Target Details
UniProt ACP31644
Gene SymbolGABRA5
Protein NameGamma-aminobutyric acid receptor subunit alpha-5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,276
  • Clinical molecules 0
  • Avg pChEMBL 7.87
Top Co-occurrence Targets
Active Molecules (1,276)
InChIKey pChEMBL Type Targets Clinical
PBUYINIRVVLBIH 9.0 Ki 4
AQKFCEWRKDXGMK 9.0 Ki 16
BQWZDXNKDYRCJK 9.0 Ki 3
IPHSQMSRIWZULE 9.0 Ki 16
IREBWVNSEHBJRT 9.0 Ki 6
KDMMIKQMHNBKAV 9.0 Ki 17
MFZNONRIQYSLMZ 9.0 Ki 6
NHJRHDMRNNOSLV 9.0 Ki 5
NLHGXPUKOAOTRO 9.0 Ki 4
NUXNKKUXSDGYTN 9.0 Ki 7
OXUTXRZFYPFZEZ 9.0 Ki 6
QRZNWQBPKJMWHT 9.0 Kd 2
RKWZHLJYVXAQQP 9.0 Ki 3
RTRIMAMBTITPNP 9.0 Ki 6
STHRYAZDXIDVJO 9.0 Ki 6
VQQCPWHLJXFLOG 9.0 Ki 3
WGRVAGIQTHEEQW 9.0 IC50 16
XKDRJZMAMYYSIZ 9.0 Ki 2
BSBLYLUAUVTSMM 9.0 IC50 16
CIGLLASOKXAMLS 9.0 Ki 7
HZDFUJFVZWUGMH 9.0 Ki 3
IVVHFTRDYKTGCC 9.0 Ki 6
LJRIFLWERUHAIZ 9.0 Ki 8
PCZLQMGFNUNVOM 9.0 Ki 6
RBJYKFLLCXRSGC 9.0 Ki 2
UVTIJQDSGQQUDX 8.9 Ki 5
AETXHLUBKZXEAA 8.9 Ki 3
CAIDJZOHDFNJOZ 8.9 Ki 4
HRJQUDZTLASEPW 8.9 Ki 6
NDFKYGUTDGWIHX 8.9 Ki 6
NEVSBYUBNOGFQJ 8.9 Ki 3
PYEJACCXPZGJAH 8.9 Ki 2
QWNIEEVMYAZTBJ 8.9 Ki 3
UMQUUXLLUHJNGK 8.9 Ki 3
WLHRDALLBOSVLX 8.9 Ki 6
WWDXVOFHKJTAKM 8.9 Ki 6
XXVQXGKSBMSCHX 8.9 Ki 6
ILFZZMYJRPZIPF 8.9 Ki 5
OIKCREAGTIJWOO 8.9 Ki 6
PURSHIRLIYVFDB 8.9 Ki 4
QSEBFHRZNPGODU 8.9 Ki 6
PISANIRNHZBQRM 8.9 Ki 4
AGSFVTKORUUQJP 8.9 Ki 7
QCQSTOYKSWTFNN 8.9 Ki 6
GLOOEDBOHDKUMM 8.9 Ki 4
AYVAVBFBOCMUHW 8.8 Ki 6
BYMDBFGHCDTBMT 8.8 IC50 16
IHAAIBPWHHEARW 8.8 Ki 3
LLJUUCOIBTZXIJ 8.8 Ki 6
MMZOMTNDPGKUIA 8.8 Ki 4
2D structure