Target Details
UniProt ACP31644
Gene SymbolGABRA5
Protein NameGamma-aminobutyric acid receptor subunit alpha-5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,276
  • Clinical molecules 0
  • Avg pChEMBL 7.87
Top Co-occurrence Targets
Active Molecules (1,276)
InChIKey pChEMBL Type Targets Clinical
HJNOESUOZGNLKO 9.2 Ki 6
NLEQOPYBIKKOPK 9.2 Ki 7
OVFRNPXWYQUNHR 9.2 Ki 4
VJMXGRAYTDRKAO 9.2 Ki 6
NZMJFRXKGUCYNP 9.2 Ki 6
BELGLGAAMPTDSH 9.2 Ki 2
CGMJQQJSWIRRRL 9.2 Ki 6
NTEUDQFHQWGEBH 9.2 Ki 5
SSJXJXJUHUAOQL 9.2 Ki 6
CMRJVDJLBFKXKL 9.2 Ki 4
NFMFVESVKLVYJR 9.2 Ki 7
DZPQKPSHACGLKC 9.1 Ki 6
QBYZDDIMNITMSB 9.1 Ki 6
SJAGJFDQMIAULO 9.1 Ki 6
HRVCUISAJOBFTQ 9.1 Ki 6
MMWKMKRWCPKFRA 9.1 Ki 6
SBDBQMZCLBOJPE 9.1 Ki 6
BJYKRVMKNGJKKZ 9.1 Ki 6
CJBGLZXUYDUSDI 9.1 Ki 2
CNEHRQMKOUFFMX 9.1 Ki 3
DQKNTSFPZMVKNA 9.1 Ki 3
GXPHYMCBGKIIKN 9.1 Ki 3
IRYAGFJMRZLHGE 9.1 Ki 6
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
VZKRZUPJCVFVGR 9.1 IC50 16
YTGZSWOWFGVAFH 9.1 Ki 7
BPKZCNBWMWKTIB 9.1 Ki 4
FLTOAJWVMNMXMX 9.1 Ki 6
NURMFSYNABAOFU 9.1 Ki 6
XIDCXRFZRFADDU 9.1 Ki 4
DGBIGWXXNGSACT 9.1 Ki 16
PKSKIVNMTHKBOS 9.1 Ki 2
QORLMYYHZLDYOR 9.1 Ki 9
CHMFFBQMSYJXTP 9.1 Ki 6
IPEQYLWHCRAOTC 9.1 Ki 6
JNJUWXAKLRKXII 9.1 Ki 6
PZIQTZQOFYKORR 9.1 Ki 6
GCTGWUUTZLTQAR 9.1 Ki 6
VCAOZNYTIATHLZ 9.1 Ki 2
WLZXRXFLGSQYFP 9.1 Ki 4
YJZGQBGGTBIAOP 9.1 IC50 16
ZAKVPALBELHKFH 9.1 Ki 6
AAXTWJHZRVXBFG 9.0 Ki 4
CDRADZRGYBTOKU 9.0 Ki 6
OBPPXGLDCMXNDT 9.0 Ki 6
GXKGSEUULCEOTM 9.0 Ki 5
ZDLKXIOQJJRYCW 9.0 Ki 6
GWERFVJRQFKXQG 9.0 Ki 5
2D structure