Target Details
| UniProt AC | P32238 |
|---|---|
| Gene Symbol | CCKAR |
| Protein Name | Cholecystokinin receptor type A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) PF09193 (CholecysA-Rec_N) |
Summary
- Multi-target molecules 343
- Clinical molecules 242
- Avg pChEMBL 7.65
KEGG Pathways (5)
Active Molecules (343)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IZTQOLKUZKXIRV
|
11.1 | pIC50 | 2 | Yes | |
MAZYNSFCRNJVOU
|
10.5 | IC50 | 2 | — | |
ZFTPEIAEGCLUII
|
10.2 | pIC50 | 2 | Yes | |
LQEROZJFLGEKCE
|
10.2 | IC50 | 2 | — | |
YXNZPENQMVNHAZ
|
10.2 | IC50 | 2 | — | |
QPEUEORJEDJUHX
|
10.1 | IC50 | 2 | — | |
IUSFSIDKWAJIKQ
|
10.1 | IC50 | 2 | — | |
QPEUEORJEDJUHX
|
10.1 | IC50 | 2 | — | |
IFELUJVLOCAXCD
|
10.1 | IC50 | 2 | — | |
WNWLMMMHXDFXKP
|
10.1 | IC50 | 2 | — | |
VKDAZGQQWPSRFA
|
10.0 | pIC50 | 2 | Yes | |
YJRSAZMDFOJHLB
|
10.0 | pIC50 | 2 | Yes | |
BMZYXLWLLWZVBA
|
9.9 | IC50 | 2 | — | |
KYIGOCCCBXRHNJ
|
9.9 | IC50 | 43 | — | |
ADFBVAUNEXEYJP
|
9.8 | pIC50 | 2 | Yes | |
CSXIDZJPJYRGSK
|
9.8 | pIC50 | 2 | Yes | |
NFHRQQKPEBFUJK
|
9.7 | IC50 | 2 | Yes | |
DNKPXDLQYBBMPC
|
9.7 | pIC50 | 2 | Yes | |
SLFCKQWVMXDHDU
|
9.7 | IC50 | 2 | — | |
CSXIDZJPJYRGSK
|
9.6 | pIC50 | 2 | Yes | |
CNWXJSZWVGJITL
|
9.6 | pIC50 | 2 | Yes | |
GHEUKVOXUQUGLZ
|
9.6 | IC50 | 2 | — | |
UDFKASJOSSYSOL
|
9.6 | IC50 | 2 | — | |
SFJVTILNSUYYFI
|
9.6 | pIC50 | 2 | Yes | |
BFIXTZFVFDMGQQ
|
9.6 | IC50 | 2 | — | |
LXWCNCKGNPJZAA
|
9.6 | IC50 | 2 | — | |
QUSCQANKQSFCGJ
|
9.6 | pIC50 | 2 | Yes | |
PBVOPXCIKKBKIX
|
9.5 | pIC50 | 2 | Yes | |
ZANFFYJCTUAWAK
|
9.5 | pIC50 | 2 | Yes | |
XYEJNVLBRMQKPD
|
9.5 | IC50 | 2 | — | |
QPRHQFFOOJJWON
|
9.3 | pIC50 | 2 | Yes | |
NACOKSRFWNZWTN
|
9.3 | pIC50 | 2 | Yes | |
DLRAUJSCRJKHJV
|
9.3 | pIC50 | 2 | Yes | |
WLTSODCLBUFUDX
|
9.3 | pIC50 | 2 | Yes | |
GUXRAKLYIXOIFQ
|
9.2 | pIC50 | 2 | Yes | |
KJQHRGYUFQCLJG
|
9.2 | pIC50 | 4 | Yes | |
LWZREZWAQQSATC
|
9.2 | pIC50 | 2 | Yes | |
OGBLGSTXVFINII
|
9.2 | pIC50 | 2 | Yes | |
WSTOKXRJTCQBGW
|
9.2 | pIC50 | 2 | Yes | |
NLKGFOOGBGCDAL
|
9.2 | pIC50 | 2 | Yes | |
IJHCWGDIGBABKC
|
9.1 | pIC50 | 3 | Yes | |
JMDKMESJXNSGPX
|
9.1 | IC50 | 4 | Yes | |
YJPQVTKXGCBSPW
|
9.1 | pIC50 | 2 | Yes | |
ZINWBFHVGIYPGZ
|
9.1 | IC50 | 2 | — | |
MQIOWUHVKXZQPM
|
9.1 | pIC50 | 2 | Yes | |
IRCIITOKKBCNGO
|
9.1 | pIC50 | 2 | Yes | |
NWLBBDKAIZNTHK
|
9.1 | pIC50 | 2 | Yes | |
OCVIYTKLKRGXCI
|
9.0 | IC50 | 2 | — | |
AGBJVABYWAWOKN
|
9.0 | pIC50 | 2 | Yes | |
ARYXAMNDWNZMBO
|
9.0 | pIC50 | 2 | Yes |