Target Details
UniProt ACP31644
Gene SymbolGABRA5
Protein NameGamma-aminobutyric acid receptor subunit alpha-5
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,276
  • Clinical molecules 0
  • Avg pChEMBL 7.87
Top Co-occurrence Targets
Active Molecules (1,276)
InChIKey pChEMBL Type Targets Clinical
KPKJEFIYLPVANT 9.4 Ki 4
KVQKVRWATUWLAO 9.4 Ki 5
BUTCFAZTKZDYCN 9.4 Ki 6
HGJUDXDUSGEVOX 9.4 Ki 6
HNGRWUCKESPKRC 9.4 Ki 6
PWTUVRWHZWTHMS 9.4 Ki 2
QUUNMICPMYIHFS 9.4 IC50 16
TXIWNLQFRATZFL 9.4 Ki 4
VMDUABMKBUKKPG 9.4 IC50 16
YTUMMZANIYQNOM 9.4 Ki 8
IHDXFSAXAJRBOG 9.4 Ki 5
AHTXTFPELOVMKB 9.4 Ki 6
SNVZCVVNVLIROS 9.3 Ki 6
YKYOQIXTECBVBB 9.3 Ki 7
XKENJWNGLCKOBP 9.3 IC50 16
YKKWBLSUYZOORV 9.3 Ki 6
IXGIOXIKQZCZIK 9.3 Ki 8
KIDPGPYNXRNUGP 9.3 Ki 3
NJUMMJUUDUYSKB 9.3 IC50 16
WDTNKNNGHGOKBH 9.3 Ki 9
AJWPZYMLAILYCO 9.3 Ki 5
ANARVVNNNQSSPE 9.3 Ki 3
AOZALWRGTMILIK 9.3 Ki 6
BPTASZCHRIMWEF 9.3 Ki 6
FPRLTMYWIBRCQM 9.3 Ki 3
HJIQKECDKLWXGE 9.3 Kd 2
HOQUSTXYXSUJDG 9.3 Ki 6
LLHQBHOWDZNCNK 9.3 Ki 5
LWUDDYHYYNNIQI 9.3 Ki 7
MZGKIGRVCYKVPS 9.3 Ki 6
QGOAGGOYLMIFPI 9.3 Ki 6
UIKTZQCQKHUZHT 9.3 Ki 3
UJBOQYCZTOTBAN 9.3 Ki 4
XXRKXVKJMSIZSM 9.3 Ki 6
GFQMHVYMEKXHDT 9.3 Ki 6
RJOMRLSAWXNFSU 9.3 Ki 4
KSYVJHGNJMYDIQ 9.3 Ki 6
YZRXMMCBUVDBFF 9.3 Ki 6
DXPCEAZKJSYFJM 9.3 Ki 6
FHXDHVUQGGBLGD 9.3 Ki 4
BLJPKQXXDFIIFR 9.2 IC50 16
GIUPLTIPPKYWPM 9.2 Ki 3
GRHSJPRDKRVXDK 9.2 Ki 6
GTOBFJHFOZIFFU 9.2 Ki 5
KCEIOBKDDQAYCM 9.2 Ki 5
LULPFCFGFHHBEZ 9.2 Ki 3
OABMKUYJAYGQHV 9.2 Ki 3
OFBIFZUFASYYRE 9.2 Ki 16
SPUDBCPXWITYDE 9.2 Ki 3
XHCCKQJTDGEMHT 9.2 Ki 3
2D structure