Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CQUWKHKELQQYRI
|
9.0 | IC50 | 4 | — | |
CQUWKHKELQQYRI
|
9.0 | IC50 | 4 | — | |
VLKJKVMACAESPP
|
9.0 | pIC50 | 2 | Yes | |
TVNLSGMCRJXNND
|
9.0 | pIC50 | 2 | Yes | |
CMYDNIJMVCZZQK
|
9.0 | pIC50 | 2 | Yes | |
KDFQABSFVYLGPM
|
9.0 | pIC50 | 2 | Yes | |
KKPFQTRKARZYLE
|
9.0 | pIC50 | 3 | Yes | |
ROJMLIUODNIIEZ
|
8.9 | IC50 | 2 | — | |
KSAGKPZDJHLHBS
|
8.9 | pIC50 | 4 | Yes | |
IEJRYJFWTCKXSD
|
8.8 | pIC50 | 2 | Yes | |
ZYFZAOVAALGAJO
|
8.8 | pIC50 | 2 | Yes | |
LFIFGNCFEBAIHA
|
8.8 | pIC50 | 4 | Yes | |
UGINDELNLJSTRU
|
8.8 | pIC50 | 2 | Yes | |
KKPFQTRKARZYLE
|
8.8 | pIC50 | 4 | Yes | |
LFIFGNCFEBAIHA
|
8.8 | pIC50 | 3 | Yes | |
NENKRICCIWXRGU
|
8.8 | Ki | 4 | Yes | |
OFQAQYAFHZCAOX
|
8.8 | pIC50 | 2 | Yes | |
OGWBASUUCLOVLN
|
8.7 | pIC50 | 2 | Yes | |
FVTWFHUCJJXREC
|
8.7 | pIC50 | 2 | Yes | |
QRYOMNSPKSJSKG
|
8.7 | pIC50 | 2 | Yes | |
ZANGNFNVUAPKGY
|
8.7 | pIC50 | 2 | Yes | |
IJHCWGDIGBABKC
|
8.7 | pIC50 | 3 | Yes | |
LGRKVVHGUJOXEN
|
8.7 | pIC50 | 4 | Yes | |
CYCOQCORURTMQB
|
8.7 | IC50 | 2 | — | |
JHFTVYNYYKDISE
|
8.7 | pIC50 | 2 | Yes | |
JJAYAAFBSRHMID
|
8.7 | pIC50 | 2 | Yes | |
CLMCTKVZMVJCQP
|
8.6 | pIC50 | 2 | Yes | |
QOSWNOTZBYMOLA
|
8.6 | pIC50 | 2 | Yes | |
BFSMHEBYNOKMKU
|
8.6 | pIC50 | 2 | Yes | |
GCLKVXOCZDHVEF
|
8.5 | IC50 | 2 | — | |
CXNFPROZKYIEPE
|
8.5 | pIC50 | 2 | Yes | |
DZFMLNMPSVVWNC
|
8.5 | pIC50 | 2 | Yes | |
JMFXHOKUYGTFJU
|
8.5 | pIC50 | 2 | Yes | |
KONMZUWCOVKBMG
|
8.4 | IC50 | 2 | — | |
VLKJKVMACAESPP
|
8.4 | Ki | 2 | Yes | |
VLKJKVMACAESPP
|
8.4 | Ki | 2 | — | |
RKKAWDULAQHRCY
|
8.4 | pIC50 | 2 | Yes | |
QWOAONQRBDJQTC
|
8.4 | pIC50 | 2 | Yes | |
BERNHFOYDVXQGI
|
8.4 | pIC50 | 2 | Yes | |
LJAZTWRBCMHLKX
|
8.4 | pIC50 | 2 | Yes | |
IBOMYHWWSMSHBV
|
8.4 | pIC50 | 2 | Yes | |
STEAMACHIRWBBH
|
8.3 | IC50 | 3 | — | |
NXHWDEQNHXTHJU
|
8.3 | pIC50 | 3 | Yes | |
DAZGMBOFHKYQHK
|
8.3 | pIC50 | 2 | Yes | |
FNRFRMQWGSYIMM
|
8.3 | IC50 | 2 | — | |
PFOLRJQYZKGBLP
|
8.3 | pIC50 | 2 | Yes | |
QAZGXXFYHAMXIB
|
8.3 | pIC50 | 2 | Yes | |
STEAMACHIRWBBH
|
8.3 | IC50 | 2 | — | |
XLWHWNHGNRPPBH
|
8.3 | Ki | 2 | Yes | |
KYWMQIRORZGHDH
|
8.3 | IC50 | 2 | Yes |