNIIEZ 8.9 IC50 2
KSAGKPZDJHLHBS 8.9 pIC50 4 Yes
IEJRYJFWTCKXSD 8.8 pIC50 2 Yes
ZYFZAOVAALGAJO 8.8 pIC50 2 Yes
LFIFGNCFEBAIHA 8.8 pIC50 4 Yes
UGINDELNLJSTRU 8.8 pIC50 2 Yes
KKPFQTRKARZYLE 8.8 pIC50 4 Yes
LFIFGNCFEBAIHA 8.8 pIC50 3 Yes
NENKRICCIWXRGU 8.8 Ki 4 Yes
OFQAQYAFHZCAOX 8.8 pIC50 2 Yes
OGWBASUUCLOVLN 8.7 pIC50 2 Yes
FVTWFHUCJJXREC 8.7 pIC50 2 Yes
QRYOMNSPKSJSKG 8.7 pIC50 2 Yes
ZANGNFNVUAPKGY 8.7 pIC50 2 Yes
IJHCWGDIGBABKC 8.7 pIC50 3 Yes
LGRKVVHGUJOXEN 8.7 pIC50 4 Yes
CYCOQCORURTMQB 8.7 IC50 2
JHFTVYNYYKDISE 8.7 pIC50 2 Yes
JJAYAAFBSRHMID 8.7 pIC50 2 Yes
CLMCTKVZMVJCQP 8.6 pIC50 2 Yes
QOSWNOTZBYMOLA 8.6 pIC50 2 Yes
BFSMHEBYNOKMKU 8.6 pIC50 2 Yes
GCLKVXOCZDHVEF 8.5 IC50 2
CXNFPROZKYIEPE 8.5 pIC50 2 Yes
DZFMLNMPSVVWNC 8.5 pIC50 2 Yes
JMFXHOKUYGTFJU 8.5 pIC50 2 Yes
KONMZUWCOVKBMG 8.4 IC50 2
VLKJKVMACAESPP 8.4 Ki 2 Yes
VLKJKVMACAESPP 8.4 Ki 2
RKKAWDULAQHRCY 8.4 pIC50 2 Yes
QWOAONQRBDJQTC 8.4 pIC50 2 Yes
BERNHFOYDVXQGI 8.4 pIC50 2 Yes
LJAZTWRBCMHLKX 8.4 pIC50 2 Yes
IBOMYHWWSMSHBV 8.4 pIC50 2 Yes
STEAMACHIRWBBH 8.3 IC50 3
NXHWDEQNHXTHJU 8.3 pIC50 3 Yes
DAZGMBOFHKYQHK 8.3 pIC50 2 Yes
FNRFRMQWGSYIMM 8.3 IC50 2
PFOLRJQYZKGBLP 8.3 pIC50 2 Yes
QAZGXXFYHAMXIB 8.3 pIC50 2 Yes
STEAMACHIRWBBH 8.3 IC50 2
XLWHWNHGNRPPBH 8.3 Ki 2 Yes
KYWMQIRORZGHDH 8.3 IC50 2 Yes
2D structure