Target Details
UniProt ACP31645
Gene SymbolSLC6A4
Protein NameSodium-dependent serotonin transporter
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF03491 (5HT_transport_N) PF00209 (SNF)
Summary
  • Multi-target molecules 3,668
  • Clinical molecules 120
  • Avg pChEMBL 7.53
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (3,668)
InChIKey pChEMBL Type Targets Clinical
YVKDUIAAPBKHMJ 11.0 Ki 3
YVKDUIAAPBKHMJ 11.0 Ki 3
KPKLDBBNSFWOFA 10.9 Ki 3
VGVAYDIHTPWEKS 10.5 Ki 3
GZWPHROGQGOESZ 10.4 Ki 3
PETAHELMBJGYJY 10.4 Ki 3
GZWPHROGQGOESZ 10.3 Ki 3
ZGPGDMLZVXIWAH 10.3 Ki 2
ZRZJDCNJTXKTEF 10.2 Ki 2
AEYFRZGFXCIRPL 10.1 Ki 3
QRRDJSMVPRYYBA 10.1 Ki 3
RXBAZUHMGOEBGO 10.1 Ki 3
RXBAZUHMGOEBGO 10.1 Ki 3
VNJFIBFHISUZRV 10.1 Ki 4
GAMXLCNZCZEZGS 10.1 Ki 3
WDZSPNFWRVITEJ 10.0 Ki 2
KMNJYBBPXRFSBY 10.0 Ki 3
XFIVQANHMYEPDG 10.0 Ki 2
AYGLZYIWAZBQDC 10.0 IC50 7
ABXUYGWOEIXKBD 10.0 Ki 3
UMYMNRFUWNCPOG 9.9 Ki 2
JNLXUEPMJIMNHM 9.9 Ki 3
RXJIAQGHWRMBEZ 9.9 IC50 2
IBZJKEOJOGAMGJ 9.8 Ki 11 Yes
ZSANFFXRVWPAJC 9.8 Ki 4
GGDBEAVVGFNWIA 9.8 Ki 6
YDNOASAJYGOBQG 9.7 Ki 3
AHEMMEONOCHONP 9.7 Ki 3
AHOUBRCZNHFOSL 9.7 Ki 13
HRCVSENKVJEEJB 9.7 Ki 3
HRJQWACHSNEZEE 9.7 Ki 3
JTZODQOWHKXAGE 9.7 Ki 3
PJIMUTYPWDGKIC 9.7 Ki 3
PYIBCEOJEPANCH 9.7 Ki 3
SVFXPTLYMIXFRX 9.7 Ki 3
CLVQITJMWWKDJN 9.7 Ki 2
CMJSIPQFDNXSOL 9.7 IC50 4
SNNRWIBSGBMYRF 9.7 Ki 3
SNNRWIBSGBMYRF 9.6 Ki 2
FCVAOOZCNCHWJQ 9.6 Ki 3
WEGCLSBGECOYJJ 9.6 Ki 2
FXPKVPDERQMXMV 9.6 Ki 3
GRCVTMNCDBAKJY 9.6 Ki 3
GXWUVPPXUBCALT 9.6 Ki 3
JQQXRQMPNKINQO 9.6 Ki 3
NRTIMMZNHIFNOB 9.6 Ki 3
PWAQSKSFOYUNMV 9.6 Ki 3
SDAMYSWGWHXMRT 9.6 Ki 9
YKDPKVFUKKJFFE 9.6 Ki 3
CDWCEOHVRGUKCE 9.6 Ki 2
2D structure